Consensus-Based Pharmacophore Mapping for New Set of

CoMSA IVE-PLS MIC MTT assay antistaphylococcal activity antitubercular activity hydroxynaphthalenecarboxamides lipophilicity similarity-activity landscape index

Journal

International journal of molecular sciences
ISSN: 1422-0067
Titre abrégé: Int J Mol Sci
Pays: Switzerland
ID NLM: 101092791

Informations de publication

Date de publication:
09 Sep 2020
Historique:
received: 03 08 2020
revised: 01 09 2020
accepted: 07 09 2020
entrez: 12 9 2020
pubmed: 13 9 2020
medline: 6 3 2021
Statut: epublish

Résumé

A series of twenty-two novel

Identifiants

pubmed: 32916824
pii: ijms21186583
doi: 10.3390/ijms21186583
pmc: PMC7555178
pii:
doi:

Substances chimiques

Anti-Infective Agents 0
Naphthalenes 0
naphthalene-2-carboxamide 0

Types de publication

Journal Article

Langues

eng

Sous-ensembles de citation

IM

Références

J Comput Aided Mol Des. 2008 Feb;22(2):81-9
pubmed: 18189157
Future Sci OA. 2019 Jan 18;5(2):FSO363
pubmed: 30828462
Bioorg Med Chem Lett. 2016 Aug 15;26(16):3862-5
pubmed: 27432762
SAR QSAR Environ Res. 2009;20(3-4):241-66
pubmed: 19544191
J Chem Inf Model. 2006 Nov-Dec;46(6):2310-8
pubmed: 17125174
Methods Mol Biol. 2011;672:39-100
pubmed: 20838964
Drug Discov Today. 2003 Jul 1;8(13):594-602
pubmed: 12850335
Bioorg Med Chem. 2013 Nov 1;21(21):6574-81
pubmed: 24045008
Curr Med Chem. 2018;25(38):4972-5006
pubmed: 28925868
Methods Mol Biol. 2013;930:3-27
pubmed: 23086835
Nat Rev Drug Discov. 2012 Apr 30;11(5):355-65
pubmed: 22543468
Anal Chem. 1996 Nov 1;68(21):3851-8
pubmed: 21619260
SAR QSAR Environ Res. 2017 Jun;28(6):427-449
pubmed: 28573881
J Chem Inf Model. 2008 Mar;48(3):465-75
pubmed: 18302356
J Chem Inf Model. 2007 Jul-Aug;47(4):1469-80
pubmed: 17567123
Future Med Chem. 2009 Jun;1(3):451-66
pubmed: 21426126
Molecules. 2019 Aug 18;24(16):
pubmed: 31426567
Molecules. 2017 Nov 14;22(11):
pubmed: 29135926
J Chem Inf Comput Sci. 2004 Jul-Aug;44(4):1423-35
pubmed: 15272850
PLoS Pathog. 2010 Apr 08;6(4):e1000855
pubmed: 20386717
Bioorg Med Chem. 2015 May 1;23(9):2035-43
pubmed: 25819330
Molecules. 2017 Oct 12;22(10):
pubmed: 29023407
Molecules. 2011 Mar 14;16(3):2414-30
pubmed: 21403599
J Comput Aided Mol Des. 2003 Feb-Apr;17(2-4):83-92
pubmed: 13677477
Int J Mol Sci. 2020 May 12;21(10):
pubmed: 32408543
Molecules. 2013 Jul 08;18(7):7977-97
pubmed: 23884130
Med Chem. 2015;11(2):156-64
pubmed: 25134428
Nat Rev Drug Discov. 2003 Mar;2(3):192-204
pubmed: 12612645
Drug Discov Today. 2009 Jul;14(13-14):698-705
pubmed: 19410012
Int J Tuberc Lung Dis. 1998 Dec;2(12):1011-6
pubmed: 9869118
Eur J Pharm Sci. 2015 Sep 18;77:197-207
pubmed: 26079401
SAR QSAR Environ Res. 2018 Oct;29(10):801-821
pubmed: 30230355
Molecules. 2018 Dec 11;23(12):
pubmed: 30544967
Drug Discov Today. 2000 Feb;5(2):49-58
pubmed: 10652455
Bioorg Med Chem. 2013 Nov 1;21(21):6531-41
pubmed: 24075143
Bioorg Med Chem Lett. 2017 May 1;27(9):1881-1885
pubmed: 28363749
Int J Mol Sci. 2019 Oct 29;20(21):
pubmed: 31671776
Curr Opin Chem Biol. 2004 Jun;8(3):255-63
pubmed: 15183323
Bioorg Med Chem. 2015 Aug 1;23(15):4188-4196
pubmed: 26183541
J Chem Inf Model. 2008 Aug;48(8):1716-28
pubmed: 18686944
J Cheminform. 2009 Jun 10;1(1):8
pubmed: 20298526
Bioorg Med Chem Lett. 2011 Aug 1;21(15):4564-7
pubmed: 21724391
Trends Pharmacol Sci. 2006 Mar;27(3):149-57
pubmed: 16483674
Molecules. 2015 May 27;20(6):9767-87
pubmed: 26023938
J Chem Inf Model. 2005 Sep-Oct;45(5):1447-55
pubmed: 16180922
Molecules. 2013 Aug 06;18(8):9397-419
pubmed: 23924993
J Innate Immun. 2016;8(2):111-20
pubmed: 26845587
Curr Comput Aided Drug Des. 2012 Jun;8(2):107-27
pubmed: 22497466
Int J Mol Sci. 2016 Jul 28;17(8):
pubmed: 27483236
Int J Mol Sci. 2018 Aug 07;19(8):
pubmed: 30087309
Molecules. 2016 Aug 16;21(8):
pubmed: 27537867
J Chem Inf Comput Sci. 2003 May-Jun;43(3):819-28
pubmed: 12767139
Sci Rep. 2019 Apr 23;9(1):6387
pubmed: 31011161
Diagn Microbiol Infect Dis. 2002 Dec;44(4):363-6
pubmed: 12543542
J Mol Graph Model. 2002 Jan;20(4):269-76
pubmed: 11858635

Auteurs

Andrzej Bak (A)

Department of Chemistry, University of Silesia, Szkolna 9, 40007 Katowice, Poland.

Jiri Kos (J)

Division of Biologically Active Complexes and Molecular Magnets, Regional Centre of Advanced Technologies and Materials, Faculty of Science, Palacky University, Slechtitelu 27, 78371 Olomouc, Czech Republic.

Hana Michnova (H)

Division of Biologically Active Complexes and Molecular Magnets, Regional Centre of Advanced Technologies and Materials, Faculty of Science, Palacky University, Slechtitelu 27, 78371 Olomouc, Czech Republic.

Tomas Gonec (T)

Department of Chemical Drugs, Faculty of Pharmacy, Masaryk University, Palackeho 1, 60200 Brno, Czech Republic.

Sarka Pospisilova (S)

Division of Biologically Active Complexes and Molecular Magnets, Regional Centre of Advanced Technologies and Materials, Faculty of Science, Palacky University, Slechtitelu 27, 78371 Olomouc, Czech Republic.

Violetta Kozik (V)

Department of Chemistry, University of Silesia, Szkolna 9, 40007 Katowice, Poland.

Alois Cizek (A)

Department of Infectious Diseases and Microbiology, Faculty of Veterinary Medicine, University of Veterinary and Pharmaceutical Sciences, Palackeho 1946/1, 61242 Brno, Czech Republic.

Adam Smolinski (A)

Central Mining Institute, Pl. Gwarków 1, 40-166 Katowice, Poland.

Josef Jampilek (J)

Division of Biologically Active Complexes and Molecular Magnets, Regional Centre of Advanced Technologies and Materials, Faculty of Science, Palacky University, Slechtitelu 27, 78371 Olomouc, Czech Republic.

Articles similaires

Vancomycin Polyesters Anti-Bacterial Agents Models, Theoretical Drug Liberation
Biofilms Candida albicans Quorum Sensing Candida glabrata Menthol

Two codependent routes lead to high-level MRSA.

Abimbola Feyisara Adedeji-Olulana, Katarzyna Wacnik, Lucia Lafage et al.
1.00
Methicillin-Resistant Staphylococcus aureus Penicillin-Binding Proteins Peptidoglycan Bacterial Proteins Anti-Bacterial Agents

Naturally derived 3-aminoquinuclidine salts as new promising therapeutic agents.

Doris Crnčević, Alma Ramić, Andreja Radman Kastelic et al.
1.00
Humans Microbial Sensitivity Tests Anti-Bacterial Agents Biofilms Quinuclidines

Classifications MeSH