DPP10 is a new regulator of Nav1.5 channels in human heart.


Journal

International journal of cardiology
ISSN: 1874-1754
Titre abrégé: Int J Cardiol
Pays: Netherlands
ID NLM: 8200291

Informations de publication

Date de publication:
01 06 2019
Historique:
received: 20 06 2018
revised: 14 12 2018
accepted: 27 12 2018
pubmed: 15 1 2019
medline: 7 1 2020
entrez: 15 1 2019
Statut: ppublish

Résumé

Cardiac accessory β-subunits are part of macromolecular Nav1.5 channel complexes modulating biophysical properties and contributing to arrhythmias. Recent studies demonstrated the structural interaction between β-subunits of Na We assessed DPP10 expression in the healthy and diseased human heart and we studied the functional effects of DPP10 on the Na DPP10 mRNA and proteins were detected in human ventricle, with higher levels in patients with heart failure. In rat cardiomyocytes, DPP10ad significantly reduced upstroke velocity of action potentials indicating reduction in Na We provide first evidence that DPP10 interacts with Nav1.5 channels, linking Na

Sections du résumé

BACKGROUND
Cardiac accessory β-subunits are part of macromolecular Nav1.5 channel complexes modulating biophysical properties and contributing to arrhythmias. Recent studies demonstrated the structural interaction between β-subunits of Na
METHODS
We assessed DPP10 expression in the healthy and diseased human heart and we studied the functional effects of DPP10 on the Na
RESULTS
DPP10 mRNA and proteins were detected in human ventricle, with higher levels in patients with heart failure. In rat cardiomyocytes, DPP10ad significantly reduced upstroke velocity of action potentials indicating reduction in Na
CONCLUSION
We provide first evidence that DPP10 interacts with Nav1.5 channels, linking Na

Identifiants

pubmed: 30638748
pii: S0167-5273(18)34013-0
doi: 10.1016/j.ijcard.2018.12.072
pii:
doi:

Substances chimiques

NAV1.5 Voltage-Gated Sodium Channel 0
RNA 63231-63-0
DPP10 protein, human EC 3.4.14.-
Dipeptidyl-Peptidases and Tripeptidyl-Peptidases EC 3.4.14.-

Types de publication

Journal Article

Langues

eng

Sous-ensembles de citation

IM

Pagination

68-73

Commentaires et corrections

Type : CommentIn

Informations de copyright

Copyright © 2019 Elsevier B.V. All rights reserved.

Auteurs

Fabian Belau (F)

Rudolf-Boehm-Institute of Pharmacology and Toxicology, Leipzig University, Leipzig, Germany.

Katharina Metzner (K)

Rudolf-Boehm-Institute of Pharmacology and Toxicology, Leipzig University, Leipzig, Germany.

Torsten Christ (T)

Institute of Experimental Pharmacology and Toxicology, DZHK (German Center for Cardiovascular Research), partner site Hamburg/Kiel/Lübeck, University Medical Center Hamburg Eppendorf, Hamburg, Germany.

Ursula Ravens (U)

Department of Physiology, TU Dresden, Dresden, Germany; Institute of Experimental Cardiovascular Medicine, University Heart Centre Freiburg-Bad Krozingen, Freiburg, Germany.

Michael Schaefer (M)

Rudolf-Boehm-Institute of Pharmacology and Toxicology, Leipzig University, Leipzig, Germany.

Stephan Künzel (S)

Department of Pharmacology and Toxicology, TU Dresden, Dresden, Germany.

Wener Li (W)

Department of Pharmacology and Toxicology, TU Dresden, Dresden, Germany.

Erich Wettwer (E)

Institute of Pharmacology, West German Heart and Vascular Center, University Duisburg-Essen, Essen, Germany.

Dobromir Dobrev (D)

Institute of Pharmacology, West German Heart and Vascular Center, University Duisburg-Essen, Essen, Germany.

Ali El-Armouche (A)

Department of Pharmacology and Toxicology, TU Dresden, Dresden, Germany.

Susanne Kämmerer (S)

Rudolf-Boehm-Institute of Pharmacology and Toxicology, Leipzig University, Leipzig, Germany; Department of Pharmacology and Toxicology, TU Dresden, Dresden, Germany. Electronic address: susanne.kaemmerer@tu-dresden.de.

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Classifications MeSH