Extraordinary therapeutic effect of PSMA radioligand therapy in treatment-refractory progressive metastatic prostate cancer with the transketolase inhibitor benfo-oxythiamine as a radiosensitizer-A case report.

177Lu-PSMA TKTL1 benfo-oxythiamine case report metastatic castration-resistant prostate cancer radiosensitizer thiamine antagonist transketolase

Journal

Frontiers in medicine
ISSN: 2296-858X
Titre abrégé: Front Med (Lausanne)
Pays: Switzerland
ID NLM: 101648047

Informations de publication

Date de publication:
2024
Historique:
received: 09 07 2024
accepted: 28 08 2024
medline: 24 10 2024
pubmed: 24 10 2024
entrez: 24 10 2024
Statut: epublish

Résumé

Herein we report, for the first time, the therapeutic response of a prostate cancer patient with the thiamine antagonist benfo-oxythiamine (B-OT) added to prostate-specific membrane antigen (PSMA)-targeted radioligand therapy (PRLT). The patient was initially diagnosed as pT3b pN0 (0/7) M0 L0 V0 R0 G3, Gleason score 5 + 5 = 10, with an initial prostate-specific antigen (PSA) level of 4.05 ng/ml. Shortly after radical prostatectomy,

Identifiants

pubmed: 39444815
doi: 10.3389/fmed.2024.1462234
pmc: PMC11496175
doi:

Types de publication

Case Reports Journal Article

Langues

eng

Pagination

1462234

Informations de copyright

Copyright © 2024 Kramer, Zhang and Baum.

Déclaration de conflit d'intérêts

RB is a shareholder of Benfovir AG and Oxy5 OncoMedical AG. The remaining authors declare that the research was conducted in the absence of any commercial or financial relationships that could be construed as a potential conflict of interest.

Auteurs

Carsten S Kramer (CS)

CURANOSTICUM Wiesbaden-Frankfurt, Center for Advanced Radiomolecular Precision Oncology, Wiesbaden, Germany.

Jingjing Zhang (J)

Department of Diagnostic Radiology, Clinical Imaging Research Centre, National University of Singapore, Singapore, Singapore.

Richard P Baum (RP)

CURANOSTICUM Wiesbaden-Frankfurt, Center for Advanced Radiomolecular Precision Oncology, Wiesbaden, Germany.

Classifications MeSH