Modeling the nonlinear behavior of a bioactive peptide in reversed-phase gradient elution chromatography.

Adsorption isotherms Gradient elution Inverse method Pharmaceutical peptides Preparative chromatography Reversed-phase liquid chromatography (RP-LC)

Journal

Journal of chromatography. A
ISSN: 1873-3778
Titre abrégé: J Chromatogr A
Pays: Netherlands
ID NLM: 9318488

Informations de publication

Date de publication:
12 Apr 2020
Historique:
received: 22 10 2019
revised: 09 12 2019
accepted: 12 12 2019
pubmed: 26 12 2019
medline: 18 6 2020
entrez: 26 12 2019
Statut: ppublish

Résumé

The thermodynamic behavior of octreotide, a cyclic octapeptide with important pharmaceutical functions, has been simulated under reversed-phase gradient elution conditions. To this end, adsorption behavior was firstly investigated in isocratic conditions, under a variety of water/acetonitrile + 0.02% (v/v) trifluoroacetic acid (TFA) mixtures as mobile phase by using a Langmuir isotherm. Organic modifier was varied in the range between 23 and 28% (v/v). Adsorption isotherms were determined by means of the so-called Inverse Method (IM) with a minimum amount of peptide. The linear solvent strength (LSS) model was used to find the correlation between isotherm parameters and mobile phase composition. This study contributes to enlarge our knowledge on the chromatographic behavior under nonlinear gradient conditions of peptides. In particular, it focuses on a cyclic octapeptide.

Identifiants

pubmed: 31874699
pii: S0021-9673(19)31237-3
doi: 10.1016/j.chroma.2019.460789
pii:
doi:

Substances chimiques

Peptides 0
Solvents 0
Water 059QF0KO0R

Types de publication

Journal Article

Langues

eng

Sous-ensembles de citation

IM

Pagination

460789

Informations de copyright

Copyright © 2019. Published by Elsevier B.V.

Déclaration de conflit d'intérêts

Declaration of Competing Interest None.

Auteurs

Chiara De Luca (C)

Dept. of Chemistry and Pharmaceutical Sciences, University of Ferrara, via L. Borsari 46, Ferrara 44121, Italy.

Simona Felletti (S)

Dept. of Chemistry and Pharmaceutical Sciences, University of Ferrara, via L. Borsari 46, Ferrara 44121, Italy.

Marco Macis (M)

Fresenius Kabi iPSUM, via San Leonardo 23, Villadose, Rovigo 45010, Italy.

Walter Cabri (W)

Fresenius Kabi iPSUM, via San Leonardo 23, Villadose, Rovigo 45010, Italy.

Giulio Lievore (G)

Dept. of Chemistry and Pharmaceutical Sciences, University of Ferrara, via L. Borsari 46, Ferrara 44121, Italy.

Tatiana Chenet (T)

Dept. of Chemistry and Pharmaceutical Sciences, University of Ferrara, via L. Borsari 46, Ferrara 44121, Italy.

Luisa Pasti (L)

Dept. of Chemistry and Pharmaceutical Sciences, University of Ferrara, via L. Borsari 46, Ferrara 44121, Italy.

Massimo Morbidelli (M)

Dept. of Chemistry and Applied Biosciences, Institute for Chemical and Bioengineering, ETH Zurich, Vladimir-Prelog-Weg 1, Zurich 8093, Switzerland.

Alberto Cavazzini (A)

Dept. of Chemistry and Pharmaceutical Sciences, University of Ferrara, via L. Borsari 46, Ferrara 44121, Italy. Electronic address: cvz@unife.it.

Martina Catani (M)

Dept. of Chemistry and Pharmaceutical Sciences, University of Ferrara, via L. Borsari 46, Ferrara 44121, Italy. Electronic address: ctnmtn@unife.it.

Antonio Ricci (A)

Fresenius Kabi iPSUM, via San Leonardo 23, Villadose, Rovigo 45010, Italy.

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Classifications MeSH