PDE4 inhibition as a therapeutic strategy for improvement of pulmonary dysfunctions in Covid-19 and cigarette smoking.
Angiotensin-Converting Enzyme Inhibitors
/ pharmacology
Animals
COVID-19
/ epidemiology
Cigarette Smoking
/ drug therapy
Humans
Lung
/ drug effects
Lung Diseases
/ drug therapy
Peptidyl-Dipeptidase A
/ metabolism
Phosphodiesterase 4 Inhibitors
/ pharmacology
Respiratory Distress Syndrome
/ drug therapy
COVID-19 Drug Treatment
Angiotensin-converting enzyme 2 (ACE2)
COVID-19
Cigarette smoking (CS)
Inflammation
PDE4
Respiratory epithelial cells
Journal
Biochemical pharmacology
ISSN: 1873-2968
Titre abrégé: Biochem Pharmacol
Pays: England
ID NLM: 0101032
Informations de publication
Date de publication:
03 2021
03 2021
Historique:
received:
23
11
2020
revised:
15
01
2021
accepted:
19
01
2021
pubmed:
31
1
2021
medline:
7
4
2021
entrez:
30
1
2021
Statut:
ppublish
Résumé
Angiotensin-converting enzyme 2 (ACE2) is the binding-site and entry-point for SARS-CoV-2 in human and highly expressed in the lung. Cigarette smoking (CS) is the leading cause of pulmonary and cardiovascular diseases. Chronic CS leads to upregulation of bronchial ACE2 inducing a high vulnerability in COVID-19 smoker patients. Interestingly, CS-induced dysregulation of pulmonary renin-angiotensin system (RAS) in part contributing into the potential pathogenesis COVID-19 pneumonia and acute respiratory distress syndrome (ARDS). Since, CS-mediated ACE2 activations is not the main pathway for increasing the risk of COVID-19, it appeared that AngII/AT
Identifiants
pubmed: 33515531
pii: S0006-2952(21)00027-7
doi: 10.1016/j.bcp.2021.114431
pmc: PMC7842152
pii:
doi:
Substances chimiques
Angiotensin-Converting Enzyme Inhibitors
0
Phosphodiesterase 4 Inhibitors
0
Peptidyl-Dipeptidase A
EC 3.4.15.1
Types de publication
Journal Article
Review
Langues
eng
Sous-ensembles de citation
IM
Pagination
114431Informations de copyright
Crown Copyright © 2021. Published by Elsevier Inc. All rights reserved.
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