MAHOGANY: margetuximab combination in HER2+ unresectable/metastatic gastric/gastroesophageal junction adenocarcinoma.


Journal

Future oncology (London, England)
ISSN: 1744-8301
Titre abrégé: Future Oncol
Pays: England
ID NLM: 101256629

Informations de publication

Date de publication:
Apr 2021
Historique:
pubmed: 3 12 2020
medline: 16 10 2021
entrez: 2 12 2020
Statut: ppublish

Résumé

Standard-of-care, first-line therapy for patients with advanced HER2+ gastric/gastroesophageal junction adenocarcinoma is chemotherapy plus trastuzumab, a monoclonal antibody (mAb) targeting HER2. Margetuximab is an Fc-optimized mAb that binds HER2. Retifanlimab, a humanized IgG4 mAb, binds to PD-1 and blocks its interaction with PD-L1/2. Tebotelimab, an IgG4κ bispecific DART

Identifiants

pubmed: 33263418
doi: 10.2217/fon-2020-1007
doi:

Substances chimiques

Antibodies, Monoclonal 0
Biomarkers, Tumor 0
Receptor, ErbB-2 EC 2.7.10.1
margetuximab K911R84KEW

Banques de données

ClinicalTrials.gov
['NCT04082364']

Types de publication

Clinical Trial, Phase II Clinical Trial, Phase III Journal Article Randomized Controlled Trial

Langues

eng

Sous-ensembles de citation

IM

Pagination

1155-1164

Subventions

Organisme : MacroGenics, Inc.

Auteurs

Daniel Vt Catenacci (DV)

Department of Medicine, Section of Hematology & Oncology, University of Chicago, Chicago, IL 60637, USA.

Minori Rosales (M)

Clinical Research, MacroGenics, Inc., Rockville, MD 20850, USA.

Hyun Cheol Chung (HC)

Yonsei Cancer Center, University College of Medicine, Seoul 03722, Korea.

Harry H Yoon (H)

Mayo Clinic Cancer Center, Rochester, MN 55905, USA.

Lin Shen (L)

Peking University Cancer Hospital & Institute, Beijing 100142, China.

Markus Moehler (M)

University Medical Center Mainz, Mainz 55131, Germany.

Yoon-Koo Kang (YK)

Asan Medical Center, University of Ulsan College of Medicine, Seoul 05505, Korea.

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Classifications MeSH