Benzoxaboroles: New Potent Inhibitors of the Carbonic Anhydrases of the Pathogenic Bacterium


Journal

ACS medicinal chemistry letters
ISSN: 1948-5875
Titre abrégé: ACS Med Chem Lett
Pays: United States
ID NLM: 101521073

Informations de publication

Date de publication:
12 Nov 2020
Historique:
received: 20 07 2020
accepted: 09 09 2020
entrez: 20 11 2020
pubmed: 21 11 2020
medline: 21 11 2020
Statut: epublish

Résumé

A series of urea/thiourea substituted benzoxaboroles was investigated for the inhibition of the three carbonic anhydrases encoded by

Identifiants

pubmed: 33214840
doi: 10.1021/acsmedchemlett.0c00403
pmc: PMC7667823
doi:

Types de publication

Journal Article

Langues

eng

Pagination

2277-2284

Déclaration de conflit d'intérêts

The authors declare no competing financial interest.

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Auteurs

Alessandro Bonardi (A)

Department of NEUROFARBA, Section of Pharmaceutical and Nutraceutical Sciences, University of Florence, 50121 Florence, Italy.
Department of NEUROFARBA, Section of Pharmaceutical and Nutraceutical Sciences, Laboratory of Molecular Modeling Cheminformatics & QSAR, University of Florence, 50121 Florence, Italy.

Alessio Nocentini (A)

Department of NEUROFARBA, Section of Pharmaceutical and Nutraceutical Sciences, Laboratory of Molecular Modeling Cheminformatics & QSAR, University of Florence, 50121 Florence, Italy.
IBMM, Univ Montpellier, CNRS, ENSCM, 34296 Montpellier, France.

Roberta Cadoni (R)

IBMM, Univ Montpellier, CNRS, ENSCM, 34296 Montpellier, France.

Sonia Del Prete (S)

Istituto di Bioscienze e Biorisorse, CNR, Via Pietro Castellino 111, 80131 Napoli, Italy.

Pascal Dumy (P)

IBMM, Univ Montpellier, CNRS, ENSCM, 34296 Montpellier, France.

Clemente Capasso (C)

Istituto di Bioscienze e Biorisorse, CNR, Via Pietro Castellino 111, 80131 Napoli, Italy.

Paola Gratteri (P)

Department of NEUROFARBA, Section of Pharmaceutical and Nutraceutical Sciences, Laboratory of Molecular Modeling Cheminformatics & QSAR, University of Florence, 50121 Florence, Italy.

Claudiu T Supuran (CT)

Department of NEUROFARBA, Section of Pharmaceutical and Nutraceutical Sciences, University of Florence, 50121 Florence, Italy.

Jean-Yves Winum (JY)

IBMM, Univ Montpellier, CNRS, ENSCM, 34296 Montpellier, France.

Classifications MeSH