A Bifunctional NAD


Journal

ACS chemical biology
ISSN: 1554-8937
Titre abrégé: ACS Chem Biol
Pays: United States
ID NLM: 101282906

Informations de publication

Date de publication:
19 02 2021
Historique:
pubmed: 2 2 2021
medline: 29 6 2021
entrez: 1 2 2021
Statut: ppublish

Résumé

Protein poly-ADP-ribosylation (PARylation) is a heterogeneous and dynamic post-translational modification regulated by various writers, readers, and erasers. It participates in a variety of biological events and is involved in many human diseases. Currently, tools and technologies have yet to be developed for unambiguously defining readers and erasers of individual PARylated proteins or cognate PARylated proteins for known readers and erasers. Here, we report the generation of a bifunctional nicotinamide adenine dinucleotide (NAD

Identifiants

pubmed: 33524253
doi: 10.1021/acschembio.0c00937
pmc: PMC7909001
mid: NIHMS1669996
doi:

Substances chimiques

Azides 0
Cross-Linking Reagents 0
Proteome 0
NAD 0U46U6E8UK
Diazomethane 60A625P70P
PARP1 protein, human EC 2.4.2.30
Poly (ADP-Ribose) Polymerase-1 EC 2.4.2.30

Types de publication

Journal Article Research Support, N.I.H., Extramural Research Support, Non-U.S. Gov't

Langues

eng

Sous-ensembles de citation

IM

Pagination

389-396

Subventions

Organisme : NIDDK NIH HHS
ID : P30 DK048522
Pays : United States
Organisme : NIGMS NIH HHS
ID : R35 GM137901
Pays : United States

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Auteurs

Albert T Lam (AT)

Department of Pharmacology and Pharmaceutical Sciences, School of Pharmacy, University of Southern California, Los Angeles, California 90089, United States.

Xiao-Nan Zhang (XN)

Department of Pharmacology and Pharmaceutical Sciences, School of Pharmacy, University of Southern California, Los Angeles, California 90089, United States.

Valentine V Courouble (VV)

Department of Molecular Medicine, The Scripps Research Institute, Jupiter, Florida 33458, United States.

Timothy S Strutzenberg (TS)

Department of Molecular Medicine, The Scripps Research Institute, Jupiter, Florida 33458, United States.

Hua Pei (H)

Titus Family Department of Clinical Pharmacy, School of Pharmacy, University of Southern California, Los Angeles, California 90089, United States.

Bangyan L Stiles (BL)

Department of Pharmacology and Pharmaceutical Sciences, School of Pharmacy, University of Southern California, Los Angeles, California 90089, United States.

Stan G Louie (SG)

Titus Family Department of Clinical Pharmacy, School of Pharmacy, University of Southern California, Los Angeles, California 90089, United States.

Patrick R Griffin (PR)

Department of Molecular Medicine, The Scripps Research Institute, Jupiter, Florida 33458, United States.

Yong Zhang (Y)

Department of Pharmacology and Pharmaceutical Sciences, School of Pharmacy, University of Southern California, Los Angeles, California 90089, United States.
Department of Chemistry, Dornsife College of Letters, Arts and Sciences, University of Southern California, Los Angeles, California 90089, United States.
Norris Comprehensive Cancer Center, University of Southern California, Los Angeles, California 90089, United States.
Research Center for Liver Diseases, University of Southern California, Los Angeles, California 90089, United States.

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Classifications MeSH