Davis-Beirut Reaction: Diverse Chemistries of Highly Reactive Nitroso Intermediates in Heterocycle Synthesis.


Journal

Accounts of chemical research
ISSN: 1520-4898
Titre abrégé: Acc Chem Res
Pays: United States
ID NLM: 0157313

Informations de publication

Date de publication:
20 08 2019
Historique:
pubmed: 23 7 2019
medline: 7 8 2020
entrez: 23 7 2019
Statut: ppublish

Résumé

Indazoles are an important class of nitrogen heterocycles because of their excellent performance in biologically relevant applications, such as in chemical biology and medicinal chemistry. In these applications, convenient synthesis using commercially available and diverse building blocks is highly desirable. Within this broad class, 2

Identifiants

pubmed: 31328502
doi: 10.1021/acs.accounts.9b00220
pmc: PMC6702092
mid: NIHMS1044831
doi:

Substances chimiques

Amines 0
Indazoles 0
Nitroso Compounds 0

Types de publication

Journal Article Research Support, N.I.H., Extramural Research Support, Non-U.S. Gov't Review

Langues

eng

Sous-ensembles de citation

IM

Pagination

2256-2265

Subventions

Organisme : NIDDK NIH HHS
ID : P30 DK072517
Pays : United States
Organisme : NIDDK NIH HHS
ID : R01 DK067003
Pays : United States

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Auteurs

Jie S Zhu (JS)

Department of Chemistry , University of California Davis , 1 Shields Avenue , Davis California 95616 , United States.

Makhluf J Haddadin (MJ)

Department of Chemistry , American University of Beirut , Beirut , Lebanon.

Mark J Kurth (MJ)

Department of Chemistry , University of California Davis , 1 Shields Avenue , Davis California 95616 , United States.

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