Diagnoses of Pathological States Based on Acetylcholinesterase and Butyrylcholinesterase.

Acetylcholinesterase anesthesia butyrylcholinesterase diagnosis liver function test myorelaxant nerve agent neurotransmission pesticide poisoning.

Journal

Current medicinal chemistry
ISSN: 1875-533X
Titre abrégé: Curr Med Chem
Pays: United Arab Emirates
ID NLM: 9440157

Informations de publication

Date de publication:
2020
Historique:
received: 01 07 2018
revised: 16 01 2019
accepted: 17 01 2019
pubmed: 2 2 2019
medline: 6 8 2020
entrez: 2 2 2019
Statut: ppublish

Résumé

Two cholinesterases exist: Acetylcholinesterase (AChE) and butyrylcholinesterase (BChE). While AChE plays a crucial role in neurotransmissions, BChE has no specific function apart from the detoxification of some drugs and secondary metabolites from plants. Thus, both AChE and BChE can serve as biochemical markers of various pathologies. Poisoning by nerve agents like sarin, soman, tabun, VX, novichok and overdosing by drugs used in some neurodegenerative disorders like Alzheimer´s disease and myasthenia gravis, as well as poisoning by organophosphorus pesticides are relevant to this issue. But it appears that changes in these enzymes take place in other processes including oxidative stress, inflammation, some types of cancer and genetically conditioned diseases. In this review, the cholinesterases are introduced, the mechanism of inhibitors action is explained and the relations between the cholinesterases and pathologies are explained.

Identifiants

pubmed: 30706778
pii: CMC-EPUB-96228
doi: 10.2174/0929867326666190130161202
doi:

Substances chimiques

Cholinesterase Inhibitors 0
Pesticides 0
Acetylcholinesterase EC 3.1.1.7
Butyrylcholinesterase EC 3.1.1.8

Types de publication

Journal Article Review

Langues

eng

Sous-ensembles de citation

IM

Pagination

2994-3011

Informations de copyright

Copyright© Bentham Science Publishers; For any queries, please email at epub@benthamscience.net.

Auteurs

Miroslav Pohanka (M)

Faculty of Military Health Sciences, University of Defence, Trebesska 1575, 50001 Hradec Kralove, Czech Republic.

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Classifications MeSH