Epigenetic Regulation of Multidrug Resistance Protein 1 and Breast Cancer Resistance Protein Transporters by Histone Deacetylase Inhibition.
ATP Binding Cassette Transporter, Subfamily B
/ genetics
ATP Binding Cassette Transporter, Subfamily G, Member 2
/ genetics
Acetylation
/ drug effects
Animals
Drug Resistance
/ drug effects
Epigenesis, Genetic
/ drug effects
Histone Deacetylase Inhibitors
/ pharmacology
Histone Deacetylases
/ metabolism
Histones
/ metabolism
Humans
Models, Animal
Neoplasm Proteins
/ genetics
Journal
Drug metabolism and disposition: the biological fate of chemicals
ISSN: 1521-009X
Titre abrégé: Drug Metab Dispos
Pays: United States
ID NLM: 9421550
Informations de publication
Date de publication:
06 2020
06 2020
Historique:
received:
07
11
2019
accepted:
13
02
2020
pubmed:
21
3
2020
medline:
20
7
2021
entrez:
21
3
2020
Statut:
ppublish
Résumé
Multidrug resistance protein 1 (MDR1,
Identifiants
pubmed: 32193359
pii: dmd.119.089953
doi: 10.1124/dmd.119.089953
pmc: PMC7250367
doi:
Substances chimiques
ABCB1 protein, human
0
ABCG2 protein, human
0
ATP Binding Cassette Transporter, Subfamily B
0
ATP Binding Cassette Transporter, Subfamily G, Member 2
0
Histone Deacetylase Inhibitors
0
Histones
0
Neoplasm Proteins
0
Histone Deacetylases
EC 3.5.1.98
Types de publication
Journal Article
Research Support, N.I.H., Extramural
Review
Langues
eng
Sous-ensembles de citation
IM
Pagination
459-480Subventions
Organisme : NIEHS NIH HHS
ID : P30 ES005022
Pays : United States
Organisme : NIEHS NIH HHS
ID : R01 ES021800
Pays : United States
Informations de copyright
Copyright © 2020 by The American Society for Pharmacology and Experimental Therapeutics.
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