Contalactone, a contaminant formed during chemical synthesis of the strigolactone reference GR24 is also a strigolactone mimic.

Arabidopsis thaliana Medicago truncatula Pisum sativum Plant hormone Rhizophagus irregularis Root parasitic plants Strigolactone mimics Structural determination α/β-hydrolase

Journal

Phytochemistry
ISSN: 1873-3700
Titre abrégé: Phytochemistry
Pays: England
ID NLM: 0151434

Informations de publication

Date de publication:
Dec 2019
Historique:
received: 12 06 2019
revised: 28 08 2019
accepted: 28 08 2019
pubmed: 10 9 2019
medline: 18 12 2019
entrez: 10 9 2019
Statut: ppublish

Résumé

Strigolactone (SL) plant hormones control plant architecture and are key players in both symbiotic and parasitic interactions. GR24, a synthetic SL analog, is the worldwide reference compound used in all bioassays for investigating the role of SLs in plant development and in rhizospheric interactions. In 2012, the first characterization of the SL receptor reported the detection of an unknown compound after incubation of GR24 samples with the SL receptor. We reveal here the origin of this compound (P270), which comes from a by-product formed during GR24 chemical synthesis. We present the identification of this by-product, named contalactone. A proposed chemical pathway for its formation is provided as well as an evaluation of its bioactivity on pea, Arabidopsis, root parasitic plant seeds and AM fungi, characterizing it as a SL mimic. Quality of GR24 samples can be easily checked by carrying out microscale hydrolysis in a basic aqueous medium to easily detect P270 as indicator of the presence of the contalactone impurity. In all cases, before being used for bioassays, GR24 must be careful purified by preparative HPLC.

Identifiants

pubmed: 31499274
pii: S0031-9422(19)30548-5
doi: 10.1016/j.phytochem.2019.112112
pii:
doi:

Substances chimiques

GR24 strigolactone 0
Heterocyclic Compounds, 3-Ring 0
Lactones 0

Types de publication

Journal Article

Langues

eng

Sous-ensembles de citation

IM

Pagination

112112

Informations de copyright

Copyright © 2019 Elsevier Ltd. All rights reserved.

Auteurs

Alexandre de Saint Germain (A)

Institut Jean-Pierre Bourgin, INRA, AgroParisTech, CNRS, Université Paris-Saclay, 78000, Versailles, France. Electronic address: Alexandre.De-Saint-Germain@inra.fr.

Pascal Retailleau (P)

Institut de Chimie des Substances Naturelles, CNRS UPR2301, Univ. Paris-Sud, Université Paris-Saclay, 1 Av. de la Terrasse, F-91198, Gif-sur-Yvette, France. Electronic address: Pascal.RETAILLEAU@cnrs.fr.

Stéphanie Norsikian (S)

Institut de Chimie des Substances Naturelles, CNRS UPR2301, Univ. Paris-Sud, Université Paris-Saclay, 1 Av. de la Terrasse, F-91198, Gif-sur-Yvette, France. Electronic address: Stephanie.NORSIKIAN@cnrs.fr.

Vincent Servajean (V)

Institut de Chimie des Substances Naturelles, CNRS UPR2301, Univ. Paris-Sud, Université Paris-Saclay, 1 Av. de la Terrasse, F-91198, Gif-sur-Yvette, France. Electronic address: Vincent.SERVAJEAN@cnrs.fr.

Franck Pelissier (F)

Institut de Chimie des Substances Naturelles, CNRS UPR2301, Univ. Paris-Sud, Université Paris-Saclay, 1 Av. de la Terrasse, F-91198, Gif-sur-Yvette, France. Electronic address: Franck.PELISSIER@cnrs.fr.

Vincent Steinmetz (V)

Institut de Chimie des Substances Naturelles, CNRS UPR2301, Univ. Paris-Sud, Université Paris-Saclay, 1 Av. de la Terrasse, F-91198, Gif-sur-Yvette, France. Electronic address: Vincent.STEINMETZ@cnrs.fr.

Jean-Paul Pillot (JP)

Institut Jean-Pierre Bourgin, INRA, AgroParisTech, CNRS, Université Paris-Saclay, 78000, Versailles, France. Electronic address: jean-paul.pillot@inra.fr.

Soizic Rochange (S)

Laboratoire de Recherche en Sciences Végétales, Université de Toulouse, CNRS, UPS, 24 Chemin de Borde Rouge, Auzeville, BP42617, 31326, Castanet Tolosan, France. Electronic address: rochange@lrsv.ups-tlse.fr.

Jean-Bernard Pouvreau (JB)

Université de Nantes, Laboratoire de Biologie et Pathologie Végétales, LBPV, EA 1157, F-44000, Nantes, France. Electronic address: Jean-Bernard.Pouvreau@univ-nantes.fr.

François-Didier Boyer (FD)

Institut Jean-Pierre Bourgin, INRA, AgroParisTech, CNRS, Université Paris-Saclay, 78000, Versailles, France; Institut de Chimie des Substances Naturelles, CNRS UPR2301, Univ. Paris-Sud, Université Paris-Saclay, 1 Av. de la Terrasse, F-91198, Gif-sur-Yvette, France. Electronic address: francois-didier.boyer@cnrs.fr.

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Classifications MeSH