Accueil
Ester Colarusso
Ester Colarusso
Affiliations
Department of Pharmacy, University of Salerno, Via Giovanni Paolo II, 132, 84084 Fisciano, Italy. Electronic address: ecolarusso@unisa.it.
Publications (11)
2-Substituted 1,5-benzothiazepine-based HDAC inhibitors exert anticancer activities on human solid and acute myeloid leukemia cell lines.
Bioorganic & medicinal chemistry
Avec:
Simona De Vita
,
Sara Meninno
,
Lucia Capasso
,
Ester Colarusso
,
Maria Giovanna Chini
,
Gianluigi Lauro
,
Romolo Rinaldi
,
Annalisa De Cicco
,
Veronica Sian
,
Stefania Terracciano
,
Angela Nebbioso
,
Alessandra Lattanzi
,
Giuseppe Bifulco
Repositioning of Small Molecules through the Inverse Virtual Screening in silico Tool: Case of Benzothiazole-Based Inhibitors of Soluble Epoxide Hydrolase (sEH).
ChemPlusChem
Avec:
Erica Gazzillo
,
Ester Colarusso
,
Assunta Giordano
,
Maria Giovanna Chini
,
Marianna Potenza
,
Robert Klaus Hofstetter
,
Maria Iorizzi
,
Oliver Werz
,
Gianluigi Lauro
,
Giuseppe Bifulco
PharmaCore: The Automatic Generation of 3D Structure-Based Pharmacophore Models from Protein/Ligand Complexes.
Journal of chemical information and modeling
Avec:
Simona De Vita
,
Ester Colarusso
,
Maria Giovanna Chini
,
Giuseppe Bifulco
,
Gianluigi Lauro
Identification of Novel Bromodomain-Containing Protein 4 (BRD4) Binders through 3D Pharmacophore-Based Repositioning Screening Campaign.
Molecules (Basel, Switzerland)
Avec:
Ester Colarusso
,
Erica Gazzillo
,
Eleonora Boccia
,
Stefania Terracciano
,
Ines Bruno
,
Giuseppe Bifulco
,
Maria Giovanna Chini
,
Gianluigi Lauro
In Silico Design, Chemical Synthesis, Biophysical and In Vitro Evaluation for the Identification of 1-ethyl-1H-pyrazolo[3,4-b]pyridine-based BRD9 Binders.
ChemPlusChem
Avec:
Ester Colarusso
,
Erica Gazzillo
,
Martina Pierri
,
Dafne Ruggiero
,
Maria Giovanna Chini
,
Ines Bruno
,
Giuseppe Bifulco
,
Stefania Terracciano
,
Gianluigi Lauro
Chemical Profiling of Polar Lipids and the Polyphenolic Fraction of Commercial Italian
Biomolecules
Avec:
Vadym Samukha
,
Francesca Fantasma
,
Gilda D'Urso
,
Ester Colarusso
,
Anna Schettino
,
Noemi Marigliano
,
Maria Giovanna Chini
,
Gabriella Saviano
,
Vincenzo De Felice
,
Gianluigi Lauro
,
Francesco Maione
,
Giuseppe Bifulco
,
Agostino Casapullo
,
Maria Iorizzi
Identification of 2,4,5-trisubstituted-2,4-dihydro-3H-1,2,4-triazol-3-one-based small molecules as selective BRD9 binders.
European journal of medicinal chemistry
Avec:
Ester Colarusso
,
Sara Ceccacci
,
Maria Chiara Monti
,
Erica Gazzillo
,
Assunta Giordano
,
Maria Giovanna Chini
,
Maria Grazia Ferraro
,
Marialuisa Piccolo
,
Dafne Ruggiero
,
Carlo Irace
,
Stefania Terracciano
,
Ines Bruno
,
Giuseppe Bifulco
,
Gianluigi Lauro
Unemployment Status Subsequent to Cancer Diagnosis and Therapies: A Systematic Review and Meta-Analysis.
Cancers
Avec:
Martina Chimienti
,
Giustino Morlino
,
Fabio Ingravalle
,
Antonio Vinci
,
Emilio Colarusso
,
Carolina De Santo
,
Valeria Formosa
,
Lavinia Gentile
,
Grazia Lorusso
,
Claudia Mosconi
,
Martina Scaramella
,
Virginia Rosca
,
Elena Veneziano
,
Francesco Torino
,
Leonardo Emberti Gialloreti
,
Leonardo Palombi
Targeting mPGES-1 by a Combinatorial Approach: Identification of the Aminobenzothiazole Scaffold to Suppress PGE
ACS medicinal chemistry letters
Avec:
Maria G Chini
,
Assunta Giordano
,
Marianna Potenza
,
Stefania Terracciano
,
Katrin Fischer
,
Maria C Vaccaro
,
Ester Colarusso
,
Ines Bruno
,
Raffaele Riccio
,
Andreas Koeberle
,
Oliver Werz
,
Giuseppe Bifulco
Exploring the chemical space of functionalized [1,2,4]triazolo[4,3-a]quinoxaline-based compounds targeting the bromodomain of BRD9.
Bioorganic chemistry
Avec:
Erica Gazzillo
,
Martina Pierri
,
Ester Colarusso
,
Maria Giovanna Chini
,
Maria Grazia Ferraro
,
Marialuisa Piccolo
,
Carlo Irace
,
Ines Bruno
,
Giuseppe Bifulco
,
Stefania Terracciano
,
Gianluigi Lauro
Identification and Development of BRD9 Chemical Probes.
Pharmaceuticals (Basel, Switzerland)
Avec:
Ester Colarusso
,
Maria Giovanna Chini
,
Giuseppe Bifulco
,
Gianluigi Lauro
,
Assunta Giordano
Réseau de co-auteurs
Giuseppe Bifulco
10 collaborations
Maria Giovanna Chini
9 collaborations
Gianluigi Lauro
9 collaborations
Stefania Terracciano
6 collaborations
Erica Gazzillo
5 collaborations
Ines Bruno
5 collaborations
Assunta Giordano
4 collaborations
Simona De Vita
2 collaborations
Marianna Potenza
2 collaborations
Maria Iorizzi
2 collaborations
Oliver Werz
2 collaborations
Martina Pierri
2 collaborations
Dafne Ruggiero
2 collaborations
Maria Grazia Ferraro
2 collaborations
Marialuisa Piccolo
2 collaborations
Carlo Irace
2 collaborations
Sara Meninno
1 collaboration
Lucia Capasso
1 collaboration
Romolo Rinaldi
1 collaboration
Annalisa De Cicco
1 collaboration
Veronica Sian
1 collaboration
Angela Nebbioso
1 collaboration
Alessandra Lattanzi
1 collaboration
Robert Klaus Hofstetter
1 collaboration
Eleonora Boccia
1 collaboration
Vadym Samukha
1 collaboration
Francesca Fantasma
1 collaboration
Gilda D'Urso
1 collaboration
Anna Schettino
1 collaboration
Noemi Marigliano
1 collaboration
Gabriella Saviano
1 collaboration
Vincenzo De Felice
1 collaboration
Francesco Maione
1 collaboration
Agostino Casapullo
1 collaboration
Sara Ceccacci
1 collaboration
Maria Chiara Monti
1 collaboration
Martina Chimienti
1 collaboration
Giustino Morlino
1 collaboration
Fabio Ingravalle
1 collaboration
Antonio Vinci
1 collaboration
Emilio Colarusso
1 collaboration
Carolina De Santo
1 collaboration
Valeria Formosa
1 collaboration
Lavinia Gentile
1 collaboration
Grazia Lorusso
1 collaboration
Claudia Mosconi
1 collaboration
Martina Scaramella
1 collaboration
Virginia Rosca
1 collaboration
Elena Veneziano
1 collaboration
Francesco Torino
1 collaboration
Leonardo Emberti Gialloreti
1 collaboration
Leonardo Palombi
1 collaboration
Maria G Chini
1 collaboration
Katrin Fischer
1 collaboration
Maria C Vaccaro
1 collaboration
Raffaele Riccio
1 collaboration
Andreas Koeberle
1 collaboration