Modes of Accessing Bicarbonate for the Regulation of Membrane Guanylate Cyclase (ROS-GC) in Retinal Rods and Cones.
Acetazolamide
/ pharmacology
Ambystoma
Animals
Bicarbonates
/ metabolism
COS Cells
Carbon Dioxide
/ metabolism
Carbonic Anhydrase Inhibitors
/ pharmacology
Carbonic Anhydrases
/ genetics
Cattle
Cell Membrane
/ drug effects
Chlorocebus aethiops
Cyclic GMP
/ metabolism
Gene Expression
Guanylate Cyclase
/ genetics
Mice
Receptors, Cell Surface
/ metabolism
Recombinant Proteins
/ metabolism
Retinal Cone Photoreceptor Cells
/ cytology
Retinal Rod Photoreceptor Cells
/ cytology
Tissue Culture Techniques
Vision, Ocular
/ drug effects
bicarbonate
cone
receptor guanylate cyclase
retina
rod
visual transduction
Journal
eNeuro
ISSN: 2373-2822
Titre abrégé: eNeuro
Pays: United States
ID NLM: 101647362
Informations de publication
Date de publication:
Historique:
received:
11
10
2018
revised:
20
12
2018
accepted:
15
01
2019
entrez:
21
2
2019
pubmed:
21
2
2019
medline:
19
4
2019
Statut:
epublish
Résumé
The membrane guanylate cyclase, ROS-GC, that synthesizes cyclic GMP for use as a second messenger for visual transduction in retinal rods and cones, is stimulated by bicarbonate. Bicarbonate acts directly on ROS-GC1, because it enhanced the enzymatic activity of a purified, recombinant fragment of bovine ROS-GC1 consisting solely of the core catalytic domain. Moreover, recombinant ROS-GC1 proved to be a true sensor of bicarbonate, rather than a sensor for CO
Identifiants
pubmed: 30783616
doi: 10.1523/ENEURO.0393-18.2019
pii: eN-NWR-0393-18
pmc: PMC6378327
pii:
doi:
Substances chimiques
Bicarbonates
0
Carbonic Anhydrase Inhibitors
0
Receptors, Cell Surface
0
Recombinant Proteins
0
Carbon Dioxide
142M471B3J
Carbonic Anhydrases
EC 4.2.1.1
Guanylate Cyclase
EC 4.6.1.2
Cyclic GMP
H2D2X058MU
Acetazolamide
O3FX965V0I
Types de publication
Journal Article
Research Support, N.I.H., Extramural
Langues
eng
Sous-ensembles de citation
IM
Subventions
Organisme : NEI NIH HHS
ID : R01 EY023980
Pays : United States
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