Lipid-Lowering Agents.


Journal

Circulation research
ISSN: 1524-4571
Titre abrégé: Circ Res
Pays: United States
ID NLM: 0047103

Informations de publication

Date de publication:
02 2019
Historique:
entrez: 1 2 2019
pubmed: 1 2 2019
medline: 16 11 2019
Statut: ppublish

Résumé

Several new or emerging drugs for dyslipidemia owe their existence, in part, to human genetic evidence, such as observations in families with rare genetic disorders or in Mendelian randomization studies. Much effort has been directed to agents that reduce LDL (low-density lipoprotein) cholesterol, triglyceride, and Lp[a] (lipoprotein[a]), with some sustained programs on agents to raise HDL (high-density lipoprotein) cholesterol. Lomitapide, mipomersen, AAV8.TBG.hLDLR, inclisiran, bempedoic acid, and gemcabene primarily target LDL cholesterol. Alipogene tiparvovec, pradigastat, and volanesorsen primarily target elevated triglycerides, whereas evinacumab and IONIS-ANGPTL3-L

Identifiants

pubmed: 30702996
doi: 10.1161/CIRCRESAHA.118.313171
doi:

Substances chimiques

ALN-PCS 0
Antibodies, Monoclonal 0
Anticholesteremic Agents 0
BMS201038 0
Benzimidazoles 0
Caproates 0
Cholesterol, HDL 0
Cholesterol, LDL 0
Dicarboxylic Acids 0
Fatty Acids 0
Hypolipidemic Agents 0
ISIS 304801 0
Lipoprotein(a) 0
Oligonucleotides 0
RNA, Small Interfering 0
8-hydroxy-2,2,14,14-tetramethylpentadecanedioic acid 1EJ6Z6Q368
mipomersen 9GJ8S4GU0M
gemcabene B96UX1DDKS
Diacylglycerol O-Acyltransferase EC 2.3.1.20
Ezetimibe EOR26LQQ24
evinacumab T8B2ORP1DW

Types de publication

Journal Article Research Support, N.I.H., Extramural Research Support, Non-U.S. Gov't

Langues

eng

Sous-ensembles de citation

IM

Pagination

386-404

Subventions

Organisme : CIHR
Pays : Canada
Organisme : NHLBI NIH HHS
ID : P01 HL088093
Pays : United States
Organisme : NHLBI NIH HHS
ID : P01 HL055798
Pays : United States
Organisme : NHLBI NIH HHS
ID : R01 HL106579
Pays : United States
Organisme : NHLBI NIH HHS
ID : R01 HL078610
Pays : United States
Organisme : NHLBI NIH HHS
ID : R01 HL124174
Pays : United States

Commentaires et corrections

Type : ErratumIn

Auteurs

Robert A Hegele (RA)

From the Department of Medicine and Robarts Research Institute, Schulich School of Medicine and Dentistry, Western University, London, Ontario, Canada (R.A.H.).

Sotirios Tsimikas (S)

Sulpizio Cardiovascular Center, Vascular Medicine Program, University of California San Diego, La Jolla (S.T.).

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Classifications MeSH