Enabling adoption of 2D-NMR for the higher order structure assessment of monoclonal antibody therapeutics.

NISTmAb chemometrics comparability higher order structure monoclonal antibody (mAb) therapeutics nuclear magnetic resonance spectroscopy (NMR)

Journal

mAbs
ISSN: 1942-0870
Titre abrégé: MAbs
Pays: United States
ID NLM: 101479829

Informations de publication

Date de publication:
01 2019
Historique:
pubmed: 21 12 2018
medline: 16 7 2019
entrez: 21 12 2018
Statut: ppublish

Résumé

The increased interest in using monoclonal antibodies (mAbs) as a platform for biopharmaceuticals has led to the need for new analytical techniques that can precisely assess physicochemical properties of these large and very complex drugs for the purpose of correctly identifying quality attributes (QA). One QA, higher order structure (HOS), is unique to biopharmaceuticals and essential for establishing consistency in biopharmaceutical manufacturing, detecting process-related variations from manufacturing changes and establishing comparability between biologic products. To address this measurement challenge, two-dimensional nuclear magnetic resonance spectroscopy (2D-NMR) methods were introduced that allow for the precise atomic-level comparison of the HOS between two proteins, including mAbs. Here, an inter-laboratory comparison involving 26 industrial, government and academic laboratories worldwide was performed as a benchmark using the NISTmAb, from the National Institute of Standards and Technology (NIST), to facilitate the translation of the 2D-NMR method into routine use for biopharmaceutical product development. Two-dimensional

Identifiants

pubmed: 30570405
doi: 10.1080/19420862.2018.1544454
pmc: PMC6343768
doi:

Substances chimiques

Antibodies, Monoclonal 0

Types de publication

Journal Article Research Support, Non-U.S. Gov't Research Support, U.S. Gov't, Non-P.H.S.

Langues

eng

Sous-ensembles de citation

IM

Pagination

94-105

Références

Prog Nucl Magn Reson Spectrosc. 2014 Nov;83:21-41
pubmed: 25456315
J Biomol NMR. 2012 Apr;52(4):315-27
pubmed: 22331404
Prog Nucl Magn Reson Spectrosc. 2013 Aug;73:1-16
pubmed: 23962882
Sci Rep. 2016 Aug 31;6:32201
pubmed: 27578487
J Biomol NMR. 1995 Nov;6(3):277-93
pubmed: 8520220
J Pharm Biomed Anal. 2019 Jan 30;163:144-152
pubmed: 30296716
J Biomol NMR. 1998 Jul;12(1):1-23
pubmed: 9729785
Pharm Res. 2015 Oct;32(10):3365-75
pubmed: 26043856
J Pharm Sci. 2017 Dec;106(12):3486-3498
pubmed: 28843351
Anal Chem. 2015 Apr 7;87(7):3556-61
pubmed: 25728213
J Biomol NMR. 2005 Dec;33(4):199-211
pubmed: 16341750
J Pharm Sci. 2015 Apr;104(4):1240-5
pubmed: 25711138
Bioinformatics. 2015 Apr 15;31(8):1325-7
pubmed: 25505092
Pharm Res. 2016 Feb;33(2):462-75
pubmed: 26453189
J Pharm Biomed Anal. 2018 Jan 5;147:367-377
pubmed: 28760370
Int J Pharm. 2016 Dec 30;515(1-2):390-402
pubmed: 27773853
MAbs. 2018 Feb/Mar;10(2):183-203
pubmed: 29300693
Anal Bioanal Chem. 2018 Mar;410(8):2127-2139
pubmed: 29411089
Anal Chem. 2017 Nov 7;89(21):11839-11845
pubmed: 28937210
J Am Chem Soc. 2010 Feb 24;132(7):2145-7
pubmed: 20121194
J Pharm Sci. 2016 Dec;105(12):3465-3470
pubmed: 27743675
Anal Bioanal Chem. 2018 Mar;410(8):2067-2078
pubmed: 29430600
Nat Rev Drug Discov. 2012 Jun 29;11(7):527-40
pubmed: 22743980
Anal Chem. 2008 Apr 1;80(7):2623-7
pubmed: 18321136
J Magn Reson. 2015 Dec;261:19-26
pubmed: 26524650
Methods Enzymol. 2016;566:3-34
pubmed: 26791974
Nat Biotechnol. 2016 Feb;34(2):139-41
pubmed: 26849514
Protein Expr Purif. 2015 Nov;115:1-10
pubmed: 26256059

Auteurs

Robert G Brinson (RG)

a Institute of Bioscience and Biotechnology Research , National Institute of Standards and Technology and the University of Maryland , Rockville , MD , USA.

John P Marino (JP)

a Institute of Bioscience and Biotechnology Research , National Institute of Standards and Technology and the University of Maryland , Rockville , MD , USA.

Frank Delaglio (F)

a Institute of Bioscience and Biotechnology Research , National Institute of Standards and Technology and the University of Maryland , Rockville , MD , USA.

Luke W Arbogast (LW)

a Institute of Bioscience and Biotechnology Research , National Institute of Standards and Technology and the University of Maryland , Rockville , MD , USA.

Ryan M Evans (RM)

b Applied and Computational Mathematics Division , National Institute of Standards and Technology , Gaithersburg , MD , USA.

Anthony Kearsley (A)

b Applied and Computational Mathematics Division , National Institute of Standards and Technology , Gaithersburg , MD , USA.

Geneviève Gingras (G)

c Centre for Biologics Evaluation, Biologics and Genetic Therapies Directorate , Health Canada , Ottawa , ON , Canada.

Houman Ghasriani (H)

c Centre for Biologics Evaluation, Biologics and Genetic Therapies Directorate , Health Canada , Ottawa , ON , Canada.

Yves Aubin (Y)

c Centre for Biologics Evaluation, Biologics and Genetic Therapies Directorate , Health Canada , Ottawa , ON , Canada.

Gregory K Pierens (GK)

d The Centre for Advanced Imaging , The University of Queensland , St Lucia , QLD , Australia.

Xinying Jia (X)

d The Centre for Advanced Imaging , The University of Queensland , St Lucia , QLD , Australia.

Mehdi Mobli (M)

d The Centre for Advanced Imaging , The University of Queensland , St Lucia , QLD , Australia.

Hamish G Grant (HG)

e Bio21 Molecular Science & Biotechnology Institute , The University of Melbourne , Victoria , Australia.

David W Keizer (DW)

e Bio21 Molecular Science & Biotechnology Institute , The University of Melbourne , Victoria , Australia.

Kristian Schweimer (K)

f Lehrstuhl Biopolymere , Universitaet Bayreuth , Bayreuth , Germany.

Jonas Ståhle (J)

g Department of Organic Chemistry , Arrhenius Laboratory, Stockholm University , Stockholm , Sweden.

Göran Widmalm (G)

g Department of Organic Chemistry , Arrhenius Laboratory, Stockholm University , Stockholm , Sweden.

Edward R Zartler (ER)

h Analytical R&D , Pfizer Essential Health , Lake Forest , IL , USA.

Chad W Lawrence (CW)

i Pacific Northwest National Laboratory , Earth and Biological Sciences Directorate , Richland , DC , USA.

Patrick N Reardon (PN)

i Pacific Northwest National Laboratory , Earth and Biological Sciences Directorate , Richland , DC , USA.

John R Cort (JR)

i Pacific Northwest National Laboratory , Earth and Biological Sciences Directorate , Richland , DC , USA.

Ping Xu (P)

j Department of Downstream Processing and Analytics , Human Health Therapeutics Research Centre, National Research Council of Canada , Montreal , Quebec , Canada.

Feng Ni (F)

j Department of Downstream Processing and Analytics , Human Health Therapeutics Research Centre, National Research Council of Canada , Montreal , Quebec , Canada.

Saeko Yanaka (S)

k Institute for Molecular Science and Exploratory Research Center on Life and Living Systems , National Institutes of Natural Sciences , Myodaiji, Okazaki , Japan.

Koichi Kato (K)

k Institute for Molecular Science and Exploratory Research Center on Life and Living Systems , National Institutes of Natural Sciences , Myodaiji, Okazaki , Japan.

Stuart R Parnham (SR)

l Department of Biochemistry and Molecular Biology , Medical University of South Carolina , Charleston , SC , USA.

Desiree Tsao (D)

m Analytical Development , Momenta Pharmaceuticals , Cambridge , MA , USA.

Andreas Blomgren (A)

n Laboratory Unit , Swedish Medical Products Agency, Laboratory , Uppsala , Sweden.

Torgny Rundlöf (T)

n Laboratory Unit , Swedish Medical Products Agency, Laboratory , Uppsala , Sweden.

Nils Trieloff (N)

o NMR-supported Structural Biology , Leibniz-Forschungsinstitut für Molekulare Pharmakologie (FMP) , Berlin , Germany.

Peter Schmieder (P)

o NMR-supported Structural Biology , Leibniz-Forschungsinstitut für Molekulare Pharmakologie (FMP) , Berlin , Germany.

Alfred Ross (A)

p Roche Pharmaceutical Research & Early Development , Pre-Clinical CMC, Roche Innovation Center Basel , Basel , Switzerland.

Ken Skidmore (K)

q Analytical Operations , Genentech , South San Francisco , CA , USA.

Kang Chen (K)

r Center for Drug Evaluation and Research , Food and Drug Administration , Maryland , USA.

David Keire (D)

r Center for Drug Evaluation and Research , Food and Drug Administration , Maryland , USA.

Darón I Freedberg (DI)

s Center for Biologics Evaluation and Research , Food and Drug Administration , Maryland , USA.

Thea Suter-Stahel (T)

t Department of Biology , Institute of Molecular Biology and Biophysics , ETH Zurich, Zurich , Switzerland.

Gerhard Wider (G)

t Department of Biology , Institute of Molecular Biology and Biophysics , ETH Zurich, Zurich , Switzerland.

Gregor Ilc (G)

u NMR Centre , EN-FIST Centre of Excellence , Ljubljana , Slovenia.
v NMR Centre , National Institute of Chemistry , Ljubljana , Slovenia.

Janez Plavec (J)

u NMR Centre , EN-FIST Centre of Excellence , Ljubljana , Slovenia.
v NMR Centre , National Institute of Chemistry , Ljubljana , Slovenia.

Scott A Bradley (SA)

w Eli Lilly and Company , Lilly Corporate Center , Indianapolis , IN , USA.

Donna M Baldisseri (DM)

x MRS - Application Science , Bruker BioSpin Corporation , Billerica , MA , USA.

Mauricio Luis Sforça (ML)

y Brazilian Biosciences National Laboratory (LNBio), Brazilian Center for Research in Energy and Materials (CNPEM) , Campinas, Brazil.

Ana Carolina de Mattos Zeri (ACM)

z Brazilian Synchrotron Light Laboratory (LNLS), Brazilian Center for Research in Energy and Materials (CNPEM) , Campinas, Brazil , CEP.

Julie Yu Wei (JY)

aa Protein Product Development , Biogen Inc ., Cambridge , MA , USA.

Christina M Szabo (CM)

ab Baxter Pharmaceuticals R&D , Baxter Healthcare , Round Lake, IL , USA.

Carlos A Amezcua (CA)

ab Baxter Pharmaceuticals R&D , Baxter Healthcare , Round Lake, IL , USA.

John B Jordan (JB)

ac Global Regulatory and R&D Policy , Amgen Inc ., Thousand Oaks , CA , USA.

Mats Wikström (M)

ad Higher Order Structure, Attribute Sciences , Amgen Inc ., Thousand Oaks , CA , USA.

Articles similaires

[Redispensing of expensive oral anticancer medicines: a practical application].

Lisanne N van Merendonk, Kübra Akgöl, Bastiaan Nuijen
1.00
Humans Antineoplastic Agents Administration, Oral Drug Costs Counterfeit Drugs

Smoking Cessation and Incident Cardiovascular Disease.

Jun Hwan Cho, Seung Yong Shin, Hoseob Kim et al.
1.00
Humans Male Smoking Cessation Cardiovascular Diseases Female
Humans United States Aged Cross-Sectional Studies Medicare Part C
1.00
Humans Yoga Low Back Pain Female Male

Classifications MeSH