Determinants of Successful Use of Sirolimus in Renal Transplant Patients.


Journal

Transplantation proceedings
ISSN: 1873-2623
Titre abrégé: Transplant Proc
Pays: United States
ID NLM: 0243532

Informations de publication

Date de publication:
Dec 2020
Historique:
received: 30 01 2020
accepted: 13 02 2020
pubmed: 5 6 2020
medline: 16 2 2021
entrez: 5 6 2020
Statut: ppublish

Résumé

Sirolimus is an established immunosuppressant in renal transplantation with antineoplastic and antiviral features, but side effects like proteinuria limit its use. The aim of this retrospective multicenter observational study is to define predictors for determining which patients most likely benefit from a sirolimus-based therapy. All patients from 10 German centers that were switched to a sirolimus-containing maintenance immunosuppression in 2000 to 2008 after 3 months or later post-transplantation were enrolled (n = 726). Observation times after switching to sirolimus ranged from 4 days to 9 years (median: 24.3 months). With multinomial logistic regression, risk factors for the endpoints terminal graft failure and withdrawal of sirolimus therapy compared to successful therapy were identified. Successful sirolimus therapy was observed in 304 patients. Forty patients died with functioning graft. Therapy failures included graft loss (n = 106) and sirolimus-discontinuation for various reasons (n = 276). Successful sirolimus-use was predicted in 83% and graft failure in 65%, whereas prediction of deliberate sirolimus-discontinuation was poor (48%). Most favorable results for sirolimus-use were observed in patients switched in 2006 to 2008. Using ROC analysis, an estimated glomerular filtration rate (eGFR) below 32 mL/min was shown to be the cut-off in patients withdrawing from therapy as a result of renal reasons, as well as in patients with graft loss. Proteinuria above 151 mg/L was shown to be predictive for patients with graft failure. eGFR and proteinuria are the major determinants for successful sirolimus-therapy. Our findings help stratifying patients who will benefit most from this therapy and avoid toxicities in patients without potential benefits for this therapy.

Sections du résumé

BACKGROUND BACKGROUND
Sirolimus is an established immunosuppressant in renal transplantation with antineoplastic and antiviral features, but side effects like proteinuria limit its use. The aim of this retrospective multicenter observational study is to define predictors for determining which patients most likely benefit from a sirolimus-based therapy.
METHODS METHODS
All patients from 10 German centers that were switched to a sirolimus-containing maintenance immunosuppression in 2000 to 2008 after 3 months or later post-transplantation were enrolled (n = 726). Observation times after switching to sirolimus ranged from 4 days to 9 years (median: 24.3 months). With multinomial logistic regression, risk factors for the endpoints terminal graft failure and withdrawal of sirolimus therapy compared to successful therapy were identified.
RESULTS RESULTS
Successful sirolimus therapy was observed in 304 patients. Forty patients died with functioning graft. Therapy failures included graft loss (n = 106) and sirolimus-discontinuation for various reasons (n = 276). Successful sirolimus-use was predicted in 83% and graft failure in 65%, whereas prediction of deliberate sirolimus-discontinuation was poor (48%). Most favorable results for sirolimus-use were observed in patients switched in 2006 to 2008. Using ROC analysis, an estimated glomerular filtration rate (eGFR) below 32 mL/min was shown to be the cut-off in patients withdrawing from therapy as a result of renal reasons, as well as in patients with graft loss. Proteinuria above 151 mg/L was shown to be predictive for patients with graft failure.
CONCLUSIONS CONCLUSIONS
eGFR and proteinuria are the major determinants for successful sirolimus-therapy. Our findings help stratifying patients who will benefit most from this therapy and avoid toxicities in patients without potential benefits for this therapy.

Identifiants

pubmed: 32493677
pii: S0041-1345(19)31510-6
doi: 10.1016/j.transproceed.2020.02.159
pii:
doi:

Substances chimiques

Immunosuppressive Agents 0
Sirolimus W36ZG6FT64

Types de publication

Journal Article Multicenter Study Observational Study

Langues

eng

Sous-ensembles de citation

IM

Pagination

3103-3111

Informations de copyright

Copyright © 2020 The Authors. Published by Elsevier Inc. All rights reserved.

Auteurs

Marcel G Naik (MG)

Medical Department, Division of Nephrology and Internal Intensive Care Medicine, Charite University Medicine Berlin, Germany. Electronic address: marcel.naik@charite.de.

Jan Steffen Jürgensen (JS)

Medical Department, Division of Nephrology and Internal Intensive Care Medicine, Charite University Medicine Berlin, Germany; Division of Nephrology, EBC University Berlin and Klinikum, Stuttgart, Germany.

Wolfgang Arns (W)

Transplant Centre Cologne, Cologne General Hospital, Cologne, Germany.

Edin Basic (E)

Pfizer Pharma GmbH, Berlin, Germany.

Klemens Budde (K)

Medical Department, Division of Nephrology and Internal Intensive Care Medicine, Charite University Medicine Berlin, Germany.

Frank Eitner (F)

Division of Nephrology and Clinical Immunology, RWTH Aachen University, Aachen, Germany.

Michael Fischereder (M)

Department of Medicine IV, University Hospital LMU, Munich, Germany.

Jan Goßmann (J)

Division of Nephrology, Transplant Care Centre Frankfurt, Frankfurt, Germany.

Katharina M Heller (KM)

Division of Nephrology, Department of Medicine, University of Erlangen, Erlangen, Germany.

Nils Heyne (N)

Division of Nephrology, Universitätsklinikum Tübingen, Tübingen, Germany.

Christian Morath (C)

Division of Nephrology, University of Heidelberg, Heidelberg, Germany.

Udo Riester (U)

Pfizer Pharma GmbH, Berlin, Germany.

Fritz Diekmann (F)

Department of Nephrology and Kidney Transplantation, Hospital Clinic, Barcelona, Spain.

Wilfried Gwinner (W)

Division of Nephrology, Hannover Medical School, Hannover, Germany.

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Classifications MeSH