ABC transporters Mdr1a/1b, Bcrp1, Mrp2 and Mrp3 determine the sensitivity to PhIP/DSS-induced colon carcinogenesis and inflammation.


Journal

Archives of toxicology
ISSN: 1432-0738
Titre abrégé: Arch Toxicol
Pays: Germany
ID NLM: 0417615

Informations de publication

Date de publication:
03 2019
Historique:
received: 10 10 2018
accepted: 10 01 2019
pubmed: 1 2 2019
medline: 19 5 2020
entrez: 1 2 2019
Statut: ppublish

Résumé

2-Amino-1-methyl-6-phenylimidazo[4,5-b]pyridine (PhIP) is an abundant dietary carcinogen, formed during high-temperature cooking of meat. In this study, we investigated whether clinically relevant ATP-binding cassette (ABC) efflux transporters can modulate PhIP-induced colorectal carcinogenesis in vivo using wild-type (WT), Bcrp1

Identifiants

pubmed: 30701287
doi: 10.1007/s00204-019-02394-w
pii: 10.1007/s00204-019-02394-w
doi:

Substances chimiques

ATP-Binding Cassette Transporters 0
Carcinogens 0
Imidazoles 0
Dextran Sulfate 9042-14-2
2-amino-1-methyl-6-phenylimidazo(4,5-b)pyridine 909C6UN66T

Types de publication

Journal Article Research Support, Non-U.S. Gov't

Langues

eng

Sous-ensembles de citation

IM

Pagination

775-790

Auteurs

S Durmus (S)

Division of Pharmacology, The Netherlands Cancer Institute, Plesmanlaan 121, 1066 CX, Amsterdam, The Netherlands.
Department of Medical Biochemistry, Faculty of Medicine, Istinye University, Istanbul, Turkey.

M van der Valk (M)

Department of Animal Pathology, The Netherlands Cancer Institute, Amsterdam, The Netherlands.

S F Teunissen (SF)

Department of Pharmacy and Pharmacology, The Netherlands Cancer Institute, Amsterdam, The Netherlands.

J Y Song (JY)

Department of Animal Pathology, The Netherlands Cancer Institute, Amsterdam, The Netherlands.

E Wagenaar (E)

Division of Pharmacology, The Netherlands Cancer Institute, Plesmanlaan 121, 1066 CX, Amsterdam, The Netherlands.

J H Beijnen (JH)

Department of Pharmacy and Pharmacology, The Netherlands Cancer Institute, Amsterdam, The Netherlands.
Department of Pharmaceutical Sciences, Utrecht University, Utrecht, The Netherlands.

A H Schinkel (AH)

Division of Pharmacology, The Netherlands Cancer Institute, Plesmanlaan 121, 1066 CX, Amsterdam, The Netherlands. a.schinkel@nki.nl.

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Classifications MeSH