Optimizing the Synthetic Route of Chromone-2-carboxylic Acids: A Step forward to Speed-Up the Discovery of Chromone-Based Multitarget-Directed Ligands.

chromone-2-carboxylic acids microwave-assisted reaction multitarget ligands

Journal

Molecules (Basel, Switzerland)
ISSN: 1420-3049
Titre abrégé: Molecules
Pays: Switzerland
ID NLM: 100964009

Informations de publication

Date de publication:
20 Nov 2019
Historique:
received: 13 09 2019
revised: 26 10 2019
accepted: 19 11 2019
entrez: 24 11 2019
pubmed: 24 11 2019
medline: 15 4 2020
Statut: epublish

Résumé

6-Bromochromone-2-carboxylic acid (

Identifiants

pubmed: 31757041
pii: molecules24234214
doi: 10.3390/molecules24234214
pmc: PMC6930484
pii:
doi:

Substances chimiques

Chromones 0
Ligands 0
chromone-2-carboxylic acid 4940-39-0

Types de publication

Journal Article

Langues

eng

Sous-ensembles de citation

IM

Subventions

Organisme : FEDER funds through the Operational Programme Competitiveness Factors-COMPETE and national funds by FCT - Foundation for Science and Technology
ID : UID/QUI/00081/2019 and FEDER/COMPETE POCI-01-0145-FEDER-028397

Déclaration de conflit d'intérêts

The authors declare no conflict of interest.

Références

Chem Rev. 1996 Dec 19;96(8):3147-3176
pubmed: 11848856
Drug Discov Today. 2002 Mar 15;7(6):373-80
pubmed: 11893546
J Org Chem. 2009 Apr 3;74(7):2755-9
pubmed: 19323574
Front Chem. 2018 Apr 23;6:126
pubmed: 29740575
Chem Rev. 2014 May 14;114(9):4960-92
pubmed: 24555663
J Med Chem. 2017 Oct 12;60(19):7941-7957
pubmed: 28537720
Eur J Med Chem. 2018 Oct 5;158:781-800
pubmed: 30245401
Drug Discov Today Technol. 2005 Summer;2(2):155-61
pubmed: 24981843

Auteurs

Fernando Cagide (F)

CIQUP/Department of Chemistry and Biochemistry, Faculty of Sciences, University of Porto, Rua do Campo Alegre, 4169-007 Porto, Portugal.

Catarina Oliveira (C)

CIQUP/Department of Chemistry and Biochemistry, Faculty of Sciences, University of Porto, Rua do Campo Alegre, 4169-007 Porto, Portugal.

Fernanda Borges (F)

CIQUP/Department of Chemistry and Biochemistry, Faculty of Sciences, University of Porto, Rua do Campo Alegre, 4169-007 Porto, Portugal.

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Classifications MeSH