Correlation between the potency of hallucinogens in the mouse head-twitch response assay and their behavioral and subjective effects in other species.
Animals
Discrimination Learning
/ drug effects
Dose-Response Relationship, Drug
Hallucinogens
/ administration & dosage
Head Movements
/ drug effects
Humans
Magnetometry
/ instrumentation
Male
Mice
Mice, Inbred C57BL
Rats
Receptor, Serotonin, 5-HT2A
/ physiology
Serotonin 5-HT2 Receptor Agonists
/ administration & dosage
Species Specificity
Behavioral model
DMT
DOM
Head shake
Mescaline
N,N-dimethyltryptamine
NBOMe
Psilocybin
Psychedelic
Journal
Neuropharmacology
ISSN: 1873-7064
Titre abrégé: Neuropharmacology
Pays: England
ID NLM: 0236217
Informations de publication
Date de publication:
01 05 2020
01 05 2020
Historique:
received:
22
10
2019
revised:
28
12
2019
accepted:
31
12
2019
pubmed:
10
1
2020
medline:
24
4
2021
entrez:
10
1
2020
Statut:
ppublish
Résumé
Serotonergic hallucinogens such as lysergic acid diethylamide (LSD) induce head twitches in rodents via 5-HT
Identifiants
pubmed: 31917152
pii: S0028-3908(19)30504-0
doi: 10.1016/j.neuropharm.2019.107933
pmc: PMC9191653
mid: NIHMS1564203
pii:
doi:
Substances chimiques
Hallucinogens
0
Receptor, Serotonin, 5-HT2A
0
Serotonin 5-HT2 Receptor Agonists
0
Types de publication
Journal Article
Research Support, N.I.H., Extramural
Langues
eng
Sous-ensembles de citation
IM
Pagination
107933Subventions
Organisme : NIDA NIH HHS
ID : R01 DA041336
Pays : United States
Organisme : NIMH NIH HHS
ID : T32 MH018399
Pays : United States
Informations de copyright
Published by Elsevier Ltd.
Déclaration de conflit d'intérêts
Declaration of competing interest None.
Références
Pharmacol Ther. 2006 Mar;109(3):325-38
pubmed: 16023217
Proc Natl Acad Sci U S A. 2009 Nov 17;106(46):19575-80
pubmed: 19889983
Eur J Pharmacol. 2008 Oct 10;594(1-3):32-8
pubmed: 18703043
J Psychopharmacol. 2016 Dec;30(12):1181-1197
pubmed: 27909165
Int J Neuropsychopharmacol. 2018 Oct 1;21(10):926-931
pubmed: 29850881
Cell Rep. 2018 Jun 12;23(11):3170-3182
pubmed: 29898390
J Med Chem. 1985 Sep;28(9):1252-5
pubmed: 4032428
J Med Chem. 1995 Mar 17;38(6):958-66
pubmed: 7699712
Pharmacol Rev. 2016 Apr;68(2):264-355
pubmed: 26841800
Life Sci. 1984 Dec 17;35(25):2505-11
pubmed: 6513725
ACS Chem Neurosci. 2015 Jul 15;6(7):1165-75
pubmed: 25547199
Eur J Pharmacol. 1983 Jan 21;86(3-4):453-9
pubmed: 6572591
Psychopharmacology (Berl). 2002 Oct;164(1):93-107
pubmed: 12373423
Pharmacol Biochem Behav. 1982 Oct;17(4):603-7
pubmed: 6965276
Psychopharmacology (Berl). 1980;68(2):159-62
pubmed: 6776559
Mol Pharmacol. 2006 Dec;70(6):1956-64
pubmed: 17000863
Behav Brain Res. 1996;73(1-2):121-4
pubmed: 8788488
J Med Chem. 2003 Jul 31;46(16):3526-35
pubmed: 12877591
Pharmacol Biochem Behav. 2008 Jan;88(3):358-65
pubmed: 17905422
Psychopharmacology (Berl). 2010 Apr;209(2):163-74
pubmed: 20165943
Neuropharmacology. 2014 Feb;77:200-7
pubmed: 24012658
Psychopharmacology (Berl). 1995 Oct;121(3):347-56
pubmed: 8584617
J Med Chem. 2000 Nov 30;43(24):4701-10
pubmed: 11101361
Br J Pharmacol Chemother. 1963 Feb;20:106-20
pubmed: 14023050
J Med Chem. 1997 Sep 12;40(19):2997-3008
pubmed: 9301661
Eur J Pharmacol. 1983 Jul 22;91(2-3):189-96
pubmed: 6617740
Psychopharmacology (Berl). 1982;76(2):130-5
pubmed: 6805022
Pharmacol Biochem Behav. 1994 Mar;47(3):667-73
pubmed: 8208787
Science. 1982 Apr 30;216(4545):535-7
pubmed: 7071600
Behav Brain Res. 2015 Jan 15;277:99-120
pubmed: 25036425
J Pharmacol Exp Ther. 1995 Apr;273(1):101-12
pubmed: 7714755
Drug Test Anal. 2019 Aug;11(8):1122-1133
pubmed: 31083768
ACS Chem Neurosci. 2013 Jan 16;4(1):96-109
pubmed: 23336049
Neuropsychopharmacology. 1996 Apr;14(4):233-41
pubmed: 8924191
Behav Brain Res. 2019 Feb 1;359:828-835
pubmed: 30053461
Psychopharmacologia. 1971;20(1):66-76
pubmed: 5565748
Neuropharmacology. 2011 Sep;61(3):503-12
pubmed: 21352832
Arch Gen Psychiatry. 1966 Sep;15(3):320-9
pubmed: 5330062
Psychopharmacology (Berl). 1980;68(3):209-15
pubmed: 6771804
J Med Chem. 2006 Jan 12;49(1):318-28
pubmed: 16392816
Med Res Rev. 1983 Jul-Sep;3(3):289-340
pubmed: 6350763
J Psychopharmacol. 2014 Nov;28(11):983-92
pubmed: 25213996
Pharmacol Biochem Behav. 2007 Oct;87(4):472-80
pubmed: 17688928
Neuropharmacology. 2011 Sep;61(3):364-81
pubmed: 21256140
Psychopharmacology (Berl). 1982;76(1):20-5
pubmed: 6805003
CMAJ. 2003 May 27;168(11):1439-42
pubmed: 12771076
Neuropsychopharmacology. 2008 Aug;33(9):2206-16
pubmed: 17957214
Eur Neuropsychopharmacol. 2016 Jul;26(7):1161-75
pubmed: 27039035
Pharmacol Biochem Behav. 1998 May;60(1):83-90
pubmed: 9610928
Curr Biol. 2017 Feb 6;27(3):451-457
pubmed: 28132813
Biochem Pharmacol. 1991 Jun 1;41(11):1739-44
pubmed: 1828347
J Med Chem. 1992 Jan 24;35(2):203-11
pubmed: 1732537
Neuropharmacology. 2019 Jan;144:368-376
pubmed: 30385253
J Pharmacol Exp Ther. 2010 Dec;335(3):728-34
pubmed: 20858706
Pharmacol Biochem Behav. 1990 Aug;36(4):901-6
pubmed: 2145593
Emerg Med J. 2007 Apr;24(4):e20
pubmed: 17384366
Pharmacopsychiatria. 1981 Sep;14(5):162-6
pubmed: 7291300
Am J Psychiatry. 1976 Feb;133(2):203-8
pubmed: 1062171
Pharmacol Biochem Behav. 1985 Dec;23(6):937-41
pubmed: 2934750
Biol Psychiatry. 1982 Jul;17(7):807-14
pubmed: 6126227
Neuropsychopharmacology. 2000 Nov;23(5):569-76
pubmed: 11027922
Psychopharmacologia. 1973;33(2):117-34
pubmed: 4272898
J Psychopharmacol. 2014 Jun;28(6):545-52
pubmed: 24785760
Pharmacol Biochem Behav. 2001 Jul-Aug;69(3-4):643-52
pubmed: 11509227
Drug Test Anal. 2016 Sep;8(9):891-902
pubmed: 26456305
Eur J Pharmacol. 1987 Aug 21;140(3):323-30
pubmed: 3653248
ACS Chem Neurosci. 2018 Jul 18;9(7):1582-1590
pubmed: 29664276
J Pharmacol Exp Ther. 2014 Dec;351(3):485-91
pubmed: 25271256
J Psychopharmacol. 2011 Nov;25(11):1548-61
pubmed: 21148021
Neuropharmacology. 1981 May;20(5):473-5
pubmed: 7242868
J Ment Sci. 1959 Jan;105(438):171-81
pubmed: 13641966
Neuroreport. 1998 Dec 1;9(17):3897-902
pubmed: 9875725
Pharmacol Biochem Behav. 2006 Jan;83(1):122-9
pubmed: 16460788
J Med Chem. 1999 Mar 25;42(6):1106-11
pubmed: 10090793
Front Mol Neurosci. 2018 Sep 04;11:312
pubmed: 30233313
Behav Pharmacol. 2011 Sep;22(5-6):415-29
pubmed: 21808191
Neuron. 2007 Feb 1;53(3):439-52
pubmed: 17270739
NIDA Res Monogr. 1978;(22):27-37
pubmed: 101882
Psychopharmacology (Berl). 2017 Jul;234(13):2031-2046
pubmed: 28386699
J Nerv Ment Dis. 1967 Oct;145(4):306-13
pubmed: 6076017
J Med Chem. 1998 Dec 17;41(26):5148-9
pubmed: 9857084
J Pharmacol Exp Ther. 2011 Jul;338(1):280-9
pubmed: 21474568
Life Sci. 1978 Oct 9;23(14):1499-506
pubmed: 713706
J Med Chem. 1991 Jan;34(1):276-81
pubmed: 1992127
Drug Test Anal. 2012 Jul-Aug;4(7-8):556-76
pubmed: 22517680
J Med Chem. 1994 Dec 9;37(25):4346-51
pubmed: 7996545
Neuropharmacology. 1986 Nov;25(11):1289-91
pubmed: 3796801
Psychopharmacology (Berl). 1981;74(2):173-6
pubmed: 6168003
Neuropharmacology. 2016 Aug;107:364-375
pubmed: 27020041
J Clin Psychiatry. 2006 Nov;67(11):1735-40
pubmed: 17196053
J Med Chem. 1995 Sep 1;38(18):3593-601
pubmed: 7658446
Neuropharmacology. 2014 Aug;83:18-27
pubmed: 24680675
Neuropharmacology. 2018 Nov;142:240-250
pubmed: 29501528
Neuropharmacology. 2013 Jul;70:112-21
pubmed: 23353901
Behav Pharmacol. 2017 Aug;28(5):375-385
pubmed: 28537942
Pharmacol Biochem Behav. 1982 Apr;16(4):557-9
pubmed: 7071089
Psychopharmacology (Berl). 2019 Feb;236(2):799-808
pubmed: 30298278
Am J Drug Alcohol Abuse. 2017 Jan;43(1):55-60
pubmed: 27441452
Prog Neuropsychopharmacol Biol Psychiatry. 1998 May;22(4):649-63
pubmed: 9682278
Neuropharmacology. 2018 Nov;142:231-239
pubmed: 29499272
J Psychopharmacol. 2015 Mar;29(3):289-99
pubmed: 25586396
Commun Psychopharmacol. 1980;4(5):363-9
pubmed: 6949674
Psychopharmacology (Berl). 1995 Oct;121(3):357-63
pubmed: 8584618
Commun Psychopharmacol. 1980;4(6):501-6
pubmed: 7297054
Psychopharmacologia. 1967;11(1):65-78
pubmed: 5302272
Biochem Pharmacol. 2008 Jan 1;75(1):17-33
pubmed: 17977517
Drug Test Anal. 2017 Jan;9(1):38-50
pubmed: 27265891
Psychopharmacology (Berl). 2015 Jan;232(1):275-84
pubmed: 24985890
Arch Gen Psychiatry. 1973 Jun;28(6):817-21
pubmed: 4575167
J Psychopharmacol. 2016 Dec;30(12):1165-1180
pubmed: 27909164
Exp Brain Res. 2013 Aug;228(4):481-91
pubmed: 23727882
Psychopharmacology (Berl). 2013 Jun;227(4):727-39
pubmed: 23407781
J Med Chem. 1996 Jul 19;39(15):2953-61
pubmed: 8709129
Psychopharmacology (Berl). 1989;97(2):206-12
pubmed: 2471220
J Psychopharmacol. 2019 Mar;33(3):406-414
pubmed: 30789291
Mol Pharmacol. 1982 Mar;21(2):301-14
pubmed: 7099138
Arch Gen Psychiatry. 2011 Jan;68(1):71-8
pubmed: 20819978
PLoS One. 2010 Feb 02;5(2):e9019
pubmed: 20126400
Drug Test Anal. 2018 Feb;10(2):310-322
pubmed: 28585392
J Pharmacol Exp Ther. 2007 Jun;321(3):1054-61
pubmed: 17337633
Neurosci Biobehav Rev. 1982 Winter;6(4):529-36
pubmed: 7177512
J Med Chem. 2002 Sep 12;45(19):4344-9
pubmed: 12213075
J Med Chem. 2006 Jul 13;49(14):4269-74
pubmed: 16821786
Pharmacol Biochem Behav. 1988 Jul;30(3):597-601
pubmed: 3211969
Psychopharmacology (Berl). 2005 Jul;180(3):427-35
pubmed: 15723230
ACS Chem Neurosci. 2019 Jul 17;10(7):3261-3270
pubmed: 30829033
Biochem Pharmacol. 1983 Apr 1;32(7):1267-73
pubmed: 6573879
NIDA Res Monogr. 1989;94:43-67
pubmed: 2575229
Brain Res Mol Brain Res. 2003 Jul 23;115(2):162-72
pubmed: 12877987
Curr Top Behav Neurosci. 2018;36:1-43
pubmed: 28401524
Psychopharmacology (Berl). 1996 Nov;128(2):198-205
pubmed: 8956381
J Med Chem. 1982 Oct;25(10):1163-8
pubmed: 7143352
Psychopharmacology (Berl). 1990;100(3):417-25
pubmed: 2138338