Mitophagy protects against statin-mediated skeletal muscle toxicity.


Journal

FASEB journal : official publication of the Federation of American Societies for Experimental Biology
ISSN: 1530-6860
Titre abrégé: FASEB J
Pays: United States
ID NLM: 8804484

Informations de publication

Date de publication:
11 2019
Historique:
pubmed: 1 8 2019
medline: 9 6 2020
entrez: 1 8 2019
Statut: ppublish

Résumé

The deleterious effects of statins on skeletal muscle are well known, but the mechanism associated with these effects remains unresolved. Statins are associated with mitochondrial damage, which may contribute to muscle myopathy. Here we demonstrate that simvastatin induces mitophagy in skeletal muscle cells and hypothesized that attenuating this process by silencing the mitophagy adapter p62/sequestosome-1 (SQSTM1) might mitigate myotoxicity. Surprisingly, silencing p62/SQSTM1 in differentiated C2C12 muscle cells exacerbated rather than attenuated myotoxicity. This inhibition of mitophagy in the face of statin challenge correlated with increased release of cytochrome

Identifiants

pubmed: 31365836
doi: 10.1096/fj.201900807RR
pmc: PMC6902735
doi:

Substances chimiques

Hydroxymethylglutaryl-CoA Reductase Inhibitors 0
Sequestosome-1 Protein 0
Sqstm1 protein, mouse 0
Cytochromes c 9007-43-6
Simvastatin AGG2FN16EV
L-Lactate Dehydrogenase EC 1.1.1.27
Ubiquitin-Protein Ligases EC 2.3.2.27
parkin protein EC 2.3.2.27
Caspase 3 EC 3.4.22.-

Types de publication

Journal Article Research Support, Non-U.S. Gov't

Langues

eng

Sous-ensembles de citation

IM

Pagination

11857-11869

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Auteurs

Mridula Ramesh (M)

Donald P. Shiley BioScience Center, San Diego State University, San Diego, California, USA.

Juliane C Campos (JC)

Cedars-Sinai Medical Center, Los Angeles, California, USA.
Institute of Biomedical Sciences, University of Sao Paulo, Sao Paulo, Brazil.

Pamela Lee (P)

Donald P. Shiley BioScience Center, San Diego State University, San Diego, California, USA.

Yang Song (Y)

Cedars-Sinai Medical Center, Los Angeles, California, USA.

Genaro Hernandez (G)

Donald P. Shiley BioScience Center, San Diego State University, San Diego, California, USA.

Jon Sin (J)

Cedars-Sinai Medical Center, Los Angeles, California, USA.

Kyle C Tucker (KC)

Cedars-Sinai Medical Center, Los Angeles, California, USA.

Hannaneh Saadaeijahromi (H)

Cedars-Sinai Medical Center, Los Angeles, California, USA.

Michael Gurney (M)

Donald P. Shiley BioScience Center, San Diego State University, San Diego, California, USA.

Julio C B Ferreira (JCB)

Institute of Biomedical Sciences, University of Sao Paulo, Sao Paulo, Brazil.

Allen M Andres (AM)

Cedars-Sinai Medical Center, Los Angeles, California, USA.

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Classifications MeSH