Accueil
Fumihito Ushiyama
Fumihito Ushiyama
Affiliations
Taisho Pharmaceutical Co., Ltd, 1-403 Yoshino-Cho, Kita-Ku, Saitama 331-9530, Japan. Electronic address: f-ushiyama@taisho.co.jp.
Publications (5)
Lead optimization of 2-hydroxymethyl imidazoles as non-hydroxamate LpxC inhibitors: Discovery of TP0586532.
Bioorganic & medicinal chemistry
Avec:
Fumihito Ushiyama
,
Hajime Takashima
,
Yohei Matsuda
,
Yuya Ogata
,
Naoki Sasamoto
,
Risa Kurimoto-Tsuruta
,
Kaori Ueki
,
Nozomi Tanaka-Yamamoto
,
Mayumi Endo
,
Masashi Mima
,
Kiyoko Fujita
,
Iichiro Takata
,
Satoshi Tsuji
,
Haruhiro Yamashita
,
Hirotoshi Okumura
,
Katsumasa Otake
,
Hiroyuki Sugiyama
Lead optimization of 8-(methylamino)-2-oxo-1,2-dihydroquinolines as bacterial type II topoisomerase inhibitors.
Bioorganic & medicinal chemistry
Avec:
Fumihito Ushiyama
,
Hideaki Amada
,
Yasuhiro Mihara
,
Tomoki Takeuchi
,
Nozomi Tanaka-Yamamoto
,
Masashi Mima
,
Masafumi Kamitani
,
Reiko Wada
,
Yunoshin Tamura
,
Mayumi Endo
,
Aiko Masuko
,
Iichiro Takata
,
Kosuke Hitaka
,
Hiroyuki Sugiyama
,
Norikazu Ohtake
Fragment-Based Discovery of Novel Non-Hydroxamate LpxC Inhibitors with Antibacterial Activity.
Journal of medicinal chemistry
Avec:
Yousuke Yamada
,
Hajime Takashima
,
David Lee Walmsley
,
Fumihito Ushiyama
,
Yohei Matsuda
,
Harumi Kanazawa
,
Toru Yamaguchi-Sasaki
,
Nozomi Tanaka-Yamamoto
,
Junya Yamagishi
,
Risa Kurimoto-Tsuruta
,
Yuya Ogata
,
Norikazu Ohtake
,
Hayley Angove
,
Lisa Baker
,
Richard Harris
,
Alba Macias
,
Alan Robertson
,
Allan Surgenor
,
Hayato Watanabe
,
Koichiro Nakano
,
Masashi Mima
,
Kunihiko Iwamoto
,
Atsushi Okada
,
Iichiro Takata
,
Kosuke Hitaka
,
Akihiro Tanaka
,
Kiyoko Fujita
,
Hiroyuki Sugiyama
,
Roderick E Hubbard
Lead Identification of 8-(Methylamino)-2-oxo-1,2-dihydroquinoline Derivatives as DNA Gyrase Inhibitors: Hit-to-Lead Generation Involving Thermodynamic Evaluation.
ACS omega
Avec:
Fumihito Ushiyama
,
Hideaki Amada
,
Tomoki Takeuchi
,
Nozomi Tanaka-Yamamoto
,
Harumi Kanazawa
,
Koichiro Nakano
,
Masashi Mima
,
Aiko Masuko
,
Iichiro Takata
,
Kosuke Hitaka
,
Kunihiko Iwamoto
,
Hiroyuki Sugiyama
,
Norikazu Ohtake
Antimicrobial agents and chemotherapy
Avec:
Aiko Masuko
,
Iichiro Takata
,
Kiyoko Fujita
,
Hirotoshi Okumura
,
Fumihito Ushiyama
,
Hideaki Amada
,
Hiroyuki Sugiyama
Réseau de co-auteurs
Iichiro Takata
5 collaborations
Hiroyuki Sugiyama
5 collaborations
Nozomi Tanaka-Yamamoto
4 collaborations
Masashi Mima
4 collaborations
Kiyoko Fujita
3 collaborations
Hideaki Amada
3 collaborations
Aiko Masuko
3 collaborations
Kosuke Hitaka
3 collaborations
Norikazu Ohtake
3 collaborations
Hajime Takashima
2 collaborations
Yohei Matsuda
2 collaborations
Yuya Ogata
2 collaborations
Risa Kurimoto-Tsuruta
2 collaborations
Mayumi Endo
2 collaborations
Hirotoshi Okumura
2 collaborations
Tomoki Takeuchi
2 collaborations
Harumi Kanazawa
2 collaborations
Koichiro Nakano
2 collaborations
Kunihiko Iwamoto
2 collaborations
Naoki Sasamoto
1 collaboration
Kaori Ueki
1 collaboration
Satoshi Tsuji
1 collaboration
Haruhiro Yamashita
1 collaboration
Katsumasa Otake
1 collaboration
Yasuhiro Mihara
1 collaboration
Masafumi Kamitani
1 collaboration
Reiko Wada
1 collaboration
Yunoshin Tamura
1 collaboration
Yousuke Yamada
1 collaboration
David Lee Walmsley
1 collaboration
Toru Yamaguchi-Sasaki
1 collaboration
Junya Yamagishi
1 collaboration
Hayley Angove
1 collaboration
Lisa Baker
1 collaboration
Richard Harris
1 collaboration
Alba Macias
1 collaboration
Alan Robertson
1 collaboration
Allan Surgenor
1 collaboration
Hayato Watanabe
1 collaboration
Atsushi Okada
1 collaboration
Akihiro Tanaka
1 collaboration
Roderick E Hubbard
1 collaboration