Pharmacokinetic equivalence of CT-P17 to high-concentration (100 mg/ml) reference adalimumab: A randomized phase I study in healthy subjects.


Journal

Clinical and translational science
ISSN: 1752-8062
Titre abrégé: Clin Transl Sci
Pays: United States
ID NLM: 101474067

Informations de publication

Date de publication:
07 2021
Historique:
revised: 02 11 2020
received: 29 09 2020
accepted: 09 12 2020
pubmed: 28 1 2021
medline: 15 2 2022
entrez: 27 1 2021
Statut: ppublish

Résumé

This study aimed to demonstrate pharmacokinetic (PK) equivalence of a single dose of the proposed adalimumab biosimilar CT-P17 to United States-licensed adalimumab (US-adalimumab) and European Union-approved adalimumab (EU-adalimumab). This double-blind, parallel-group, phase I trial (clinicaltrials.gov NCT03970824) was conducted at 10 hospitals (Republic of Korea), in which healthy subjects (1:1:1) were randomized to receive a single 40 mg (100 mg/ml) subcutaneous injection of CT-P17, US-adalimumab, or EU-adalimumab. Primary end points were PK equivalence in terms of: area under the concentration-time curve from time zero to infinity (AUC

Identifiants

pubmed: 33503313
doi: 10.1111/cts.12967
pmc: PMC8301575
doi:

Substances chimiques

Adalimumab FYS6T7F842
Biosimilar Pharmaceuticals 0
Tumor Necrosis Factor Inhibitors 0
CT-P17 0

Banques de données

ClinicalTrials.gov
['NCT03970824']

Types de publication

Clinical Trial, Phase I Equivalence Trial Journal Article Multicenter Study Randomized Controlled Trial Research Support, Non-U.S. Gov't

Langues

eng

Sous-ensembles de citation

IM

Pagination

1280-1291

Subventions

Organisme : Celltrion, Inc.

Informations de copyright

© 2021 Celltrion, Inc. Clinical and Translational Science published by Wiley Periodicals LLC on behalf of the American Society for Clinical Pharmacology and Therapeutics.

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Auteurs

Kyung-Sang Yu (KS)

Seoul National University College of Medicine and Hospital, Seoul, Korea.

In-Jin Jang (IJ)

Seoul National University College of Medicine and Hospital, Seoul, Korea.

Hyeong-Seok Lim (HS)

Asan Medical Center, College of Medicine, University of Ulsan, Seoul, Korea.

Jang Hee Hong (JH)

Chungnam National University Hospital, Daejeon, Korea.

Min-Gul Kim (MG)

College of Medicine, Jeonbuk National University, Jeonbuk, Korea.

Min Kyu Park (MK)

Chungbuk National University Hospital, Cheongju, Korea.

Doo-Yeoun Cho (DY)

CHA Bundang Medical Center, CHA University, Seongnam, Korea.

Min Soo Park (MS)

Severance Hospital, Yonsei University College of Medicine, Seoul, Korea.

Jae Yong Chung (JY)

Seoul National University Bundang Hospital, Seongnam, Korea.

Jong-Lyul Ghim (JL)

Inje University Busan Paik Hospital, Busan, Korea.

SeungHwan Lee (S)

Seoul National University College of Medicine and Hospital, Seoul, Korea.

Seok Kyu Yoon (SK)

Asan Medical Center, College of Medicine, University of Ulsan, Seoul, Korea.

In Sun Kwon (IS)

Chungnam National University Hospital, Daejeon, Korea.

Sang Joon Lee (SJ)

Celltrion, Inc., Incheon, Korea.

Sung Hyun Kim (SH)

Celltrion, Inc., Incheon, Korea.

Yun Ju Bae (YJ)

Celltrion, Inc., Incheon, Korea.

Jung Bin Cha (JB)

Celltrion, Inc., Incheon, Korea.

Daniel E Furst (DE)

University of California, Los Angeles, California, USA.
University of Washington, Seattle, Washington, USA.
University of Florence, Florence, Italy.

Edward Keystone (E)

Mount Sinai Hospital, University of Toronto, Toronto, Canada.

Jonathan Kay (J)

University of Massachusetts Medical School and UMass Memorial Medical Center, Worcester, Massachusetts, USA.

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Classifications MeSH