Mutation-specific effects of NRAS oncogenes in colorectal cancer cells.


Journal

Advances in biological regulation
ISSN: 2212-4934
Titre abrégé: Adv Biol Regul
Pays: England
ID NLM: 101572336

Informations de publication

Date de publication:
01 2021
Historique:
received: 07 12 2020
accepted: 21 12 2020
pubmed: 13 1 2021
medline: 28 10 2021
entrez: 12 1 2021
Statut: ppublish

Résumé

In colorectal cancer (CRC), the prevalence of NRAS mutations (5-9%) is inferior to that of KRAS mutations (40-50%). NRAS mutations feature lately during tumour progression and drive resistance to anti-EGFR therapy in KRAS wild-type tumours. To elucidate specific functions of NRAS mutations in CRC, we expressed doxycycline-inducible G12D and Q61K mutations in the CRC cell line Caco-2. A focused phospho-proteome analysis based on the Bio-Plex platform, which interrogated the activity of MAPK, PI3K, mTOR, STAT, p38, JNK and ATF2, did not reveal significant differences between Caco-2 cells expressing NRAS

Identifiants

pubmed: 33431353
pii: S2212-4926(20)30089-0
doi: 10.1016/j.jbior.2020.100778
pii:
doi:

Substances chimiques

Chemokines 0
Cytokines 0
Membrane Proteins 0
GTP Phosphohydrolases EC 3.6.1.-
NRAS protein, human EC 3.6.1.-

Types de publication

Journal Article Research Support, Non-U.S. Gov't

Langues

eng

Sous-ensembles de citation

IM

Pagination

100778

Informations de copyright

Copyright © 2020. Published by Elsevier Ltd.

Auteurs

Natalia Kuhn (N)

Laboratory of Molecular Tumor Pathology and Cancer Systems Biology, Institute of Pathology, Charité Universitätsmedizin Berlin, Charitéplatz 1, D-10117, Berlin, Germany.

Bertram Klinger (B)

Laboratory of Molecular Tumor Pathology and Cancer Systems Biology, Institute of Pathology, Charité Universitätsmedizin Berlin, Charitéplatz 1, D-10117, Berlin, Germany; Integrative Research Institute Life Sciences, Humboldt University Berlin, Philippstraße 13, Building 18, D-10115, Berlin, Germany.

Florian Uhlitz (F)

Laboratory of Molecular Tumor Pathology and Cancer Systems Biology, Institute of Pathology, Charité Universitätsmedizin Berlin, Charitéplatz 1, D-10117, Berlin, Germany; Integrative Research Institute Life Sciences, Humboldt University Berlin, Philippstraße 13, Building 18, D-10115, Berlin, Germany.

Anja Sieber (A)

Laboratory of Molecular Tumor Pathology and Cancer Systems Biology, Institute of Pathology, Charité Universitätsmedizin Berlin, Charitéplatz 1, D-10117, Berlin, Germany; Integrative Research Institute Life Sciences, Humboldt University Berlin, Philippstraße 13, Building 18, D-10115, Berlin, Germany.

Maria Rivera (M)

Experimental Pharmacology and Oncology GmbH, Berlin-Buch, Robert-Rössle-Str. 10, D-13125, Berlin, Buch, Germany.

Kathleen Klotz-Noack (K)

Laboratory of Molecular Tumor Pathology and Cancer Systems Biology, Institute of Pathology, Charité Universitätsmedizin Berlin, Charitéplatz 1, D-10117, Berlin, Germany.

Iduna Fichtner (I)

Experimental Pharmacology and Oncology GmbH, Berlin-Buch, Robert-Rössle-Str. 10, D-13125, Berlin, Buch, Germany.

Jens Hoffmann (J)

Experimental Pharmacology and Oncology GmbH, Berlin-Buch, Robert-Rössle-Str. 10, D-13125, Berlin, Buch, Germany.

Nils Blüthgen (N)

Laboratory of Molecular Tumor Pathology and Cancer Systems Biology, Institute of Pathology, Charité Universitätsmedizin Berlin, Charitéplatz 1, D-10117, Berlin, Germany; Integrative Research Institute Life Sciences, Humboldt University Berlin, Philippstraße 13, Building 18, D-10115, Berlin, Germany.

Christine Falk (C)

Institute of Transplant Immunology, Hannover Medical School, Carl-Neuberg-Str. 1, D-30625, Hannover, Germany.

Christine Sers (C)

Laboratory of Molecular Tumor Pathology and Cancer Systems Biology, Institute of Pathology, Charité Universitätsmedizin Berlin, Charitéplatz 1, D-10117, Berlin, Germany; German Cancer Consortium (DKTK), German Cancer Research Center, Im Neuenheimer Feld 280, D-69120, Heidelberg, Germany. Electronic address: christine.sers@charite.de.

Reinhold Schäfer (R)

Laboratory of Molecular Tumor Pathology and Cancer Systems Biology, Institute of Pathology, Charité Universitätsmedizin Berlin, Charitéplatz 1, D-10117, Berlin, Germany; German Cancer Consortium (DKTK), German Cancer Research Center, Im Neuenheimer Feld 280, D-69120, Heidelberg, Germany; Comprehensive Cancer Center, Charité Universitätsmedizin Berlin, Charitéplatz 1, D-10117, Berlin, Germany. Electronic address: reinhold.schaefer@charite.de.

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Classifications MeSH