Canagliflozin and cardiovascular outcomes in Type 2 diabetes.


Journal

Future cardiology
ISSN: 1744-8298
Titre abrégé: Future Cardiol
Pays: England
ID NLM: 101239345

Informations de publication

Date de publication:
01 2021
Historique:
pubmed: 5 8 2020
medline: 26 10 2021
entrez: 5 8 2020
Statut: ppublish

Résumé

SGLT2 inhibitors have risen to prominence in recent years as Type 2 diabetes mellitus medications with favorable effects on cardiovascular (CV) and renal outcomes. Canagliflozin is a US FDA-approved SGLT2 inhibitor that has demonstrated CV and renal outcome benefits in large scale placebo-controlled randomized trials of patients with Type 2 diabetes mellitus and elevated CV risk. Canagliflozin use may also be associated with serious and nonserious adverse effects requiring ongoing monitoring in patients initiated on this medication. This paper provides a detailed overview of canagliflozin including its pharmacologic profile, clinical efficacy and safety data, with discussion of both clinical trial results, as well as real-world evidence.

Identifiants

pubmed: 32748638
doi: 10.2217/fca-2020-0029
pmc: PMC8656317
doi:

Substances chimiques

Hypoglycemic Agents 0
Sodium-Glucose Transporter 2 Inhibitors 0
Canagliflozin 0SAC974Z85

Types de publication

Journal Article Research Support, Non-U.S. Gov't

Langues

eng

Sous-ensembles de citation

IM

Pagination

39-48

Subventions

Organisme : NHLBI NIH HHS
ID : K01 HL144607
Pays : United States

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Auteurs

Ashish Sarraju (A)

Division of Cardiovascular Medicine & Cardiovascular Institute, Stanford University School of Medicine, Stanford, CA 94305, USA.

Gabriela Spencer-Bonilla (G)

Department of Medicine, Stanford University School of Medicine, Stanford, CA 94305, USA.

Fatima Rodriguez (F)

Division of Cardiovascular Medicine & Cardiovascular Institute, Stanford University School of Medicine, Stanford, CA 94305, USA.

Kenneth W Mahaffey (KW)

Division of Cardiovascular Medicine & Cardiovascular Institute, Stanford University School of Medicine, Stanford, CA 94305, USA.
Stanford Center for Clinical Research, Stanford, CA 94304, USA.

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Classifications MeSH