The FABP12/PPARγ pathway promotes metastatic transformation by inducing epithelial-to-mesenchymal transition and lipid-derived energy production in prostate cancer cells.


Journal

Molecular oncology
ISSN: 1878-0261
Titre abrégé: Mol Oncol
Pays: United States
ID NLM: 101308230

Informations de publication

Date de publication:
12 2020
Historique:
received: 15 05 2020
revised: 11 08 2020
accepted: 05 10 2020
pubmed: 9 10 2020
medline: 4 9 2021
entrez: 8 10 2020
Statut: ppublish

Résumé

Early stage localized prostate cancer (PCa) has an excellent prognosis; however, patient survival drops dramatically when PCa metastasizes. The molecular mechanisms underlying PCa metastasis are complex and remain unclear. Here, we examine the role of a new member of the fatty acid-binding protein (FABP) family, FABP12, in PCa progression. FABP12 is preferentially amplified and/or overexpressed in metastatic compared to primary tumors from both PCa patients and xenograft animal models. We show that FABP12 concurrently triggers metastatic phenotypes (induced epithelial-to-mesenchymal transition (EMT) leading to increased cell motility and invasion) and lipid bioenergetics (increased fatty acid uptake and accumulation, increased ATP production from fatty acid β-oxidation) in PCa cells, supporting increased reliance on fatty acids for energy production. Mechanistically, we show that FABP12 is a driver of PPARγ activation which, in turn, regulates FABP12's role in lipid metabolism and PCa progression. Our results point to a novel role for a FABP-PPAR pathway in promoting PCa metastasis through induction of EMT and lipid bioenergetics.

Identifiants

pubmed: 33031638
doi: 10.1002/1878-0261.12818
pmc: PMC7718947
doi:

Substances chimiques

FABP12 protein, human 0
Fatty Acid-Binding Proteins 0
Lipids 0
PPAR gamma 0

Types de publication

Journal Article Research Support, Non-U.S. Gov't

Langues

eng

Sous-ensembles de citation

IM

Pagination

3100-3120

Informations de copyright

© 2020 The Authors. Published by FEBS Press and John Wiley & Sons Ltd.

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Auteurs

Rong-Zong Liu (RZ)

Department of Oncology, Cross Cancer Institute, University of Alberta, Edmonton, AB, Canada.

Won-Shik Choi (WS)

Department of Oncology, Cross Cancer Institute, University of Alberta, Edmonton, AB, Canada.

Saket Jain (S)

Department of Oncology, Cross Cancer Institute, University of Alberta, Edmonton, AB, Canada.

Deepak Dinakaran (D)

Department of Oncology, Cross Cancer Institute, University of Alberta, Edmonton, AB, Canada.

Xia Xu (X)

Department of Oncology, Cross Cancer Institute, University of Alberta, Edmonton, AB, Canada.

Woo Hyun Han (WH)

Faculty Saint-Jean, University of Alberta, Edmonton, AB, Canada.

Xiao-Hong Yang (XH)

Department of Oncology, Cross Cancer Institute, University of Alberta, Edmonton, AB, Canada.

Darryl D Glubrecht (DD)

Department of Oncology, Cross Cancer Institute, University of Alberta, Edmonton, AB, Canada.

Ronald B Moore (RB)

Department of Oncology, Cross Cancer Institute, University of Alberta, Edmonton, AB, Canada.
Department of Surgery, University of Alberta, Edmonton, AB, Canada.

Hélène Lemieux (H)

Faculty Saint-Jean, University of Alberta, Edmonton, AB, Canada.

Roseline Godbout (R)

Department of Oncology, Cross Cancer Institute, University of Alberta, Edmonton, AB, Canada.

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