Bedaquiline, moxifloxacin, pretomanid, and pyrazinamide during the first 8 weeks of treatment of patients with drug-susceptible or drug-resistant pulmonary tuberculosis: a multicentre, open-label, partially randomised, phase 2b trial.


Journal

The Lancet. Respiratory medicine
ISSN: 2213-2619
Titre abrégé: Lancet Respir Med
Pays: England
ID NLM: 101605555

Informations de publication

Date de publication:
12 2019
Historique:
received: 11 12 2018
revised: 28 08 2019
accepted: 03 09 2019
pubmed: 17 11 2019
medline: 2 7 2020
entrez: 17 11 2019
Statut: ppublish

Résumé

New anti-tuberculosis regimens that are shorter, simpler, and less toxic than those that are currently available are needed as part of the global effort to address the tuberculosis epidemic. We aimed to investigate the bactericidal activity and safety profile of combinations of bedaquiline, pretomanid, moxifloxacin, and pyrazinamide in the first 8 weeks of treatment of pulmonary tuberculosis. In this multicentre, open-label, partially randomised, phase 2b trial, we prospectively recruited patients with drug-susceptible or rifampicin-resistant pulmonary tuberculosis from seven sites in South Africa, two in Tanzania, and one in Uganda. Patients aged 18 years or older with sputum smear grade 1+ or higher were eligible for enrolment, and a molecular assay (GeneXpert or MTBDRplus) was used to confirm the diagnosis of tuberculosis and to distinguish between drug-susceptible and rifampicin-resistant tuberculosis. Patients who were HIV positive with a baseline CD4 cell count of less than 100 cells per uL were excluded. Patients with drug-susceptible tuberculosis were randomly assigned (1:1:1) using numbered treatment packs with sequential allocation by the pharmacist to receive 56 days of treatment with standard tuberculosis therapy (oral isoniazid, rifampicin, pyrazinamide, and ethambutol; HRZE), or pretomanid (oral 200 mg daily) and pyrazinamide (oral 1500 mg daily) with either oral bedaquiline 400 mg daily on days 1-14 then 200 mg three times per week (B Between Oct 24, 2014, and Dec 15, 2015, we enrolled 180 patients with drug-susceptible tuberculosis (59 were randomly assigned to B B TB Alliance, UK Department for International Development, Bill & Melinda Gates Foundation, US Agency for International Development, Directorate General for International Cooperation of the Netherlands, Irish Aid, Australia Department of Foreign Affairs and Trade, and the Federal Ministry for Education and Research of Germany.

Sections du résumé

BACKGROUND
New anti-tuberculosis regimens that are shorter, simpler, and less toxic than those that are currently available are needed as part of the global effort to address the tuberculosis epidemic. We aimed to investigate the bactericidal activity and safety profile of combinations of bedaquiline, pretomanid, moxifloxacin, and pyrazinamide in the first 8 weeks of treatment of pulmonary tuberculosis.
METHODS
In this multicentre, open-label, partially randomised, phase 2b trial, we prospectively recruited patients with drug-susceptible or rifampicin-resistant pulmonary tuberculosis from seven sites in South Africa, two in Tanzania, and one in Uganda. Patients aged 18 years or older with sputum smear grade 1+ or higher were eligible for enrolment, and a molecular assay (GeneXpert or MTBDRplus) was used to confirm the diagnosis of tuberculosis and to distinguish between drug-susceptible and rifampicin-resistant tuberculosis. Patients who were HIV positive with a baseline CD4 cell count of less than 100 cells per uL were excluded. Patients with drug-susceptible tuberculosis were randomly assigned (1:1:1) using numbered treatment packs with sequential allocation by the pharmacist to receive 56 days of treatment with standard tuberculosis therapy (oral isoniazid, rifampicin, pyrazinamide, and ethambutol; HRZE), or pretomanid (oral 200 mg daily) and pyrazinamide (oral 1500 mg daily) with either oral bedaquiline 400 mg daily on days 1-14 then 200 mg three times per week (B
FINDINGS
Between Oct 24, 2014, and Dec 15, 2015, we enrolled 180 patients with drug-susceptible tuberculosis (59 were randomly assigned to B
INTERPRETATION
B
FUNDING
TB Alliance, UK Department for International Development, Bill & Melinda Gates Foundation, US Agency for International Development, Directorate General for International Cooperation of the Netherlands, Irish Aid, Australia Department of Foreign Affairs and Trade, and the Federal Ministry for Education and Research of Germany.

Identifiants

pubmed: 31732485
pii: S2213-2600(19)30366-2
doi: 10.1016/S2213-2600(19)30366-2
pmc: PMC7641992
pii:
doi:

Substances chimiques

Antitubercular Agents 0
Diarylquinolines 0
Nitroimidazoles 0
pretomanid 0
Pyrazinamide 2KNI5N06TI
bedaquiline 78846I289Y
Moxifloxacin U188XYD42P
Rifampin VJT6J7R4TR

Banques de données

ClinicalTrials.gov
['NCT02193776']

Types de publication

Clinical Trial, Phase II Journal Article Multicenter Study Randomized Controlled Trial Research Support, Non-U.S. Gov't

Langues

eng

Sous-ensembles de citation

IM

Pagination

1048-1058

Subventions

Organisme : Medical Research Council
ID : MC_UU_12023/27
Pays : United Kingdom

Commentaires et corrections

Type : CommentIn
Type : CommentIn

Informations de copyright

Copyright © 2019 The Author(s). Published by Elsevier Ltd. This is an Open Access article under the CC BY 4.0 license. Published by Elsevier Ltd.. All rights reserved.

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Auteurs

Conor D Tweed (CD)

MRC Clinical Trials Unit at UCL, London, UK. Electronic address: c.tweed@ucl.ac.uk.

Rodney Dawson (R)

University of Cape Town Lung Institute, Cape Town, South Africa; Division of Pulmonology, Department of Medicine, University of Cape Town, Cape Town, South Africa.

Divan A Burger (DA)

Department of Statistics, University of Pretoria, Pretoria, South Africa.

Almari Conradie (A)

TB Alliance, Pretoria, South Africa.

Angela M Crook (AM)

MRC Clinical Trials Unit at UCL, London, UK.

Carl M Mendel (CM)

Global Alliance for TB Drug Development, New York, NY, USA.

Francesca Conradie (F)

Clinical HIV Research Unit, University of Witwatersrand, Johannesburg, South Africa.

Andreas H Diacon (AH)

TASK Applied Science, Bellville, South Africa; Division of Physiology, Department of Medical Biochemistry, Stellenbosch University, Tygerberg, South Africa.

Nyanda E Ntinginya (NE)

NIMR-Mbeya Medical Research Centre, Mbeya, Tanzania.

Daniel E Everitt (DE)

Global Alliance for TB Drug Development, New York, NY, USA.

Frederick Haraka (F)

Ifakara Health Institute Bagamoyo Research and Training Center, Bagamoyo, Tanzania.

Mengchun Li (M)

Global Alliance for TB Drug Development, New York, NY, USA.

Christo H van Niekerk (CH)

TB Alliance, Pretoria, South Africa.

Alphonse Okwera (A)

Uganda Case Western Reserve University Research Collaboration, Kampala, Uganda.

Mohammed S Rassool (MS)

Clinical HIV Research Unit, Helen Joseph Hospital, Johannesburg, South Africa.

Klaus Reither (K)

Ifakara Health Institute Bagamoyo Research and Training Center, Bagamoyo, Tanzania; Swiss Tropical and Public Health Institute, Basel, Switzerland.

Modulakgotla A Sebe (MA)

The Aurum Institute, Tembisa Hospital, Tembisa, South Africa.

Suzanne Staples (S)

THINK, Durban, South Africa.

Ebrahim Variava (E)

MDR Unit, Klerksdorp Tshepong Hospital, Klerksdorp, South Africa.

Melvin Spigelman (M)

Global Alliance for TB Drug Development, New York, NY, USA.

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