Intracellular Lipopolysaccharide Sensing as a Potential Therapeutic Target for Sepsis.


Journal

Trends in pharmacological sciences
ISSN: 1873-3735
Titre abrégé: Trends Pharmacol Sci
Pays: England
ID NLM: 7906158

Informations de publication

Date de publication:
03 2019
Historique:
received: 19 09 2018
revised: 20 12 2018
accepted: 07 01 2019
pubmed: 30 1 2019
medline: 7 3 2019
entrez: 30 1 2019
Statut: ppublish

Résumé

Lipopolysaccharide (LPS) sensing in the cytosol by the noncanonical inflammasome leads to pyroptosis and NLRP3 inflammasome activation. This mechanism may be more critical for sepsis development than recognition of LPS by Toll-like receptor 4. LPS is directly binding to its intracellular receptor caspase-4/5/11, mediated by outer membrane vesicles and guanylate-binding proteins that deliver LPS to the cytosol and mediate access of caspases to LPS. Caspase-11-dependent cleavage of gasdermin D is discussed as a link between LPS-induced activation of caspases and pyroptosis or NLRP3 inflammasome activation. Finally, we highlight recently described inhibitors of cytosolic LPS-triggered noncanonical inflammasome activation that might be considered as potential drugs for the treatment of sepsis.

Identifiants

pubmed: 30691865
pii: S0165-6147(19)30001-X
doi: 10.1016/j.tips.2019.01.001
pii:
doi:

Substances chimiques

GSDMD protein, human 0
Inflammasomes 0
Intracellular Signaling Peptides and Proteins 0
Lipopolysaccharides 0
Neoplasm Proteins 0
Phosphate-Binding Proteins 0
Caspases EC 3.4.22.-

Types de publication

Journal Article Review

Langues

eng

Sous-ensembles de citation

IM

Pagination

187-197

Informations de copyright

Copyright © 2019 Elsevier Ltd. All rights reserved.

Auteurs

Anja Pfalzgraff (A)

Institute of Pharmacy (Pharmacology and Toxicology), Freie Universität Berlin, Berlin, Germany.

Günther Weindl (G)

Institute of Pharmacy (Pharmacology and Toxicology), Freie Universität Berlin, Berlin, Germany; Pharmacology and Toxicology Section, Pharmaceutical Institute, University of Bonn, Bonn, Germany. Electronic address: guenther.weindl@fu-berlin.de.

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Classifications MeSH