Venom diversity in the Neotropical scorpion genus Tityus: Implications for antivenom design emerging from molecular and immunochemical analyses across endemic areas of scorpionism.


Journal

Acta tropica
ISSN: 1873-6254
Titre abrégé: Acta Trop
Pays: Netherlands
ID NLM: 0370374

Informations de publication

Date de publication:
Apr 2020
Historique:
received: 01 11 2019
revised: 14 01 2020
accepted: 14 01 2020
pubmed: 27 1 2020
medline: 21 8 2020
entrez: 27 1 2020
Statut: ppublish

Résumé

Scorpions of the Neotropical genus Tityus are responsible for most severe envenomations in the Caribbean, South America, and Lower Central America (LCA). Although Tityus is taxonomically complex, contains high toxin polymorphism, and produces variable clinical manifestations, treatment is limited to antivenoms produced against species with restricted distributions. In this study, we explored the compositional and antigenic diversity of Tityus venoms to provide improved guidelines for the use of available antivenoms at a broader geographic scale. We used immunoblotting, competitive ELISA, and in vivo studies to compare reactivity against commercial antivenoms from Brazil, Venezuela, and Mexico, as well as MALDI-TOF mass spectrometry, cDNA sequencing, and phylogenetic analyses to assess venom sodium channel-active toxin (NaTx) content from medically important Tityus populations inhabiting Brazil, Colombia, Costa Rica, Ecuador, Panama, Trinidad and Tobago, and Venezuela. Additionally, we raised rabbit antibodies against Tityus venoms from LCA to test for cross-reactivity with congeneric species. The results suggest that Tityus spp. possess high venom antigenic diversity, underlying the existence of four toxinological regions in Tropical America, based on venom composition and immunochemical criteria: LCA/Colombia/Amazonia (Region I), Venezuela (Region II), southeast South America (Region III), and a fourth region encompassing species related to toxinologically divergent Tityus cerroazul. Importantly, our molecular and cross-reactivity results highlight the need for new antivenoms against species inhabiting Region I, where scorpions may produce venoms that are not significantly reactive against available antivenoms.

Identifiants

pubmed: 31982434
pii: S0001-706X(19)31478-0
doi: 10.1016/j.actatropica.2020.105346
pii:
doi:

Substances chimiques

Antivenins 0
Scorpion Venoms 0

Types de publication

Journal Article

Langues

eng

Sous-ensembles de citation

IM

Pagination

105346

Informations de copyright

Copyright © 2020 Elsevier B.V. All rights reserved.

Déclaration de conflit d'intérêts

Declaration of Conflict Interest None.

Auteurs

Adolfo Borges (A)

Centro para el Desarrollo de la Investigación Científica, Manduvirá 635, Asunción, Paraguay; Laboratorio de Biología Molecular de Toxinas y Receptores, Instituto de Medicina Experimental, Universidad Central de Venezuela, Caracas 1050, Venezuela. Electronic address: borges.adolfo@gmail.com.

Bruno Lomonte (B)

Instituto Clodomiro Picado, Facultad de Microbiología, Universidad de Costa Rica, San José 11501, Costa Rica. Electronic address: bruno.lomonte@ucr.ac.cr.

Yamileth Angulo (Y)

Instituto Clodomiro Picado, Facultad de Microbiología, Universidad de Costa Rica, San José 11501, Costa Rica. Electronic address: yamileth.angulo@ucr.ac.cr.

Hildaura Acosta de Patiño (H)

Centro de Investigación e Información de Medicamentos y Tóxicos, Universidad de Panamá, Ciudad de Panamá, Panamá.

Juan M Pascale (JM)

Instituto Conmemorativo Gorgas de Estudios de la Salud, Departamento de Genómica y Proteómica, Ciudad de Panamá, Panamá.

Rafael Otero (R)

Facultad de Medicina, Universidad de Antioquia, Apartado 1226 Medellín, Colombia. Electronic address: rafaotero@une.net.co.

Roberto J Miranda (RJ)

Instituto Conmemorativo Gorgas de Estudios de la Salud, Departamento de Genómica y Proteómica, Ciudad de Panamá, Panamá.

Leonardo De Sousa (L)

Grupo de Investigación en Toxinología Aplicada, Sección de Farmacología, Escuela de Ciencias de la Salud, Departamento de Ciencias Fisiológicas, Universidad de Oriente, Barcelona, Venezuela.

Matthew R Graham (MR)

Department of Biology, Eastern Connecticut State University, Willimantic, CT 06226, United States. Electronic address: grahamm@easternct.edu.

Aarón Gómez (A)

Instituto Clodomiro Picado, Facultad de Microbiología, Universidad de Costa Rica, San José 11501, Costa Rica.

Pedro P O Pardal (PPO)

Laboratory of Medical Entomology and Venomous Animals, Center of Tropical Medicine, Pará Federal University, Belém 66055-240, Pará State, Brazil. Electronic address: pepardal@ufpa.br.

Edna Ishikawa (E)

Laboratory of Medical Entomology and Venomous Animals, Center of Tropical Medicine, Pará Federal University, Belém 66055-240, Pará State, Brazil. Electronic address: ishikawa@ufpa.br.

Fabián Bonilla (F)

Instituto Clodomiro Picado, Facultad de Microbiología, Universidad de Costa Rica, San José 11501, Costa Rica. Electronic address: fabian.bonilla@ucr.ac.cr.

Adolfo Castillo (A)

Centro de Investigación e Información de Medicamentos y Tóxicos, Universidad de Panamá, Ciudad de Panamá, Panamá.

Ricardo A Machado de Avila (RAM)

Centro para el Desarrollo de la Investigación Científica, Manduvirá 635, Asunción, Paraguay; Programa de Pós-Graduação em Ciências da Saúde, Universidade do Extremo Sul Catarinense, Criciúma 88806-000, Brazil.

Juan P Gómez (JP)

Facultad de Medicina, Universidad de Antioquia, Apartado 1226 Medellín, Colombia.

Jorge A Caro-López (JA)

Facultad de Medicina, Universidad de Antioquia, Apartado 1226 Medellín, Colombia.

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