Selectivity filter instability dominates the low intrinsic activity of the TWIK-1 K2P K


Journal

The Journal of biological chemistry
ISSN: 1083-351X
Titre abrégé: J Biol Chem
Pays: United States
ID NLM: 2985121R

Informations de publication

Date de publication:
10 01 2020
Historique:
received: 14 08 2019
revised: 04 12 2019
pubmed: 7 12 2019
medline: 15 9 2020
entrez: 7 12 2019
Statut: ppublish

Résumé

Two-pore domain K

Identifiants

pubmed: 31806709
pii: S0021-9258(17)48351-7
doi: 10.1074/jbc.RA119.010612
pmc: PMC6956551
pii:
doi:

Substances chimiques

Cations, Monovalent 0
KCNK1 protein, human 0
Potassium Channels, Tandem Pore Domain 0
Rubidium MLT4718TJW
Potassium RWP5GA015D

Banques de données

PDB
['3UKM']

Types de publication

Journal Article Research Support, Non-U.S. Gov't

Langues

eng

Sous-ensembles de citation

IM

Pagination

610-618

Subventions

Organisme : Biotechnology and Biological Sciences Research Council
ID : BB/N000145/1
Pays : United Kingdom

Informations de copyright

© 2020 Nematian-Ardestani et al.

Références

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Auteurs

Ehsan Nematian-Ardestani (E)

Clarendon Laboratory, Department of Physics, University of Oxford, Oxford OX1 3PU, United Kingdom.

Firdaus Abd-Wahab (F)

Clarendon Laboratory, Department of Physics, University of Oxford, Oxford OX1 3PU, United Kingdom.

Franck C Chatelain (FC)

Université Côte d'Azur, Centre National de la Recherche Scientifique, Institut de Pharmacologie Moléculaire et Cellulaire, Labex ICST, 06560 Valbonne, France.

Han Sun (H)

Department of Structural Biology, Leibniz-Forschungsinstitut für Molekulare Pharmakologie, 13125 Berlin, Germany.

Marcus Schewe (M)

Institute of Physiology, Christian-Albrechts University of Kiel, 24118 Kiel, Germany.

Thomas Baukrowitz (T)

Institute of Physiology, Christian-Albrechts University of Kiel, 24118 Kiel, Germany.

Stephen J Tucker (SJ)

Clarendon Laboratory, Department of Physics, University of Oxford, Oxford OX1 3PU, United Kingdom. Electronic address: stephen.tucker@physics.ox.ac.uk.

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Classifications MeSH