Transient receptor potential vanilloid 4 channel participates in mouse ventricular electrical activity.
Action Potentials
/ drug effects
Animals
Calcium Channels, L-Type
/ metabolism
Calcium Signaling
/ drug effects
Computer Simulation
HEK293 Cells
Heart Rate
/ drug effects
Humans
Leucine
/ analogs & derivatives
Male
Mice, Inbred C57BL
Mice, Knockout
Models, Cardiovascular
Myocytes, Cardiac
/ drug effects
Piperidines
/ pharmacology
Quinolines
/ pharmacology
Sulfonamides
/ pharmacology
TRPV Cation Channels
/ deficiency
Time Factors
Ventricular Function, Left
/ drug effects
QT interval
TRPV4 channel
action potential
calcium transient
mathematical modeling
trpv4
trpv4−/−
Journal
American journal of physiology. Heart and circulatory physiology
ISSN: 1522-1539
Titre abrégé: Am J Physiol Heart Circ Physiol
Pays: United States
ID NLM: 100901228
Informations de publication
Date de publication:
01 03 2021
01 03 2021
Historique:
pubmed:
16
1
2021
medline:
23
3
2021
entrez:
15
1
2021
Statut:
ppublish
Résumé
The TRPV4 channel is a calcium-permeable channel (
Identifiants
pubmed: 33449852
doi: 10.1152/ajpheart.00497.2020
doi:
Substances chimiques
Calcium Channels, L-Type
0
GSK2193874
0
N-(1-((4-(2-(((2,4-dichlorophenyl)sulfonyl)amino)-3-hydroxypropanoyl)-1-piperazinyl)carbonyl)-3-methylbutyl)-1-benzothiophene-2-carboxamide
0
Piperidines
0
Quinolines
0
Sulfonamides
0
TRPV Cation Channels
0
TRPV4 protein, human
0
Trpv4 protein, mouse
0
Leucine
GMW67QNF9C
Types de publication
Journal Article
Research Support, Non-U.S. Gov't
Langues
eng
Sous-ensembles de citation
IM