Cannabidiol Inhibits SARS-CoV-2 Replication and Promotes the Host Innate Immune Response.


Journal

bioRxiv : the preprint server for biology
Titre abrégé: bioRxiv
Pays: United States
ID NLM: 101680187

Informations de publication

Date de publication:
10 Mar 2021
Historique:
entrez: 24 3 2021
pubmed: 25 3 2021
medline: 25 3 2021
Statut: epublish

Résumé

The rapid spread of COVID-19 underscores the need for new treatments. Here we report that cannabidiol (CBD), a compound produced by the cannabis plant, inhibits SARS-CoV-2 infection. CBD and its metabolite, 7-OH-CBD, but not congeneric cannabinoids, potently block SARS-CoV-2 replication in lung epithelial cells. CBD acts after cellular infection, inhibiting viral gene expression and reversing many effects of SARS-CoV-2 on host gene transcription. CBD induces interferon expression and up-regulates its antiviral signaling pathway. A cohort of human patients previously taking CBD had significantly lower SARS-CoV-2 infection incidence of up to an order of magnitude relative to matched pairs or the general population. This study highlights CBD, and its active metabolite, 7-OH-CBD, as potential preventative agents and therapeutic treatments for SARS-CoV-2 at early stages of infection.

Identifiants

pubmed: 33758843
doi: 10.1101/2021.03.10.432967
pmc: PMC7987002
pii:
doi:

Types de publication

Preprint

Langues

eng

Subventions

Organisme : NIAID NIH HHS
ID : R01 AI127518
Pays : United States
Organisme : NIGMS NIH HHS
ID : R35 GM119840
Pays : United States
Organisme : NCI NIH HHS
ID : R01 CA219815
Pays : United States
Organisme : NIAID NIH HHS
ID : R01 AI137514
Pays : United States
Organisme : NIGMS NIH HHS
ID : R01 GM121735
Pays : United States
Organisme : NIAID NIH HHS
ID : R01 AI134980
Pays : United States
Organisme : NCATS NIH HHS
ID : UL1 TR002389
Pays : United States
Organisme : NCI NIH HHS
ID : P30 CA014599
Pays : United States
Organisme : NCI NIH HHS
ID : R01 CA184494
Pays : United States

Commentaires et corrections

Type : UpdateIn

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Auteurs

Long Chi Nguyen (LC)

Ben May Department for Cancer Research, University of Chicago, Chicago, IL 60637.

Dongbo Yang (D)

Ben May Department for Cancer Research, University of Chicago, Chicago, IL 60637.

Vlad Nicolaescu (V)

Department of Microbiology, University of Chicago, Chicago, IL 60637.
Howard Taylor Ricketts Laboratory, Argonne National Laboratory, Lemont IL 60439.

Thomas J Best (TJ)

Center for Health and the Social Sciences, University of Chicago, Chicago IL 60637.

Takashi Ohtsuki (T)

College of Pharmacy, Pharmacognosy Institute, University of Illinois at Chicago, Chicago IL 60612.

Shao-Nong Chen (SN)

College of Pharmacy, Pharmacognosy Institute, University of Illinois at Chicago, Chicago IL 60612.

J Brent Friesen (JB)

College of Pharmacy, Pharmacognosy Institute, University of Illinois at Chicago, Chicago IL 60612.

Nir Drayman (N)

Pritzker School of Molecular Engineering, University of Chicago, Chicago IL 60637.

Adil Mohamed (A)

Pritzker School of Molecular Engineering, University of Chicago, Chicago IL 60637.

Christopher Dann (C)

Ben May Department for Cancer Research, University of Chicago, Chicago, IL 60637.

Diane Silva (D)

Department of Pathology, University of Chicago, Chicago IL 60637.

Haley Gula (H)

Department of Microbiology, University of Chicago, Chicago, IL 60637.
Howard Taylor Ricketts Laboratory, Argonne National Laboratory, Lemont IL 60439.

Krysten A Jones (KA)

Department of Chemistry, University of Chicago, Chicago IL 60637.

J Michael Millis (JM)

Department of Surgery, University of Chicago, Chicago IL 60637.

Bryan C Dickinson (BC)

Department of Chemistry, University of Chicago, Chicago IL 60637.

Savaş Tay (S)

Pritzker School of Molecular Engineering, University of Chicago, Chicago IL 60637.

Scott A Oakes (SA)

Department of Pathology, University of Chicago, Chicago IL 60637.

Guido F Pauli (GF)

College of Pharmacy, Pharmacognosy Institute, University of Illinois at Chicago, Chicago IL 60612.

David O Meltzer (DO)

Center for Health and the Social Sciences, University of Chicago, Chicago IL 60637.

Glenn Randall (G)

Department of Microbiology, University of Chicago, Chicago, IL 60637.
Howard Taylor Ricketts Laboratory, Argonne National Laboratory, Lemont IL 60439.

Marsha Rich Rosner (MR)

Ben May Department for Cancer Research, University of Chicago, Chicago, IL 60637.

Classifications MeSH