Insulin icodec: A novel once-weekly treatment for diabetes.

diabetes diabetes mellitus diabetes mellitus, type 1 diabetes mellitus, type 2 insulin insulin, long‐acting

Journal

Diabetic medicine : a journal of the British Diabetic Association
ISSN: 1464-5491
Titre abrégé: Diabet Med
Pays: England
ID NLM: 8500858

Informations de publication

Date de publication:
24 Jul 2024
Historique:
revised: 21 06 2024
received: 12 06 2023
accepted: 09 07 2024
medline: 24 7 2024
pubmed: 24 7 2024
entrez: 24 7 2024
Statut: aheadofprint

Résumé

To summarize the results of clinical studies of insulin icodec, an investigational insulin analog designed for once-weekly administration, in adults with type 1 and type 2 diabetes. Thirteen published articles describing clinical studies of insulin icodec were identified in PubMed, and data pertinent to key study outcomes were selected for inclusion in this review. In insulin-naïve and insulin-treated individuals, icodec demonstrated efficacy in glycaemic control superior or noninferior to that of insulins glargine U100, glargine U300 and degludec. Icodec exhibited a safety profile comparable to marketed insulins, with the exception of hypoglycaemic event rates. As a once-weekly alternative to daily basal insulin, icodec is expected to improve patient adherence and satisfaction, reducing the required number of injections per year from 365 to 52 and providing a dosing option potentially attractive to a wide range of insulin users. However, clinical data suggest a notable risk of hypoglycaemia with weekly icodec administration, especially in individuals with type 1 diabetes.

Identifiants

pubmed: 39046097
doi: 10.1111/dme.15414
doi:

Types de publication

Journal Article Review

Langues

eng

Sous-ensembles de citation

IM

Pagination

e15414

Subventions

Organisme : No funding was received.

Informations de copyright

© 2024 Diabetes UK.

Références

Kjeldsen TB, Hubálek F, Hjørringgaard CU, et al. Molecular engineering of insulin ICODEC, the first acylated insulin analog for once‐weekly administration in humans. J Med Chem. 2021;64(13):8942‐8950.
Nishimura E, Pridal L, Glendorf T, et al. Molecular and pharmacological characterization of insulin icodec: a new basal insulin analog designed for once‐weekly dosing. BMJ Open Diabetes Res Care. 2021;9(1):1‐10.
Pieber T, Asong M, Fluhr G, et al. Pharmacokinetic and pharmacodynamic properties of once‐weekly insulin icodec in individuals with type 2 diabetes. Diabetes Obes Metab. 2023;25:3716‐3723.
Hövelmann U, Engberg S, Heise T, et al. Pharmacokinetic and pharmacodynamic properties of once‐weekly insulin icodec in individuals with type 1 diabetes. Diabetes Obes Metab. 2024;26:1941‐1949.
Rosenstock J, Bajaj HS, Janež A, et al. One‐weekly insulin for type 2 diabetes without previous insulin treatment. N Engl J Med. 2020;383(22):2107‐2116.
Lingvay I, Buse JB, Franek E, et al. A randomized, open‐label comparison of once‐weekly insulin Icodec titration strategies versus once‐daily insulin glargine U100. Diabetes Care. 2021;44(7):1595‐1603.
Bajaj HS, Bergenstal RM, Christoffersen A, et al. Switching to once‐weekly insulin Icodec versus once‐daily insulin glargine U100 in type 2 diabetes inadequately controlled on daily basal insulin: a phase 2 randomized controlled trial. Diabetes Care. 2021;44(7):1586‐1594.
Rosenstock J, Bain S, Gowda A, et al. Weekly Icodec versus daily glargine U100 in type 2 diabetes without previous insulin. N Engl J Med. 2023;389(4):297‐308.
Philis‐Tsimikas A, Asong M, Franek E, et al. Switching to once‐weekly insulin icodec versus once‐daily insulin degludec in individuals with basal insulin‐treated type 2 diabetes (ONWARDS 2): a phase 3a, randomised, open label, multicentre, treat‐to‐target trial. Lancet Diabetes Endocrinol. 2023;11(5):1‐12.
Lingvay I, Asong M, Desouza C, et al. Once‐weekly insulin Icodec vs once‐daily insulin Degludec in adults with insulin‐naive type 2 diabetes: the ONWARDS 3 randomized clinical trial. JAMA. 2023;330(3):228‐237.
Mathieu C, Ásbjörnsdóttir B, Bajaj HS, et al. Switching to once‐weekly insulin icodec versus once‐daily insulin glargine U100 in individuals with basal‐bolus insulin‐ treated type 2 diabetes (ONWARDS 4): a phase 3a, randomised, open‐label, multicentre, treat‐to‐target, non‐inferiority trial. Lancet. 2023;401(10389):1‐12.
Bajaj HS, Aberle J, Davies M, et al. Once‐weekly insulin Icodec with dosing guide app versus once‐daily basal insulin analogues in insulin‐naive type 2 diabetes (ONWARDS 5). Ann Intern Med. 2023;176:1476‐1485.
Russell‐Jones D, Babazono T, Callieteau R, et al. Once‐weekly insulin icodec versus once‐daily insulin degludec as part of a basal‐bolus regimen in individuals with type 1 diabetes (ONWARDS 6): a phase 3a, randomised, open‐label, treat‐to‐target trial. Lancet. 2023;402(10413):1636‐1647.
Saisho Y. Use of diabetes treatment satisfaction questionnaire in diabetes care: importance of patient‐reported outcomes. J Environ Res Public Health. 2018;15(5):947.
Brod M, Christensen T, Hammer M, Busk AK, Bushnell DM. Examining the ability to detect change using the trim‐diabetes and trim‐diabetes device measures. Qual Life Res. 2011;20(9):1513‐1518.
Bajaj HS, Ásbjörnsdóttir B, Carstensen L, et al. Continuous glucose monitoring–based metrics and hypoglycemia duration in insulin‐experienced individuals with long‐standing type 2 diabetes switched from a daily basal insulin to once‐weekly insulin Icodec: post hoc analysis of ONWARDS 2 and ONWARDS 4. Diabetes Care. 2024;47(4):729‐738.
European Medicines Agency. Awiqli: EPAR—Medicine Overview. 2022. Accessed June 18, 2024. https://www.ema.europa.eu/en/medicines/human/EPAR/awiqli#overview
Swissmedic. Awiqli® FlexTouch®, Injection Solution in Prefilled Pen (Insulin icodecum). Accessed Jun 10 2024. https://www.swissmedic.ch/swissmedic/en/home/humanarzneimittel/authorisations/new‐medicines/awiqli‐flextouch‐injlsg‐fertigpen‐insulinum‐icodecum.html
Canadian Agency for Drugs and Technologies in Health. Insulin Icodec. Accessed June 10, 2024. https://www.cadth.ca/insulin‐icodec
United States Food and Drug Administration. Endocrinologic and Metabolic Drugs Advisory Committee (EMDAC) Meeting. 2024. Accessed Jun 10, 2024. https://www.youtube.com/watch?v=jeJQNP1Ug2I

Auteurs

Hannah Schaffner (H)

East Coast Institute for Research, Jacksonville, Florida, USA.

Jordyn Wiener (J)

College of Pharmacy Department of Pharmacy Education and Practice, University of Florida, Jacksonville, Florida, USA.

Amanda DeLuca (A)

College of Pharmacy Department of Pharmacy Education and Practice, University of Florida, Jacksonville, Florida, USA.

Ariana Genovese (A)

College of Medicine Department of Medical Education, University of South Florida, Tampa, Florida, USA.

Alexander Deeb (A)

College of Health Professions and Sciences Department of Health Sciences, University of Central Florida, Orlando, Florida, USA.

Wasim Deeb (W)

First Choice Endocrinology, Jacksonville, Florida, USA.

Mae Sheikh-Ali (M)

Northeast Florida Endocrine & Diabetes Associates, Jacksonville, Florida, USA.

David Sutton (D)

Northeast Florida Endocrine & Diabetes Associates, Jacksonville, Florida, USA.

Ashwini Gore (A)

The Jones Center, Macon, Georgia, USA.

Jason Berner (J)

Georgia Mountain Endocrinology, Canton, Georgia, USA.

Jessica Huston (J)

College of Pharmacy Department of Pharmacy Education and Practice, University of Florida, Jacksonville, Florida, USA.

Rebecca Goldfaden (R)

East Coast Institute for Research, Jacksonville, Florida, USA.

Classifications MeSH