Kinetic Analysis and Metabolism of Poly(Adenosine Diphosphate-Ribose) Polymerase-1-Targeted

18F-fluorthanatrace PARP-1 breast cancer radiotracer tissue pharmacokinetics

Journal

Journal of nuclear medicine : official publication, Society of Nuclear Medicine
ISSN: 1535-5667
Titre abrégé: J Nucl Med
Pays: United States
ID NLM: 0217410

Informations de publication

Date de publication:
30 Oct 2024
Historique:
received: 17 06 2024
accepted: 11 09 2024
medline: 31 10 2024
pubmed: 31 10 2024
entrez: 30 10 2024
Statut: aheadofprint

Résumé

The poly(adenosine diphosphate-ribose) polymerase inhibitors (PARPi) have demonstrated efficacy in ovarian, breast, and prostate cancers, but current biomarkers do not consistently predict clinical benefit.

Identifiants

pubmed: 39477499
pii: jnumed.124.268254
doi: 10.2967/jnumed.124.268254
pii:
doi:

Types de publication

Journal Article

Langues

eng

Sous-ensembles de citation

IM

Informations de copyright

© 2024 by the Society of Nuclear Medicine and Molecular Imaging.

Auteurs

Anthony J Young (AJ)

Department of Radiology, Perelman School of Medicine, University of Pennsylvania, Philadelphia, Pennsylvania.

Austin R Pantel (AR)

Department of Radiology, Perelman School of Medicine, University of Pennsylvania, Philadelphia, Pennsylvania.

Mahsa Kiani (M)

Department of Radiology, Perelman School of Medicine, University of Pennsylvania, Philadelphia, Pennsylvania.

Robert K Doot (RK)

Department of Radiology, Perelman School of Medicine, University of Pennsylvania, Philadelphia, Pennsylvania.

Sina Bagheri (S)

Department of Radiology, Perelman School of Medicine, University of Pennsylvania, Philadelphia, Pennsylvania.

Daniel A Pryma (DA)

Department of Radiology, Perelman School of Medicine, University of Pennsylvania, Philadelphia, Pennsylvania.

Michael D Farwell (MD)

Department of Radiology, Perelman School of Medicine, University of Pennsylvania, Philadelphia, Pennsylvania.

Shihong Li (S)

Department of Radiology, Perelman School of Medicine, University of Pennsylvania, Philadelphia, Pennsylvania.

Hsiaoju Lee (H)

Department of Radiology, Perelman School of Medicine, University of Pennsylvania, Philadelphia, Pennsylvania.

Erin K Schubert (EK)

Department of Radiology, Perelman School of Medicine, University of Pennsylvania, Philadelphia, Pennsylvania.

Anthony Secreto (A)

Department of Hematology and Oncology, Perelman School of Medicine, University of Pennsylvania, Philadelphia, Pennsylvania.

Samantha P Zuckerman (SP)

Department of Radiology, Perelman School of Medicine, University of Pennsylvania, Philadelphia, Pennsylvania.

Anupma Nayak (A)

Department of Pathology, Perelman School of Medicine, University of Pennsylvania, Philadelphia, Pennsylvania.

Hoon Choi (H)

Department of Radiology, Perelman School of Medicine, University of Pennsylvania, Philadelphia, Pennsylvania.

Sean Carlin (S)

Invicro LLC, Needham, Massachusetts; and.

Angela DeMichele (A)

Department of Medicine, Perelman School of Medicine, University of Pennsylvania, Philadelphia, Pennsylvania.

David A Mankoff (DA)

Department of Radiology, Perelman School of Medicine, University of Pennsylvania, Philadelphia, Pennsylvania.

Rong Zhou (R)

Department of Radiology, Perelman School of Medicine, University of Pennsylvania, Philadelphia, Pennsylvania.

Robert H Mach (RH)

Department of Radiology, Perelman School of Medicine, University of Pennsylvania, Philadelphia, Pennsylvania.

Elizabeth S McDonald (ES)

Department of Radiology, Perelman School of Medicine, University of Pennsylvania, Philadelphia, Pennsylvania; elizabeth.mcdonald@pennmedicine.upenn.edu.

Classifications MeSH