α,γ-Diketocarboxylic Acids and Their Esters Act as Carbonic Anhydrase IX and XII Selective Inhibitors.
Journal
ACS medicinal chemistry letters
ISSN: 1948-5875
Titre abrégé: ACS Med Chem Lett
Pays: United States
ID NLM: 101521073
Informations de publication
Date de publication:
11 Apr 2019
11 Apr 2019
Historique:
received:
21
01
2019
accepted:
19
02
2019
entrez:
19
4
2019
pubmed:
19
4
2019
medline:
19
4
2019
Statut:
epublish
Résumé
Among human carbonic anhydrase (CA) inhibitors, the α,γ-diketocarboxylic acids and esters are still poorly investigated. Here, we report the first compounds of this class (
Identifiants
pubmed: 30996814
doi: 10.1021/acsmedchemlett.9b00023
pmc: PMC6466837
doi:
Types de publication
Journal Article
Langues
eng
Pagination
661-665Déclaration de conflit d'intérêts
The authors declare no competing financial interest.
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