A First-in-Class Pyrazole-isoxazole Enhanced Antifungal Activity of Voriconazole: Synergy Studies in an Azole-Resistant


Journal

Journal of medicinal chemistry
ISSN: 1520-4804
Titre abrégé: J Med Chem
Pays: United States
ID NLM: 9716531

Informations de publication

Date de publication:
08 Aug 2024
Historique:
medline: 8 8 2024
pubmed: 8 8 2024
entrez: 8 8 2024
Statut: aheadofprint

Résumé

The widespread and irrational use of azole antifungal agents has led to an increase of azole-resistant

Identifiants

pubmed: 39115219
doi: 10.1021/acs.jmedchem.4c01109
doi:

Types de publication

Journal Article

Langues

eng

Sous-ensembles de citation

IM

Auteurs

Sveva Pelliccia (S)

Department of Pharmacy (DoE 2023-2027), University of Naples Federico II, via D. Montesano 49, 80131 Naples, Italy.

Pasquale Russomanno (P)

Magnetic Resonance Centre (CERM), Consorzio Interuniversitario Risonanze Magnetiche di Metallo Proteine (CIRMMP) and Department of Chemistry "Ugo Schiff", University of Florence, Via L. Sacconi 6, Sesto Fiorentino 50019, Italy.

Simona Barone (S)

Department of Pharmacy (DoE 2023-2027), University of Naples Federico II, via D. Montesano 49, 80131 Naples, Italy.

Baptiste Mateu (B)

Department of Pharmacy (DoE 2023-2027), University of Naples Federico II, via D. Montesano 49, 80131 Naples, Italy.

Antonella Ilenia Alfano (AI)

Department of Pharmacy (DoE 2023-2027), University of Naples Federico II, via D. Montesano 49, 80131 Naples, Italy.

Martina Miranda (M)

Department of Pharmaceutical and Cell Biological Chemistry, Pharmaceutical Institute, University of Bonn, An der Immenburg 4, 53121 Bonn, Germany.

Lorena Coretti (L)

Department of Pharmacy (DoE 2023-2027), University of Naples Federico II, via D. Montesano 49, 80131 Naples, Italy.

Francesca Lembo (F)

Department of Pharmacy (DoE 2023-2027), University of Naples Federico II, via D. Montesano 49, 80131 Naples, Italy.

Marialuisa Piccolo (M)

BioChemLab, Department of Pharmacy, School of Medicine and Surgery, University of Naples Federico II, via D. Montesano 49, 80131 Naples, Italy.

Carlo Irace (C)

BioChemLab, Department of Pharmacy, School of Medicine and Surgery, University of Naples Federico II, via D. Montesano 49, 80131 Naples, Italy.

Laura Friggeri (L)

Department of Cell and Development Biology, U4225 Medical Research Building III, 465 21st Avenue South Room 4160 MRB III Nashville, Tennessee 37232, United States.

Tatiana Y Hargrove (TY)

Department of Biochemistry, Vanderbilt University School of Medicine, Nashville, Tennessee 37232, United States.

Aaron Curtis (A)

Department of Biology, Maynooth University, W23 F2H6 Maynooth, Co. Kildare, Ireland.

Galina I Lepesheva (GI)

Department of Biochemistry, Vanderbilt University School of Medicine, Nashville, Tennessee 37232, United States.

Kevin Kavanagh (K)

Department of Biology, Maynooth University, W23 F2H6 Maynooth, Co. Kildare, Ireland.

Elisabetta Buommino (E)

Department of Pharmacy (DoE 2023-2027), University of Naples Federico II, via D. Montesano 49, 80131 Naples, Italy.

Margherita Brindisi (M)

Department of Pharmacy (DoE 2023-2027), University of Naples Federico II, via D. Montesano 49, 80131 Naples, Italy.

Classifications MeSH