Pembrolizumab for the First-Line Treatment of Recurrent Locally Advanced or Metastatic Merkel Cell Carcinoma: Results from the Single-Arm, Open-Label, Phase III KEYNOTE-913 Study.


Journal

American journal of clinical dermatology
ISSN: 1179-1888
Titre abrégé: Am J Clin Dermatol
Pays: New Zealand
ID NLM: 100895290

Informations de publication

Date de publication:
08 Oct 2024
Historique:
accepted: 19 08 2024
medline: 8 10 2024
pubmed: 8 10 2024
entrez: 8 10 2024
Statut: aheadofprint

Résumé

The phase III KEYNOTE-913 study was conducted to evaluate the efficacy and safety of pembrolizumab as first-line therapy in patients with advanced Merkel cell carcinoma (MCC). The aim was to report results from the primary analysis of KEYNOTE-913. Patients with recurrent locally advanced or metastatic MCC received pembrolizumab 200 mg intravenously every 3 weeks for up to 35 treatments (~ 2 years). The primary end point was objective response rate (ORR) per Response Evaluation Criteria in Solid Tumors, version 1.1 (RECIST v1.1) by blinded independent central review (BICR). Secondary end points were duration of response (DOR) and progression-free survival (PFS) per RECIST v1.1 by BICR, overall survival (OS), and safety and tolerability. Fifty-five patients were treated with pembrolizumab. The median time from first dose to data cutoff (February 15, 2024) was 50.3 months (range 38.7-59.4). The ORR was 49% (95% confidence interval [CI] 35-63), with 12 complete responses and 15 partial responses. The median DOR was 39.8 months (range 4.8-52.5+), and the 24-month DOR rate was 69%. The median PFS was 9.3 months (95% CI 3-26), and the 24-month PFS rate was 39%. The median OS was 24.3 months (95% CI 12.4 to not reached), and the 24-month OS rate was 51%. Any-grade treatment-related adverse events (AEs) occurred in 38 patients (69%); 13 patients (24%) experienced grade 3-5 AEs. The most common treatment-related AEs were fatigue (n = 12 [22%]), pruritus (n = 12 [22%]), and lipase increase (n = 10 [18%]). One patient died of treatment-related Guillain-Barré syndrome. Pembrolizumab provided durable antitumor activity and promising survival and had a manageable safety profile in patients with recurrent locally advanced or metastatic MCC, supporting its use in this population. Clinicaltrials.gov, NCT03783078.

Sections du résumé

BACKGROUND BACKGROUND
The phase III KEYNOTE-913 study was conducted to evaluate the efficacy and safety of pembrolizumab as first-line therapy in patients with advanced Merkel cell carcinoma (MCC).
OBJECTIVE OBJECTIVE
The aim was to report results from the primary analysis of KEYNOTE-913.
PATIENTS AND METHODS METHODS
Patients with recurrent locally advanced or metastatic MCC received pembrolizumab 200 mg intravenously every 3 weeks for up to 35 treatments (~ 2 years). The primary end point was objective response rate (ORR) per Response Evaluation Criteria in Solid Tumors, version 1.1 (RECIST v1.1) by blinded independent central review (BICR). Secondary end points were duration of response (DOR) and progression-free survival (PFS) per RECIST v1.1 by BICR, overall survival (OS), and safety and tolerability.
RESULTS RESULTS
Fifty-five patients were treated with pembrolizumab. The median time from first dose to data cutoff (February 15, 2024) was 50.3 months (range 38.7-59.4). The ORR was 49% (95% confidence interval [CI] 35-63), with 12 complete responses and 15 partial responses. The median DOR was 39.8 months (range 4.8-52.5+), and the 24-month DOR rate was 69%. The median PFS was 9.3 months (95% CI 3-26), and the 24-month PFS rate was 39%. The median OS was 24.3 months (95% CI 12.4 to not reached), and the 24-month OS rate was 51%. Any-grade treatment-related adverse events (AEs) occurred in 38 patients (69%); 13 patients (24%) experienced grade 3-5 AEs. The most common treatment-related AEs were fatigue (n = 12 [22%]), pruritus (n = 12 [22%]), and lipase increase (n = 10 [18%]). One patient died of treatment-related Guillain-Barré syndrome.
CONCLUSIONS CONCLUSIONS
Pembrolizumab provided durable antitumor activity and promising survival and had a manageable safety profile in patients with recurrent locally advanced or metastatic MCC, supporting its use in this population.
TRIAL REGISTRATION BACKGROUND
Clinicaltrials.gov, NCT03783078.

Identifiants

pubmed: 39377880
doi: 10.1007/s40257-024-00885-w
pii: 10.1007/s40257-024-00885-w
doi:

Banques de données

ClinicalTrials.gov
['NCT03783078']

Types de publication

Journal Article

Langues

eng

Sous-ensembles de citation

IM

Informations de copyright

© 2024. The Author(s).

Références

Mcevoy AM, Lachance K, Hippe DS, Cahill K, Moshiri Y, Lewis CW, et al. Recurrence and mortality risk of Merkel cell carcinoma by cancer stage and time from diagnosis. JAMA Dermatol. 2022;158(4):382–9.
doi: 10.1001/jamadermatol.2021.6096 pubmed: 35195657 pmcid: 8867389
Lewis CW, Qazi J, Hippe DS, Lachance K, Thomas H, Cook MM, et al. Patterns of distant metastases in 215 Merkel cell carcinoma patients: implications for prognosis and surveillance. Cancer Med. 2020;9(4):1374–82.
doi: 10.1002/cam4.2781 pubmed: 31883234
Harms KL, Healy MA, Nghiem P, Sober AJ, Johnson TM, Bichakjian CK, et al. Analysis of prognostic factors from 9387 Merkel cell carcinoma cases forms the basis for the new 8th edition AJCC staging system. Ann Surg Oncol. 2016;23(11):3564–71.
doi: 10.1245/s10434-016-5266-4 pubmed: 27198511 pmcid: 8881989
DeCaprio JA. Molecular pathogenesis of Merkel cell carcinoma. Annu Rev Pathol. 2021;16:69–91.
doi: 10.1146/annurev-pathmechdis-012419-032817
Park SY, Doolittle-Amieva C, Moshiri Y, Akaike T, Parvathaneni U, Bhatia S, et al. How we treat Merkel cell carcinoma: within and beyond current guidelines. Future Oncol. 2021;17(11):1363–77.
doi: 10.2217/fon-2020-1036 pubmed: 33511866 pmcid: 7983043
Baker M, Cordes L, Brownell I. Avelumab: a new standard for treating metastatic merkel cell carcinoma. Expert Rev Anticancer Ther. 2018;18(4):319–26.
doi: 10.1080/14737140.2018.1445528 pubmed: 29482384
Kaufman HL, Russell J, Hamid O, Bhatia S, Terheyden P, Dangelo SP, et al. Avelumab in patients with chemotherapy-refractory metastatic Merkel cell carcinoma: a multicentre, single-group, open-label, phase 2 trial. Lancet Oncol. 2016;17(10):1374–85.
doi: 10.1016/S1470-2045(16)30364-3 pubmed: 27592805 pmcid: 5587154
D’Angelo SP, Lebbé C, Mortier L, Brohl AS, Fazio N, Grob JJ, et al. First-line avelumab in a cohort of 116 patients with metastatic Merkel cell carcinoma (JAVELIN Merkel 200): primary and biomarker analyses of a phase II study. J Immunother Cancer. 2021;9(7):e002646.
doi: 10.1136/jitc-2021-002646 pubmed: 34301810 pmcid: 8311489
Nghiem PT, Bhatia S, Lipson EJ, Kudchadkar RR, Miller NJ, Annamalai L, et al. PD-1 blockade with pembrolizumab in advanced Merkel-cell carcinoma. N Engl J Med. 2016;374(26):2542–52.
doi: 10.1056/NEJMoa1603702 pubmed: 27093365 pmcid: 4927341
Bradford D, Demko S, Jin S, Mishra-Kalyani P, Beckles AR, Goldberg KB, et al. FDA accelerated approval of pembrolizumab for recurrent locally advanced or metastatic Merkel cell carcinoma. Oncologist. 2020;25(7):e1077–82.
doi: 10.1634/theoncologist.2020-0184 pubmed: 32272501 pmcid: 7356706
Nghiem P, Bhatia S, Lipson EJ, Sharfman WH, Kudchadkar RR, Brohl AS, et al. Three-year survival, correlates and salvage therapies in patients receiving first-line pembrolizumab for advanced Merkel cell carcinoma. J Immunother Cancer. 2021;9(4):e002478.
doi: 10.1136/jitc-2021-002478 pubmed: 33879601 pmcid: 8061836
Topalian SL, Bhatia S, Hollebecque A, Awada A, Boer JPD, Kudchadkar RR, et al. Abstract CT074: non-comparative, open-label, multiple cohort, phase 1/2 study to evaluate nivolumab (nivo) in patients with virus-associated tumors (CheckMate 358): efficacy and safety in Merkel cell carcinoma (MCC). Cancer Res. 2017;77(13_Supplement):CT074.
doi: 10.1158/1538-7445.AM2017-CT074
Topalian SL, Bhatia S, Amin A, Kudchadkar RR, Sharfman WH, Lebbé C, et al. Neoadjuvant nivolumab for patients with resectable Merkel cell carcinoma in the checkmate 358 trial. J Clin Oncol. 2020;38(22):2476–87.
doi: 10.1200/JCO.20.00201 pubmed: 32324435 pmcid: 7392746
Grignani G, Rutkowski P, Lebbe C, Guida M, Gaudy Marqueste C, De Braud FGM, et al. Updated results from POD1UM-201: a phase II study of retifanlimab in patients with advanced or metastatic Merkel cell carcinoma (MCC). Ann Oncol. 2023;34:S686.
doi: 10.1016/j.annonc.2023.09.2280
Miller NJ, Bhatia S, Parvathaneni U, Iyer JG, Nghiem P. Emerging and mechanism-based therapies for recurrent or metastatic Merkel cell carcinoma. Curr Treat Options Oncol. 2013;14(2):249–63.
doi: 10.1007/s11864-013-0225-9 pubmed: 23436166 pmcid: 3651762
Steuten L, Garmo V, Phatak H, Sullivan SD, Nghiem P, Ramsey SD. Treatment patterns, overall survival, and total healthcare costs of advanced Merkel cell carcinoma in the USA. Appl Health Econ Health Policy. 2019;17(5):733–40.
doi: 10.1007/s40258-019-00492-5 pubmed: 31250217 pmcid: 6748883
Iyer JG, Blom A, Doumani R, Lewis C, Tarabadkar ES, Anderson A, et al. Response rates and durability of chemotherapy among 62 patients with metastatic Merkel cell carcinoma. Cancer Med. 2016;5(9):2294–301.
doi: 10.1002/cam4.815 pubmed: 27431483 pmcid: 5055152
Cowey CL, Mahnke L, Espirito J, Helwig C, Oksen D, Bharmal M. Real-world treatment outcomes in patients with metastatic Merkel cell carcinoma treated with chemotherapy in the USA. Future Oncol. 2017;13(19):1699–710.
doi: 10.2217/fon-2017-0187 pubmed: 28605939
Nghiem P, Bhatia S, Lipson EJ, Sharfman WH, Kudchadkar RR, Brohl AS, et al. Durable tumor regression and overall survival in patients with advanced Merkel cell carcinoma receiving pembrolizumab as first-line therapy. J Clin Oncol. 2019;37(9):693–702.
doi: 10.1200/JCO.18.01896 pubmed: 30726175 pmcid: 6424137
U.S. Food & Drug Administration. FDA grants accelerated approval toretifanlimab-dlwr for metastatic or recurrent locally advanced Merkel cellcarcinoma. Silver Spring, MD: U.S. Food & Drug Administration; 2023. https://www.fda.gov/drugs/resources-information-approved-drugs/fda-grants-accelerated-approval-retifanlimab-dlwr-metastatic-or-recurrent-locally-advanced-merkel .
Lohray R, Verma KK, Wang LL, Haynes D, Lewis DJ. Avelumab for advanced Merkel cell carcinoma: global real-world data on patient response and survival. Pragmat Obs Res. 2023;14:149–54.
pubmed: 38021416 pmcid: 10658947
Bhatia S, Nghiem P, Veeranki SP, Vanegas A, Lachance K, Tachiki L, et al. Real-world clinical outcomes with avelumab in patients with Merkel cell carcinoma treated in the USA: a multicenter chart review study. J Immunother Cancer. 2022;10(8):e004904.
doi: 10.1136/jitc-2022-004904 pubmed: 35981787 pmcid: 9394192
Bhanegaonkar A, Liu FX, Boyd M, Fulcher N, Kim R, Krulewicz S, et al. Real-world clinical outcomes in patients with locally advanced or metastatic Merkel cell carcinoma treated in U.S. oncology clinical practices: results from SPEAR-Merkel. Oncologist. 2021;26(9):e1633–43.
doi: 10.1002/onco.13845 pubmed: 34101298 pmcid: 8417847
Robert C, Hwu WJ, Hamid O, Ribas A, Weber JS, Daud AI, et al. Long-term safety of pembrolizumab monotherapy and relationship with clinical outcome: a landmark analysis in patients with advanced melanoma. Eur J Cancer. 2021;144:182–91.
doi: 10.1016/j.ejca.2020.11.010 pubmed: 33360855

Auteurs

Laurent Mortier (L)

Université Lille, CHRU Lille, 42 Rue Paul Duez, Lille, France. laurent.mortier@chru-lille.fr.

Lisa Villabona (L)

Karolinska University Hospital, Akademiska stråket 13, G4:04, 17176, Stockholm, Sweden.

Ben Lawrence (B)

University of Auckland, 85 Park Rd, Auckland City Hospital 2 Park Rd, Auckland, New Zealand.

Ana Arance (A)

Hospital Clinic Barcelona and IDIBAPS, C. de Villarroel, 170, Barcelona, Spain.

Marcus O Butler (MO)

Departments of Medicine and Immunology, University of Toronto, 610 University Avenue, Toronto, ON, Canada.

Marie Beylot-Barry (M)

Centre Hospitalier Universitaire de Bordeaux, INSERM 1312, 1 Rue Jean Burguet, Bordeaux, France.

Philippe Saiag (P)

Hôpital Ambroise Paré, APHP & EA4340, University of Versailles-SQY, and Paris-Saclay University, 9 Av. Charles de Gaulle, Boulogne-Billancourt, France.

Mahtab Samimi (M)

University of Tours, France; ISP1282 INRA University of Tours, 60 Rue du Plat d'Étain, Tours, France.

Paolo A Ascierto (PA)

Istituto Nazionale Tumori IRCCS Fondazione "G. Pascale", Via Mariano Semmola, 53, Naples, Italy.

Francesca Spada (F)

Istituto Europeo di Oncologia (IEO) IRCCS, Via Giuseppe Ripamonti, 435, Milan, Italy.

Michel De Pontville (M)

Centre Hospitalier Universitaire de Caen-Hôpital Côte de Nacre, Av. de la Côte de Nacre CS 30001, Caen, France.

Michele Maio (M)

University of Siena and Center for Immuno-Oncology, University Hospital of Siena, Siena, Italy.

Alfonso Berrocal (A)

Hospital General Universitario de Valencia, Avda. Tres Cruces, 2, Valencia, Spain.

Enrique Espinosa (E)

Service of Oncology, Hospital Universitario La Paz, Universidad Autónoma de Madrid - CIBERONC, P. Castellana, 261-Madrid, Spain.

Jaume Capdevila (J)

Vall d'Hebron Institute of Oncology (VHIO), Vall d'Hebron University Hospital, Pg. de la Vall d'Hebron, 119, Barcelona, Spain.

Max Levin (M)

University of Gothenburg and Sahlgrenska University Hospital, Universitetsplatsen 1, Gothenburg, Sweden.

Debasmita Das (D)

Merck & Co., Inc., 126 E. Lincoln Ave, Rahway, NJ, USA.

Clemens Krepler (C)

Merck & Co., Inc., 126 E. Lincoln Ave, Rahway, NJ, USA.

Dmitri Grebennik (D)

Merck & Co., Inc., 126 E. Lincoln Ave, Rahway, NJ, USA.

Vanna Chiarion-Sileni (V)

Istituto Oncologico Veneto IOV-IRCCS, Via Gattamelata, 64, Padua, Italy.

Classifications MeSH