Immunometabolic modulation of retinal inflammation by CD36 ligand.


Journal

Scientific reports
ISSN: 2045-2322
Titre abrégé: Sci Rep
Pays: England
ID NLM: 101563288

Informations de publication

Date de publication:
09 09 2019
Historique:
received: 29 11 2018
accepted: 20 08 2019
entrez: 11 9 2019
pubmed: 11 9 2019
medline: 28 10 2020
Statut: epublish

Résumé

In subretinal inflammation, activated mononuclear phagocytes (MP) play a key role in the progression of retinopathies. Little is known about the mechanism involved in the loss of photoreceptors leading to vision impairment. Studying retinal damage induced by photo-oxidative stress, we observed that cluster of differentiation 36 (CD36)-deficient mice featured less subretinal MP accumulation and attenuated photoreceptor degeneration. Moreover, treatment with a CD36-selective azapeptide ligand (MPE-001) reduced subretinal activated MP accumulation in wild type mice and preserved photoreceptor layers and function as assessed by electroretinography in a CD36-dependent manner. The azapeptide modulated the transcriptome of subretinal activated MP by reducing pro-inflammatory markers. In isolated MP, MPE-001 induced dissociation of the CD36-Toll-like receptor 2 (TLR2) oligomeric complex, decreasing nuclear factor-kappa B (NF-κB) and NLR family pyrin domain containing 3 (NLRP3) inflammasome activation. In addition, MPE-001 caused an aerobic metabolic shift in activated MP, involving peroxisome proliferator-activated receptor-γ (PPAR-γ) activation, which in turn mitigated inflammation. Accordingly, PPAR-γ inhibition blocked the cytoprotective effect of MPE-001 on photoreceptor apoptosis elicited by activated MP. By altering activated MP metabolism, MPE-001 decreased immune responses to alleviate subsequent inflammation-dependent neuronal injury characteristic of various vision-threatening retinal disorders.

Identifiants

pubmed: 31501473
doi: 10.1038/s41598-019-49472-8
pii: 10.1038/s41598-019-49472-8
pmc: PMC6733801
doi:

Substances chimiques

Biomarkers 0
CD36 Antigens 0
Cytokines 0
Inflammasomes 0
Inflammation Mediators 0
Ligands 0
NLR Family, Pyrin Domain-Containing 3 Protein 0
Toll-Like Receptor 2 0

Types de publication

Journal Article Research Support, Non-U.S. Gov't

Langues

eng

Sous-ensembles de citation

IM

Pagination

12903

Subventions

Organisme : CIHR
ID : PPP-90157
Pays : Canada

Références

Infect Immun. 2004 Sep;72(9):5041-51
pubmed: 15321997
Nature. 2005 Feb 3;433(7025):523-7
pubmed: 15690042
J Nutr Biochem. 2016 May;31:137-49
pubmed: 27133433
Angew Chem Int Ed Engl. 2017 May 22;56(22):6284-6288
pubmed: 28090719
J Cell Sci. 2012 May 15;125(Pt 10):2407-15
pubmed: 22357958
Nucleic Acids Res. 2009 Jul;37(Web Server issue):W652-60
pubmed: 19429898
PLoS One. 2011;6(12):e29092
pubmed: 22216174
Prog Retin Eye Res. 2015 Mar;45:30-57
pubmed: 25476242
Am J Pathol. 2017 Oct;187(10):2208-2221
pubmed: 28739342
Circulation. 2003 Feb 25;107(7):1009-16
pubmed: 12600915
Cell Microbiol. 2009 Aug;11(8):1160-9
pubmed: 19388903
Int J Inflam. 2013;2013:503725
pubmed: 23533946
Sci Rep. 2016 Mar 15;6:23132
pubmed: 26976286
J Immunol. 2011 Dec 1;187(11):6043-51
pubmed: 22021612
Science. 2003 Jun 6;300(5625):1524-5
pubmed: 12791976
Mediators Inflamm. 2015;2015:690243
pubmed: 25698849
J Leukoc Biol. 2013 Nov;94(5):885-902
pubmed: 23990624
Prog Retin Eye Res. 2010 Mar;29(2):95-112
pubmed: 19961953
PLoS One. 2009 Oct 22;4(10):e7411
pubmed: 19847289
Prog Retin Eye Res. 2009 Sep;28(5):348-68
pubmed: 19560552
J Immunol. 2003 Nov 15;171(10):5272-6
pubmed: 14607928
J Neuroinflammation. 2015 Nov 17;12:209
pubmed: 26576678
F1000Prime Rep. 2014 Mar 03;6:13
pubmed: 24669294
Nature. 2013 Apr 11;496(7444):238-42
pubmed: 23535595
Front Physiol. 2017 Jul 19;8:508
pubmed: 28769820
Front Biosci. 2001 Oct 01;6:E72-92
pubmed: 11578954
EMBO Mol Med. 2015 Jan 20;7(2):211-26
pubmed: 25604058
Biochem J. 2015 May 1;467(3):517-27
pubmed: 25742174
J Clin Invest. 2007 Oct;117(10):2920-8
pubmed: 17909628
Invest Ophthalmol Vis Sci. 2011 Jul 29;52(8):5824-35
pubmed: 21666244
Proc Natl Acad Sci U S A. 2000 Dec 5;97(25):13766-71
pubmed: 11095740
Circ Res. 2004 Sep 17;95(6):568-78
pubmed: 15375023
Nat Rev Nephrol. 2017 Dec;13(12):769-781
pubmed: 28919632
Diabetes. 2014 Nov;63(11):3926-37
pubmed: 24947354
Nat Med. 2018 Mar;24(3):360-367
pubmed: 29377004
Nat Immunol. 2010 May;11(5):373-84
pubmed: 20404851
Infect Immun. 2004 Mar;72(3):1657-65
pubmed: 14977973
Oncotarget. 2016 Nov 22;7(47):76984-76994
pubmed: 27769068
Cardiovasc Res. 2009 Aug 1;83(3):457-64
pubmed: 19377069
Trends Immunol. 2004 Dec;25(12):677-86
pubmed: 15530839
Cell Metab. 2006 Jul;4(1):13-24
pubmed: 16814729
Mol Vis. 2005 Oct 27;11:887-95
pubmed: 16270028
Stroke. 2010 May;41(5):898-904
pubmed: 20360550
Free Radic Biol Med. 2011 Jan 1;50(1):27-36
pubmed: 20974251
Invest Ophthalmol Vis Sci. 2004 Mar;45(3):971-6
pubmed: 14985319
Annu Rev Immunol. 2006;24:353-89
pubmed: 16551253
Nat Rev Immunol. 2011 Oct 25;11(11):788-98
pubmed: 22025056
J Biol Chem. 1999 Jun 18;274(25):17406-9
pubmed: 10364168
Prog Retin Eye Res. 2017 Nov;61:98-128
pubmed: 28602950
J Biol Chem. 2012 Jul 6;287(28):23479-88
pubmed: 22613713
Exp Eye Res. 2003 Apr;76(4):463-71
pubmed: 12634111
Circ Res. 2011 Mar 4;108(5):544-54
pubmed: 21252155
Am J Pathol. 2009 Jun;174(6):2310-23
pubmed: 19435787
Nucleic Acids Res. 2018 Jul 2;46(W1):W486-W494
pubmed: 29762782
J Nat Sci. 2017 Jan;3(1):
pubmed: 28191500
Int Immunol. 2014 Oct;26(10):563-73
pubmed: 24860120
Eur J Biochem. 2000 Oct;267(19):6050-9
pubmed: 10998066
J Immunol. 2000 Jun 15;164(12):6166-73
pubmed: 10843666
Sci Rep. 2015 Sep 28;5:14488
pubmed: 26412089
Nat Immunol. 2013 Aug;14(8):812-20
pubmed: 23812099
Immunol Rev. 2017 Nov;280(1):102-111
pubmed: 29027220
Am J Pathol. 2002 Jan;160(1):101-12
pubmed: 11786404
J Clin Invest. 2009 Jan;119(1):136-45
pubmed: 19065049
Oncogene. 2008 Jan 7;27(2):168-80
pubmed: 18176598
Blood. 1996 Mar 1;87(5):2020-8
pubmed: 8634453
J Neurosci. 2015 May 6;35(18):6987-96
pubmed: 25948251
Biochem J. 2004 Sep 1;382(Pt 2):417-24
pubmed: 15176951
J Investig Med. 2008 Feb;56(2):522-7
pubmed: 18317435
J Biol Chem. 1999 Jul 2;274(27):19055-62
pubmed: 10383407
J Biol Chem. 2006 Oct 13;281(41):31002-11
pubmed: 16880211
Nat Rev Drug Discov. 2010 Apr;9(4):293-307
pubmed: 20380038
Ophthalmic Res. 1996;28(2):99-107
pubmed: 8792360
Neurobiol Aging. 2012 Aug;33(8):1769-76
pubmed: 21570740
EMBO Mol Med. 2013 Nov;5(11):1775-93
pubmed: 24142887
Int J Inflam. 2013;2013:724648
pubmed: 24109539
Mol Immunol. 2015 Feb;63(2):143-52
pubmed: 24951397
Elife. 2016 Jul 20;5:
pubmed: 27438413
J Biol Chem. 2011 Nov 18;286(46):40013-24
pubmed: 21917928
Invest Ophthalmol Vis Sci. 2001 Dec;42(13):3301-10
pubmed: 11726637
Cell Immunol. 2009;258(2):138-46
pubmed: 19423085
Cell Metab. 2010 Nov 3;12(5):467-82
pubmed: 21035758

Auteurs

Katia Mellal (K)

Faculty of Pharmacy, Université de Montréal, Montreal, Canada.

Samy Omri (S)

Maisonneuve-Rosemont Hospital, Montréal, Canada.
Mperia Therapeutics, Montréal, Canada.

Mukandila Mulumba (M)

Faculty of Pharmacy, Université de Montréal, Montreal, Canada.

Houda Tahiri (H)

Departments of Pediatrics, Ophthalmology and Pharmacology, Université de Montréal, Montreal, Canada.

Carl Fortin (C)

Faculty of Pharmacy, Université de Montréal, Montreal, Canada.

Marie-France Dorion (MF)

Faculty of Pharmacy, Université de Montréal, Montreal, Canada.

Hung Pham (H)

Faculty of Pharmacy, Université de Montréal, Montreal, Canada.

Yesica Garcia Ramos (Y)

Department of Chemistry, Université de Montréal, Montreal, Canada.

Jinqiang Zhang (J)

Department of Chemistry, Université de Montréal, Montreal, Canada.

Sheetal Pundir (S)

Departments of Pediatrics, Ophthalmology and Pharmacology, Université de Montréal, Montreal, Canada.

Jean-Sébastien Joyal (JS)

Departments of Pediatrics, Ophthalmology and Pharmacology, Université de Montréal, Montreal, Canada.

Jean-François Bouchard (JF)

Neuropharmacology Laboratory, School of Optometry, Université de Montréal, Montreal, Canada.

Florian Sennlaub (F)

Institut de la Vision, Sorbonne Universités, INSERM, CNRS, Paris, France.

Maria Febbraio (M)

Department of Dentistry, University of Alberta, Edmonton, Canada.

Pierre Hardy (P)

Departments of Pediatrics, Ophthalmology and Pharmacology, Université de Montréal, Montreal, Canada.

Simon-Pierre Gravel (SP)

Faculty of Pharmacy, Université de Montréal, Montreal, Canada.

Sylvie Marleau (S)

Faculty of Pharmacy, Université de Montréal, Montreal, Canada.

William D Lubell (WD)

Department of Chemistry, Université de Montréal, Montreal, Canada.

Sylvain Chemtob (S)

Maisonneuve-Rosemont Hospital, Montréal, Canada. sylvain.chemtob@umontreal.ca.
Departments of Pediatrics, Ophthalmology and Pharmacology, Université de Montréal, Montreal, Canada. sylvain.chemtob@umontreal.ca.

Huy Ong (H)

Faculty of Pharmacy, Université de Montréal, Montreal, Canada. huy.ong@umontreal.ca.

Articles similaires

Robotic Surgical Procedures Animals Humans Telemedicine Models, Animal

Odour generalisation and detection dog training.

Lyn Caldicott, Thomas W Pike, Helen E Zulch et al.
1.00
Animals Odorants Dogs Generalization, Psychological Smell
C-Reactive Protein Humans Biomarkers Inflammation
Animals TOR Serine-Threonine Kinases Colorectal Neoplasms Colitis Mice

Classifications MeSH