Facilitation of
Action Potentials
Animals
Anti-Arrhythmia Agents
/ pharmacology
Cells, Cultured
ERG1 Potassium Channel
/ antagonists & inhibitors
HEK293 Cells
Humans
Myocytes, Cardiac
/ drug effects
Phenethylamines
/ pharmacology
Potassium Channel Blockers
/ pharmacology
Pyrimidinones
/ pharmacology
Rabbits
Sulfonamides
/ pharmacology
Xenopus
Journal
The Journal of general physiology
ISSN: 1540-7748
Titre abrégé: J Gen Physiol
Pays: United States
ID NLM: 2985110R
Informations de publication
Date de publication:
04 02 2019
04 02 2019
Historique:
received:
30
07
2018
accepted:
06
12
2018
pubmed:
25
1
2019
medline:
1
5
2020
entrez:
25
1
2019
Statut:
ppublish
Résumé
Drug-induced block of the cardiac rapid delayed rectifying potassium current (
Identifiants
pubmed: 30674563
pii: jgp.201812192
doi: 10.1085/jgp.201812192
pmc: PMC6363420
doi:
Substances chimiques
Anti-Arrhythmia Agents
0
ERG1 Potassium Channel
0
KCNH2 protein, human
0
Phenethylamines
0
Potassium Channel Blockers
0
Pyrimidinones
0
Sulfonamides
0
nifekalant
5VZ7GZM43E
dofetilide
R4Z9X1N2ND
Types de publication
Journal Article
Research Support, N.I.H., Extramural
Research Support, Non-U.S. Gov't
Langues
eng
Sous-ensembles de citation
IM
Pagination
214-230Subventions
Organisme : NHLBI NIH HHS
ID : R01 HL128537
Pays : United States
Organisme : NHLBI NIH HHS
ID : U01 HL126273
Pays : United States
Informations de copyright
© 2019 Furutani et al.
Références
Br J Pharmacol. 2008 Aug;154(7):1528-37
pubmed: 18552873
PLoS One. 2014 Jan 10;9(1):e84595
pubmed: 24427289
Circulation. 2001 Mar 20;103(11):1585-90
pubmed: 11257089
Arzneimittelforschung. 1988 Feb;38(2):231-6
pubmed: 3370070
Annu Rev Pharmacol Toxicol. 2003;43:441-61
pubmed: 12540747
Biophys J. 2000 May;78(5):2392-404
pubmed: 10777735
Circ Arrhythm Electrophysiol. 2011 Feb;4(1):103-11
pubmed: 21078812
Sci Rep. 2017 Sep 7;7(1):10771
pubmed: 28883639
Biochem Biophys Res Commun. 2011 Nov 11;415(1):141-6
pubmed: 22020101
J Cardiovasc Pharmacol. 2011 Jan;57(1):79-85
pubmed: 20980921
J Am Coll Cardiol. 1996 Jan;27(1):84-9
pubmed: 8522715
Circulation. 1990 Feb;81(2):686-90
pubmed: 2153477
Circulation. 2005 Sep 6;112(10):1392-9
pubmed: 16129791
Am Heart J. 2014 Mar;167(3):292-300
pubmed: 24576511
Conf Proc IEEE Eng Med Biol Soc. 2013;2013:5529-32
pubmed: 24110989
Eur J Pharmacol. 2010 Apr 25;632(1-3):52-9
pubmed: 20097192
Biophys J. 1998 Jan;74(1):230-41
pubmed: 9449325
Circulation. 1995 Sep 1;92(5):1179-87
pubmed: 7648663
Circulation. 1997 Nov 18;96(10):3696-703
pubmed: 9396473
Circulation. 1996 Jan 1;93(1):168-77
pubmed: 8616924
Jpn Circ J. 2001 Jan;65(1):60-2
pubmed: 11153825
Cardiovasc Res. 2011 Jul 1;91(1):53-61
pubmed: 21300721
Fed Regist. 2005 Oct 20;70(202):61133-4
pubmed: 16237859
J Pharmacol Exp Ther. 1999 Dec;291(3):1324-36
pubmed: 10565858
J Cardiovasc Pharmacol. 2004 May;43(5):715-23
pubmed: 15071360
Circ Res. 2009 Jan 2;104(1):79-86
pubmed: 19038865
J Cardiovasc Pharmacol. 1990 Sep;16(3):401-10
pubmed: 1700210
J Am Coll Cardiol. 1995 Jul;26(1):185-92
pubmed: 7797750
Indian Heart J. 2014 Nov-Dec;66(6):640-8
pubmed: 25634399
Channels (Austin). 2007 May-Jun;1(3):198-208
pubmed: 18690032
J Physiol. 2002 Sep 1;543(Pt 2):615-31
pubmed: 12205194
Pflugers Arch. 2005 Aug;450(5):307-16
pubmed: 15952036
Br J Pharmacol. 2001 Jan;132(1):85-92
pubmed: 11156564
Am J Physiol Heart Circ Physiol. 2004 Apr;286(4):H1573-89
pubmed: 14656705
J Cardiovasc Electrophysiol. 2000 Aug;11(8):938-40
pubmed: 10969760
Br J Pharmacol. 2008 Aug;154(7):1502-7
pubmed: 18552874
J Cardiovasc Pharmacol. 2002 Nov;40(5):735-42
pubmed: 12409982
Science. 1995 Jul 7;269(5220):92-5
pubmed: 7604285
Eur J Heart Fail. 2002 Mar;4(2):201-6
pubmed: 11959050
Cardiovasc Res. 2003 Apr 1;58(1):32-45
pubmed: 12667944
IEEE J Biomed Health Inform. 2015 Jul;19(4):1308-20
pubmed: 26068919
Heart Rhythm. 2010 Dec;7(12):1891-9
pubmed: 20868774
Cell. 1999 Apr 16;97(2):175-87
pubmed: 10219239
J Gen Physiol. 1990 Jul;96(1):195-215
pubmed: 2170562
Cardiovasc Res. 1996 Jun;31(6):963-74
pubmed: 8759253
J Clin Pharmacol. 1992 Nov;32(11):964-77
pubmed: 1474169
J Am Coll Cardiol. 2005 Jan 18;45(2):300-7
pubmed: 15653031
Pflugers Arch. 1981 Aug;391(2):85-100
pubmed: 6270629
J Mol Cell Cardiol. 2018 Dec;125:18-28
pubmed: 30321537
Physiol Rev. 2007 Apr;87(2):425-56
pubmed: 17429037
Eur J Clin Pharmacol. 2001 Jun;57(3):185-209
pubmed: 11497335
J Pharmacol Exp Ther. 2003 Nov;307(2):776-84
pubmed: 12966159
Sci Rep. 2017 Oct 4;7(1):12683
pubmed: 28978927
Circulation. 2010 Mar 2;121(8):1047-60
pubmed: 20142454
Biochem Biophys Res Commun. 2012 Feb 3;418(1):161-6
pubmed: 22244872
Heart Rhythm. 2010 Aug;7(8):1093-101
pubmed: 20382266
Nature. 2006 Mar 23;440(7083):463-9
pubmed: 16554806
Eur J Clin Pharmacol. 2015 May;71(5):549-67
pubmed: 25870032
PLoS Comput Biol. 2011 May;7(5):e1002061
pubmed: 21637795
Circ Res. 1995 Jul;77(1):140-52
pubmed: 7788872
J Am Coll Cardiol. 1989 Jul;14(1):172-84
pubmed: 2661626
Nat Rev Drug Discov. 2016 Jul;15(7):457-71
pubmed: 26893184
Am J Physiol Heart Circ Physiol. 2012 Apr 15;302(8):H1636-44
pubmed: 22307670
Br J Pharmacol. 1993 May;109(1):157-63
pubmed: 7684298
Br J Pharmacol. 2012 Jan;165(2):467-78
pubmed: 21718297
Biophys J. 1995 Mar;68(3):949-64
pubmed: 7538806
N Engl J Med. 1999 Sep 16;341(12):857-65
pubmed: 10486417
Circ Res. 1993 Jan;72(1):75-83
pubmed: 8417848
Am J Physiol Heart Circ Physiol. 2006 Sep;291(3):H1088-100
pubmed: 16565318
Sci Rep. 2013;3:2100
pubmed: 23812503
Biophys J. 2010 Aug 4;99(3):765-73
pubmed: 20682253
Cell. 1995 Apr 21;81(2):299-307
pubmed: 7736582
Circ Res. 1993 Nov;73(5):857-68
pubmed: 8403256