Obtusaquinone: A Cysteine-Modifying Compound That Targets Keap1 for Degradation.
Journal
ACS chemical biology
ISSN: 1554-8937
Titre abrégé: ACS Chem Biol
Pays: United States
ID NLM: 101282906
Informations de publication
Date de publication:
19 06 2020
19 06 2020
Historique:
pubmed:
28
4
2020
medline:
13
4
2021
entrez:
28
4
2020
Statut:
ppublish
Résumé
We have previously identified the natural product obtusaquinone (OBT) as a potent antineoplastic agent with promising
Identifiants
pubmed: 32338864
doi: 10.1021/acschembio.0c00104
pmc: PMC7995447
mid: NIHMS1678726
doi:
Substances chimiques
Antineoplastic Agents
0
Cinnamates
0
Cyclohexanones
0
Kelch-Like ECH-Associated Protein 1
0
obtusaquinone
62745-67-9
Cysteine
K848JZ4886
Types de publication
Journal Article
Research Support, N.I.H., Extramural
Langues
eng
Sous-ensembles de citation
IM
Pagination
1445-1454Subventions
Organisme : NINDS NIH HHS
ID : R01 NS064983
Pays : United States
Organisme : NCRR NIH HHS
ID : S10 RR025504
Pays : United States
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