Molecular Dynamic in Ethosuximide Glass Forming Pharmaceutical as Studied by Dielectric Relaxation Spectroscopy.


Journal

Journal of pharmaceutical sciences
ISSN: 1520-6017
Titre abrégé: J Pharm Sci
Pays: United States
ID NLM: 2985195R

Informations de publication

Date de publication:
Jan 2019
Historique:
received: 21 03 2018
revised: 15 06 2018
accepted: 29 06 2018
pubmed: 17 7 2018
medline: 15 2 2020
entrez: 17 7 2018
Statut: ppublish

Résumé

Polymorphism and molecular dynamics of ethosuximide with molecules of left- and right-handed chirality have been studied in detail using dielectric spectroscopy. Density functional theory calculations of molecular conformations and dimer formation were performed to aid the interpretation of measurements. Moving window correlation analysis of the imaginary part of dielectric permittivity spectra allowed us to complete the monotropic system of phases found by the differential scanning calorimetry method. Extra transition connected with freezing-in/activation of slow molecular motions was identified in partially ordered crystal CrI phase. In high-temperature orientationally disordered CrI

Identifiants

pubmed: 30009796
pii: S0022-3549(18)30397-6
doi: 10.1016/j.xphs.2018.06.030
pii:
doi:

Substances chimiques

Ethosuximide 5SEH9X1D1D

Types de publication

Journal Article

Langues

eng

Sous-ensembles de citation

IM

Pagination

102-108

Informations de copyright

Copyright © 2019. Published by Elsevier Inc.

Auteurs

Natalia Osiecka (N)

Institute of Nuclear Physics Polish Academy of Sciences, Kraków PL-31342, Poland. Electronic address: natalia.osiecka@ifj.edu.pl.

Mirosław Gałązka (M)

Institute of Nuclear Physics Polish Academy of Sciences, Kraków PL-31342, Poland.

Monika Marzec (M)

Institute of Physics, Jagiellonian University, S. Łojasiewicza 11, Kraków 30-348, Poland.

Wojciech Zając (W)

Institute of Nuclear Physics Polish Academy of Sciences, Kraków PL-31342, Poland.

Maria Massalska-Arodź (M)

Institute of Nuclear Physics Polish Academy of Sciences, Kraków PL-31342, Poland.

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Classifications MeSH