MOMENTUM: A Phase I Trial Investigating 2 Schedules of Capecitabine With Aflibercept in Patients With Gastrointestinal and Breast Cancer.


Journal

Clinical colorectal cancer
ISSN: 1938-0674
Titre abrégé: Clin Colorectal Cancer
Pays: United States
ID NLM: 101120693

Informations de publication

Date de publication:
12 2020
Historique:
received: 23 03 2020
revised: 16 05 2020
accepted: 22 05 2020
pubmed: 8 7 2020
medline: 23 11 2021
entrez: 8 7 2020
Statut: ppublish

Résumé

Although data from preclinical and clinical studies provide a strong rationale for combining capecitabine with anti-angiogenic agents, clinical development of this fluoropyrimidine in combination with aflibercept has lagged behind other treatments. We conducted a nonrandomized, noncomparative, 2-arm, phase I trial to address this unmet need. Patients with chemorefractory gastrointestinal and breast cancer were sequentially recruited into a continuous (Arm A, starting dose 1100 mg/m Thirty-eight eligible patients were recruited of whom 33 were assessable for DLTs (15 in arm A and 18 in arm B). Fourteen had colorectal cancer, 8 gastric cancer, and 11 breast cancer. DLTs included grade 2 hand-foot syndrome, grade 2 anorexia considered unacceptable by the patient, and grade 3 hypertension. The recommended dose for phase II trials for capecitabine was established at 1300 mg/m Combining capecitabine with aflibercept is feasible and associated with a manageable safety profile and some anti-tumor activity in patients with chemorefractory gastrointestinal and breast cancer.

Sections du résumé

BACKGROUND
Although data from preclinical and clinical studies provide a strong rationale for combining capecitabine with anti-angiogenic agents, clinical development of this fluoropyrimidine in combination with aflibercept has lagged behind other treatments. We conducted a nonrandomized, noncomparative, 2-arm, phase I trial to address this unmet need.
PATIENTS AND METHODS
Patients with chemorefractory gastrointestinal and breast cancer were sequentially recruited into a continuous (Arm A, starting dose 1100 mg/m
RESULTS
Thirty-eight eligible patients were recruited of whom 33 were assessable for DLTs (15 in arm A and 18 in arm B). Fourteen had colorectal cancer, 8 gastric cancer, and 11 breast cancer. DLTs included grade 2 hand-foot syndrome, grade 2 anorexia considered unacceptable by the patient, and grade 3 hypertension. The recommended dose for phase II trials for capecitabine was established at 1300 mg/m
CONCLUSION
Combining capecitabine with aflibercept is feasible and associated with a manageable safety profile and some anti-tumor activity in patients with chemorefractory gastrointestinal and breast cancer.

Identifiants

pubmed: 32631787
pii: S1533-0028(20)30080-3
doi: 10.1016/j.clcc.2020.05.007
pii:
doi:

Substances chimiques

Recombinant Fusion Proteins 0
aflibercept 15C2VL427D
Capecitabine 6804DJ8Z9U
Receptors, Vascular Endothelial Growth Factor EC 2.7.10.1

Banques de données

ClinicalTrials.gov
['NCT01843725']
EudraCT
['2012-005169-11']

Types de publication

Clinical Trial, Phase I Journal Article

Langues

eng

Sous-ensembles de citation

IM

Pagination

311-318.e1

Informations de copyright

Copyright © 2020 Elsevier Inc. All rights reserved.

Auteurs

Silvia Camera (S)

Department of Medical Oncology, Institut Jules Bordet, Université Libre de Bruxelles (ULB), Brussels, Belgium.

Amélie Deleporte (A)

Department of Medical Oncology, Institut Jules Bordet, Université Libre de Bruxelles (ULB), Brussels, Belgium.

Giacomo Bregni (G)

Department of Medical Oncology, Institut Jules Bordet, Université Libre de Bruxelles (ULB), Brussels, Belgium.

Elena Trevisi (E)

Department of Medical Oncology, Institut Jules Bordet, Université Libre de Bruxelles (ULB), Brussels, Belgium.

Andrea Pretta (A)

Department of Medical Oncology, Institut Jules Bordet, Université Libre de Bruxelles (ULB), Brussels, Belgium.

Tugba Akin Telli (TA)

Department of Medical Oncology, Institut Jules Bordet, Université Libre de Bruxelles (ULB), Brussels, Belgium.

Laura Polastro (L)

Department of Medical Oncology, Institut Jules Bordet, Université Libre de Bruxelles (ULB), Brussels, Belgium.

Andrea Gombos (A)

Department of Medical Oncology, Institut Jules Bordet, Université Libre de Bruxelles (ULB), Brussels, Belgium.

Aline Kayumba (A)

Data Centre, Institut Jules Bordet, Université Libre de Bruxelles (ULB), Brussels, Belgium.

Lieveke Ameye (L)

Data Centre, Institut Jules Bordet, Université Libre de Bruxelles (ULB), Brussels, Belgium.

Martine Piccart-Gebhart (M)

Department of Medical Oncology, Institut Jules Bordet, Université Libre de Bruxelles (ULB), Brussels, Belgium.

Ahmad Awada (A)

Department of Medical Oncology, Institut Jules Bordet, Université Libre de Bruxelles (ULB), Brussels, Belgium.

Francesco Sclafani (F)

Department of Medical Oncology, Institut Jules Bordet, Université Libre de Bruxelles (ULB), Brussels, Belgium. Electronic address: francesco.sclafani@bordet.be.

Alain Hendlisz (A)

Department of Medical Oncology, Institut Jules Bordet, Université Libre de Bruxelles (ULB), Brussels, Belgium.

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Classifications MeSH