Hit-to-Lead Optimization of Benzoxazepinoindazoles As Human African Trypanosomiasis Therapeutics.
Journal
Journal of medicinal chemistry
ISSN: 1520-4804
Titre abrégé: J Med Chem
Pays: United States
ID NLM: 9716531
Informations de publication
Date de publication:
12 03 2020
12 03 2020
Historique:
pubmed:
2
11
2019
medline:
1
9
2020
entrez:
1
11
2019
Statut:
ppublish
Résumé
Human African trypanosomiasis (HAT) is a neglected tropical disease caused by infection with either of two subspecies of the parasite
Identifiants
pubmed: 31670951
doi: 10.1021/acs.jmedchem.9b01506
pmc: PMC8329730
mid: NIHMS1728378
doi:
Substances chimiques
Indazoles
0
Oxazepines
0
Small Molecule Libraries
0
Trypanocidal Agents
0
Types de publication
Journal Article
Research Support, N.I.H., Extramural
Research Support, Non-U.S. Gov't
Langues
eng
Sous-ensembles de citation
IM
Pagination
2527-2546Subventions
Organisme : NIAID NIH HHS
ID : R01 AI114685
Pays : United States
Organisme : NIAID NIH HHS
ID : R01 AI124046
Pays : United States
Organisme : NIAID NIH HHS
ID : R21 AI126296
Pays : United States
Organisme : NIAID NIH HHS
ID : R21 AI127594
Pays : United States
Références
PLoS Negl Trop Dis. 2014 Oct 23;8(10):e3253
pubmed: 25340575
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pubmed: 29113731
Bioorg Med Chem Lett. 2013 Nov 1;23(21):5992-6000
pubmed: 24054120
Lancet. 2017 Nov 25;390(10110):2397-2409
pubmed: 28673422
Chem Rev. 2014 Nov 26;114(22):11280-304
pubmed: 26443079
Bioorg Med Chem Lett. 2016 Jun 1;26(11):2569-76
pubmed: 27080183
ACS Chem Neurosci. 2010 Jun 16;1(6):435-49
pubmed: 22778837