Pharmacological characterization of a new series of carbamoylguanidines reveals potent agonism at the H


Journal

European journal of medicinal chemistry
ISSN: 1768-3254
Titre abrégé: Eur J Med Chem
Pays: France
ID NLM: 0420510

Informations de publication

Date de publication:
15 Mar 2021
Historique:
received: 20 11 2020
revised: 31 12 2020
accepted: 08 01 2021
pubmed: 7 2 2021
medline: 1 5 2021
entrez: 6 2 2021
Statut: ppublish

Résumé

Even today, the role of the histamine H

Identifiants

pubmed: 33548637
pii: S0223-5234(21)00039-8
doi: 10.1016/j.ejmech.2021.113190
pii:
doi:

Substances chimiques

Dopamine Agonists 0
Guanidines 0
Ligands 0
Receptors, Dopamine D3 0
Receptors, Histamine H2 0

Types de publication

Journal Article

Langues

eng

Sous-ensembles de citation

IM

Pagination

113190

Informations de copyright

Copyright © 2021 Elsevier Masson SAS. All rights reserved.

Déclaration de conflit d'intérêts

Declaration of competing interest The authors declare that they have no known competing financial interests or personal relationships that could have appeared to influence the work reported in this paper.

Auteurs

Sabrina Biselli (S)

Institute of Pharmacy, University of Regensburg, Universitätsstraße 31, D-93053, Regensburg, Germany; Agrolab Labor GmbH, 84079, Bruckberg, Germany.

Merlin Bresinsky (M)

Institute of Pharmacy, University of Regensburg, Universitätsstraße 31, D-93053, Regensburg, Germany.

Katharina Tropmann (K)

Institute of Pharmacy, University of Regensburg, Universitätsstraße 31, D-93053, Regensburg, Germany.

Lisa Forster (L)

Institute of Pharmacy, University of Regensburg, Universitätsstraße 31, D-93053, Regensburg, Germany.

Claudia Honisch (C)

Institute of Pharmacy, University of Regensburg, Universitätsstraße 31, D-93053, Regensburg, Germany; Institute of Biomolecular Chemistry - National Research Council (ICB-CNR), Padua Unit Via F. Marzolo, 1, 35131, Padova, Italy.

Armin Buschauer (A)

Institute of Pharmacy, University of Regensburg, Universitätsstraße 31, D-93053, Regensburg, Germany.

Günther Bernhardt (G)

Institute of Pharmacy, University of Regensburg, Universitätsstraße 31, D-93053, Regensburg, Germany.

Steffen Pockes (S)

Institute of Pharmacy, University of Regensburg, Universitätsstraße 31, D-93053, Regensburg, Germany; Department of Neurology, University of Minnesota, Minneapolis, MN, 55455, USA; Department of Medicinal Chemistry, Institute for Therapeutics Discovery and Development, University of Minnesota, Minneapolis, MN, 55414, USA. Electronic address: steffen.pockes@ur.de.

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Classifications MeSH