Furin-Guided Intracellular
Animals
Biomarkers, Tumor
/ genetics
Breast Neoplasms
/ diagnostic imaging
Cell Line, Tumor
Female
Furin
/ genetics
Gallium Radioisotopes
/ chemistry
Gene Expression
Heterografts
Humans
Liver
/ metabolism
Mice
Mice, Nude
Nanoparticles
/ metabolism
Positron-Emission Tomography
/ methods
Radiopharmaceuticals
/ chemical synthesis
Journal
Analytical chemistry
ISSN: 1520-6882
Titre abrégé: Anal Chem
Pays: United States
ID NLM: 0370536
Informations de publication
Date de publication:
03 12 2019
03 12 2019
Historique:
pubmed:
14
11
2019
medline:
21
10
2020
entrez:
14
11
2019
Statut:
ppublish
Résumé
Positron-emission tomography (PET) is routinely used in the clinic for tumor imaging with ultrahigh sensitivity, but tumor-targeted PET imaging probes are quite few. In this work, we rationally designed a furin-responsive radiotracer Acetyl-Arg-Val-Arg-Arg-Cys(StBu)-Lys(DOTA-
Identifiants
pubmed: 31718142
doi: 10.1021/acs.analchem.9b04788
doi:
Substances chimiques
Biomarkers, Tumor
0
Gallium Radioisotopes
0
Radiopharmaceuticals
0
FURIN protein, human
EC 3.4.21.75
Furin
EC 3.4.21.75
Types de publication
Journal Article
Research Support, Non-U.S. Gov't
Langues
eng
Sous-ensembles de citation
IM