Carfilzomib Weekly plus Melphalan and Prednisone in Newly Diagnosed Transplant-Ineligible Multiple Myeloma (IFM 2012-03): A Phase I Trial.


Journal

Clinical cancer research : an official journal of the American Association for Cancer Research
ISSN: 1557-3265
Titre abrégé: Clin Cancer Res
Pays: United States
ID NLM: 9502500

Informations de publication

Date de publication:
15 07 2019
Historique:
received: 06 11 2018
revised: 18 01 2019
accepted: 29 04 2019
pubmed: 6 5 2019
medline: 23 9 2020
entrez: 5 5 2019
Statut: ppublish

Résumé

Carfilzomib is a novel generation proteasome inhibitor. The Carmysap trial demonstrated that twice-weekly KMP (carfilzomib, melphalan, prednisone) might challenge the MPV (melphalan, prednisone, bortezomib) standard. We sought to study KMP weekly, allowing to increase carfilzomib's dose with maintained efficacy and improved safety profile. IFM2012-03, a phase I multicenter study of KMP weekly in elderly patients with newly diagnosed multiple myeloma (eNDMM), aimed to determine the MTD of carfilzomib. Carfilzomib was given intravenously at 36, 45, 56, and 70 mg/m Thirty eNDMMs were treated, 6 per cohort at 36, 45, and 56 mg/m The MTD dose of carfilzomib was 70 mg/m

Identifiants

pubmed: 31053600
pii: 1078-0432.CCR-18-3642
doi: 10.1158/1078-0432.CCR-18-3642
doi:

Substances chimiques

Oligopeptides 0
carfilzomib 72X6E3J5AR
Melphalan Q41OR9510P
Prednisone VB0R961HZT

Types de publication

Clinical Trial, Phase I Journal Article Multicenter Study Research Support, Non-U.S. Gov't

Langues

eng

Sous-ensembles de citation

IM

Pagination

4224-4230

Informations de copyright

©2019 American Association for Cancer Research.

Auteurs

Xavier Leleu (X)

Hematology and Inserm CIC 1402, CHU Poitiers, France. xavier.leleu@chu-poitiers.fr.

Guillemette Fouquet (G)

Institut Imagine, Inserm U1163 - CNRS ERL8254, Hôpital Necker, Paris, France.

Stéphanie Guidez (S)

Hematology and Inserm CIC 1402, CHU Poitiers, France.

Alain Duhamel (A)

Université de Lille, CHRU Lille, EA 2694 - Santé publique: épidémiologie et qualité des soins, Lille, France.

François Machuron (F)

Université de Lille, CHRU Lille, EA 2694 - Santé publique: épidémiologie et qualité des soins, Lille, France.

Lionel Karlin (L)

CHU Lyon Sud, France.

Brigitte Kolb (B)

CHU Reims, France.

Mourad Tiab (M)

CH la Roche Sur Yon, France.

Carla Araujo (C)

CH Bayonne, France.

Nathalie Meuleman (N)

Institut Bordet, Bruxelles, Belgium.

Jean-Valère Malfuson (JV)

CH Clamart, France.

Pascal Bourquard (P)

CHU Nîmes, France.

Pascal Lenain (P)

Centre Henri Becquerel, Rouen, France.

Murielle Roussel (M)

Cancer Research Center, Toulouse, France.

Arnaud Jaccard (A)

CHU Limoges, France.

Marie-Odile Pétillon (MO)

CHRU Lille, France.

Karim Belhadj-Merzoug (K)

CHU Henri Mondor, Créteil, France.

Gérard Lepeu (G)

CH Avignon, France.

Jean Fontan (J)

CHU Besançon, France.

Philippe Rodon (P)

CH Périgueux, France.

Anna Schmitt (A)

Institut Bergonie, Bordeaux, France.

Fritz Offner (F)

Universitair Ziekenhuis Gent, Belgium.

Laurent Voillat (L)

CH Chalon-sur-Saône, France.

Sophie Cereja (S)

CH Corbeil-Essonnes, France.

Frédérique Kuhnowski (F)

Institut Curie, Paris, France.

Sophie Rigaudeau (S)

CHU Versailles, France.

Olivier Decaux (O)

CHU de Rennes, France.

Jamile Frayfer (J)

CH Meaux, France.

Olivier Fitoussi (O)

Polyclinique Bordeaux Nord, France.

Damien Roos-Weil (D)

AP-HP Groupe Hospitalier Pitié-Salpêtrière, Paris, France.

Jean-Claude Eisenmann (JC)

CH Mulhouse, France.

Véronique Dorvaux (V)

CH Metz-Thionville, France.

Eric G Voog (EG)

Centre Jean Bernard, Le Mans, France.

Michel Attal (M)

Cancer Research Center, Toulouse, France.

Philippe Moreau (P)

CHU Nantes, France.

Hervé Avet-Loiseau (H)

Cancer Research Center, Toulouse, France.

Cyrille Hulin (C)

CHU Bordeaux, France.

Thierry Facon (T)

CHRU Lille, France.

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Classifications MeSH