Combined Activation of Guanylate Cyclase and Cyclic AMP in Lung Fibroblasts as a Novel Therapeutic Concept for Lung Fibrosis.
Cell Proliferation
/ drug effects
Cell Survival
/ drug effects
Colforsin
/ pharmacology
Collagen Type I
/ metabolism
Collagen Type III
/ metabolism
Cyclic AMP
/ genetics
Fibroblasts
/ drug effects
Fibronectins
/ metabolism
Gene Expression Regulation
/ drug effects
Guanylate Cyclase
/ genetics
Humans
Idiopathic Pulmonary Fibrosis
/ drug therapy
Lung
/ drug effects
Primary Cell Culture
Pyrazoles
/ pharmacology
Pyridines
/ pharmacology
Signal Transduction
/ drug effects
Transforming Growth Factor beta
/ genetics
beta Catenin
/ genetics
Journal
BioMed research international
ISSN: 2314-6141
Titre abrégé: Biomed Res Int
Pays: United States
ID NLM: 101600173
Informations de publication
Date de publication:
2019
2019
Historique:
received:
15
08
2018
revised:
19
12
2018
accepted:
28
01
2019
entrez:
16
4
2019
pubmed:
16
4
2019
medline:
17
8
2019
Statut:
epublish
Résumé
Remodelling of the peripheral lung tissue and fibrotic foci are the main pathologies of idiopathic pulmonary fibrosis (IPF), a disease that is difficult to treat. TGF-
Identifiants
pubmed: 30984775
doi: 10.1155/2019/1345402
pmc: PMC6431482
doi:
Substances chimiques
3-(4-Amino-5-cyclopropylpyrimidine-2-yl)-1-(2-fluorobenzyl)-1H-pyrazolo(3,4-b)pyridine
0
Collagen Type I
0
Collagen Type III
0
Fibronectins
0
Pyrazoles
0
Pyridines
0
Transforming Growth Factor beta
0
beta Catenin
0
Colforsin
1F7A44V6OU
Cyclic AMP
E0399OZS9N
Guanylate Cyclase
EC 4.6.1.2
Types de publication
Journal Article
Langues
eng
Pagination
1345402Références
Am J Respir Crit Care Med. 2001 Jan;163(1):210-7
pubmed: 11208648
Thorax. 2001 Dec;56(12):907-15
pubmed: 11713352
Br J Pharmacol. 2002 Jan;135(2):344-55
pubmed: 11815369
Am J Physiol Lung Cell Mol Physiol. 2003 Sep;285(3):L527-39
pubmed: 12598227
J Cell Physiol. 2005 Jul;204(1):146-54
pubmed: 15672417
Biol Neonate. 2006;90(2):135-44
pubmed: 16582538
J Cardiovasc Pharmacol. 2009 Feb;53(2):121-31
pubmed: 19188837
Hypertens Res. 2009 Jul;32(7):597-603
pubmed: 19424280
Ther Adv Respir Dis. 2010 Dec;4(6):367-88
pubmed: 20952439
Am J Respir Crit Care Med. 2011 Mar 15;183(6):788-824
pubmed: 21471066
J Pharmacol Exp Ther. 2011 Nov;339(2):394-402
pubmed: 21825001
J Biol Chem. 2012 Mar 2;287(10):7026-38
pubmed: 22241478
Ann Rheum Dis. 2012 Jun;71(6):1019-26
pubmed: 22294631
Int J Clin Exp Pathol. 2012;5(1):58-71
pubmed: 22295148
Eur Respir Rev. 2012 Jun 1;21(124):141-6
pubmed: 22654086
Proc Am Thorac Soc. 2012 Jul;9(3):130-6
pubmed: 22802287
Int Wound J. 2015 Jun;12(3):313-6
pubmed: 23742140
J Cell Physiol. 2014 Feb;229(2):213-24
pubmed: 23881674
Pharmacol Res. 2013 Oct;76:182-9
pubmed: 23994158
Ann Rheum Dis. 2015 Jul;74(7):1408-16
pubmed: 24567525
Eur J Pharm Sci. 2014 Jul 16;58:13-9
pubmed: 24613900
PLoS One. 2014 Apr 11;9(4):e94616
pubmed: 24728102
N Engl J Med. 2014 May 29;370(22):2083-92
pubmed: 24836312
Mol Med Rep. 2014 Aug;10(2):1030-6
pubmed: 24859686
Biochem Pharmacol. 2014 Oct 1;91(3):400-8
pubmed: 25107701
Mol Med Rep. 2015 Apr;11(4):2703-10
pubmed: 25435076
Eur Respir J. 2015 Sep;46(3):795-806
pubmed: 25976683
Am J Respir Cell Mol Biol. 2016 Jan;54(1):51-9
pubmed: 26072676
Pharmacol Res. 2015 Dec;102:310-8
pubmed: 26546746
Am J Physiol Lung Cell Mol Physiol. 2016 Apr 1;310(7):L615-29
pubmed: 26773067
J Cell Mol Med. 2017 Aug;21(8):1545-1554
pubmed: 28244647
Am J Respir Cell Mol Biol. 2017 Jul;57(1):77-90
pubmed: 28257580
Expert Rev Respir Med. 2017 Apr;11(4):299-309
pubmed: 28274188
Mediators Inflamm. 2017;2017:3520581
pubmed: 28588349
J Cell Physiol. 2018 Mar;233(3):2513-2525
pubmed: 28771711
PLoS One. 2017 Sep 5;12(9):e0183972
pubmed: 28873461
Nat Rev Drug Discov. 2017 Nov;16(11):755-772
pubmed: 28983101
Mol Biol Cell. 2017 Dec 15;28(26):3741-3755
pubmed: 29046395
Toxicol Lett. 2018 Mar 1;284:1-9
pubmed: 29195901
Sci Rep. 2018 Jan 18;8(1):1087
pubmed: 29348469
Pharmacol Ther. 2018 Jul;187:150-166
pubmed: 29458107
Respirology. 2018 Aug;23(8):756-763
pubmed: 29532550
Respir Res. 2018 Apr 7;19(1):56
pubmed: 29625570
BMC Pulm Med. 2018 Apr 27;18(1):63
pubmed: 29703175