Norditerpenoids with Selective Anti-Cholinesterase Activity from the Roots of


Journal

International journal of molecular sciences
ISSN: 1422-0067
Titre abrégé: Int J Mol Sci
Pays: Switzerland
ID NLM: 101092791

Informations de publication

Date de publication:
23 Jun 2020
Historique:
received: 08 05 2020
revised: 16 06 2020
accepted: 19 06 2020
entrez: 27 6 2020
pubmed: 27 6 2020
medline: 23 3 2021
Statut: epublish

Résumé

Inhibition of cholinesterases remains one of a few available treatment strategies for neurodegenerative dementias such as Alzheimer's disease and related conditions. The current study was inspired by previous data on anticholinesterase properties of diterpenoids from

Identifiants

pubmed: 32586060
pii: ijms21124475
doi: 10.3390/ijms21124475
pmc: PMC7352922
pii:
doi:

Substances chimiques

Cholinesterase Inhibitors 0
Diterpenes 0
Plant Extracts 0
Acetylcholinesterase EC 3.1.1.7
Butyrylcholinesterase EC 3.1.1.8

Types de publication

Journal Article

Langues

eng

Sous-ensembles de citation

IM

Subventions

Organisme : Uniwersytet Medyczny im. Piastów Slaskich we Wroclawiu
ID : SUB.D033.19.009
Organisme : Narodowe Centrum Nauki
ID : FUGA 2014/12/S/NZ9/00715
Organisme : Fundación Séneca del Centro de Coordinación de la Investigación de la Región de Murcia
ID : 20988/PI/18 and 20524/PDC/18
Organisme : Türkiye Bilimsel ve Teknolojik Araştirma Kurumu
ID : POLTUR/PLANT-ALZH/5/2015
Organisme : Ministerstwo Nauki i Szkolnictwa Wyższego
ID : 96/E-394/SPUB/2019
Organisme : Ministerio de Ciencia e Innovación
ID : CTQ2017-87974-R

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Auteurs

Sylwester Ślusarczyk (S)

Department of Pharmaceutical Biology and Botany, Wroclaw Medical University, 50556 Wroclaw, Poland.

F Sezer Senol Deniz (FS)

Department of Pharmacognosy, Faculty of Pharmacy, Gazi University, 06330 Ankara, Turkey.

Renata Abel (R)

Department of Pharmaceutical Biology and Botany, Wroclaw Medical University, 50556 Wroclaw, Poland.
Structural Bioinformatics Group, Institute for Physiology & ECRC, Charité University Medicine, 10115 Berlin, Germany.

Łukasz Pecio (Ł)

Department of Biochemistry and Crop Quality, IUNG-Institute of Soil Science and Plant Cultivation, 24100 Puławy, Poland.

Horacio Pérez-Sánchez (H)

Structural Bioinformatics and High Performance Computing Research Group, Universidad Católica San Antonio de Murcia (UCAM), 30107, Murcia, Spain.

José P Cerón-Carrasco (JP)

Reconocimiento y Encapsulación Molecular (REM), Universidad Católica San Antonio de Murcia (UCAM), 30107 Murcia, Spain.

Helena den-Haan (H)

Structural Bioinformatics and High Performance Computing Research Group, Universidad Católica San Antonio de Murcia (UCAM), 30107, Murcia, Spain.

Priyanka Banerjee (P)

Structural Bioinformatics Group, Institute for Physiology & ECRC, Charité University Medicine, 10115 Berlin, Germany.

Robert Preissner (R)

Structural Bioinformatics Group, Institute for Physiology & ECRC, Charité University Medicine, 10115 Berlin, Germany.

Edward Krzyżak (E)

Department of Inorganic Chemistry, Wroclaw Medical University, 50556 Wroclaw, Poland.

Wiesław Oleszek (W)

Department of Biochemistry and Crop Quality, IUNG-Institute of Soil Science and Plant Cultivation, 24100 Puławy, Poland.

Ilkay E Orhan (I)

Department of Pharmacognosy, Faculty of Pharmacy, Gazi University, 06330 Ankara, Turkey.

Adam Matkowski (A)

Department of Pharmaceutical Biology and Botany, Wroclaw Medical University, 50556 Wroclaw, Poland.

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Classifications MeSH