Interventional Study to Evaluate the Clinical Effects and Safety of the Nutraceutical Compound BrainUp-10® in a Cohort of Patients with Alzheimer's Disease: A Multicenter, Randomized, Double-Blind, and Placebo-Controlled Trial.


Journal

Journal of Alzheimer's disease : JAD
ISSN: 1875-8908
Titre abrégé: J Alzheimers Dis
Pays: Netherlands
ID NLM: 9814863

Informations de publication

Date de publication:
2021
Historique:
pubmed: 4 5 2021
medline: 18 9 2021
entrez: 3 5 2021
Statut: ppublish

Résumé

Clinically-evaluated nutraceuticals are candidates for Alzheimer's disease (AD) prevention and treatment. Phase I studies showed biological safety of the nutraceutical BrainUp-10®, while a pilot trial demonstrated efficacy for treatment. Cell studies demonstrated neuroprotection. BrainUp-10® blocks tau self-assembly. Apathy is the most common of behavioral alterations. The aim was to explore efficacy of BrainUp-10® in mitigating cognitive and behavioral symptoms and in providing life quality, in a cohort of Chilean patients with mild to moderate AD. The was a multicenter, randomized, double blind, placebo-controlled phase II clinical study in mild to moderate AD patients treated with BrainUp-10® daily, while controls received a placebo. Primary endpoint was Apathy (AES scale), while secondary endpoints included Mini-Mental State Examination (MMSE), Trail Making Test (TMT A and TMT B), and Neuropsychiatry Index (NPI). AD blood biomarkers were analyzed. Laboratory tests were applied to all subjects. 82 patients were enrolled. The MMSE score improved significantly at week 24 compared to baseline with tendency to increase, which met the pre-defined superiority criteria. NPI scores improved, the same for caregiver distress at 12th week (p = 0.0557), and the alimentary response (p = 0.0333). Apathy tests showed a statistically significant decrease in group treated with BrainUp-10®, with p = 0.0321 at week 4 and p = 0.0480 at week 12 treatment. A marked decrease in homocysteine was shown with BrainUp-10® (p = 0.0222). Data show that BrainUp-10® produces a statistically significant improvement in apathy, ameliorating neuropsychiatric distress of patients. There were no compound-related adverse events. BrainUp-10® technology may enable patients to receive the benefits for their cognitive and behavioral problems.

Sections du résumé

BACKGROUND
Clinically-evaluated nutraceuticals are candidates for Alzheimer's disease (AD) prevention and treatment. Phase I studies showed biological safety of the nutraceutical BrainUp-10®, while a pilot trial demonstrated efficacy for treatment. Cell studies demonstrated neuroprotection. BrainUp-10® blocks tau self-assembly. Apathy is the most common of behavioral alterations.
OBJECTIVE
The aim was to explore efficacy of BrainUp-10® in mitigating cognitive and behavioral symptoms and in providing life quality, in a cohort of Chilean patients with mild to moderate AD.
METHODS
The was a multicenter, randomized, double blind, placebo-controlled phase II clinical study in mild to moderate AD patients treated with BrainUp-10® daily, while controls received a placebo. Primary endpoint was Apathy (AES scale), while secondary endpoints included Mini-Mental State Examination (MMSE), Trail Making Test (TMT A and TMT B), and Neuropsychiatry Index (NPI). AD blood biomarkers were analyzed. Laboratory tests were applied to all subjects.
RESULTS
82 patients were enrolled. The MMSE score improved significantly at week 24 compared to baseline with tendency to increase, which met the pre-defined superiority criteria. NPI scores improved, the same for caregiver distress at 12th week (p = 0.0557), and the alimentary response (p = 0.0333). Apathy tests showed a statistically significant decrease in group treated with BrainUp-10®, with p = 0.0321 at week 4 and p = 0.0480 at week 12 treatment. A marked decrease in homocysteine was shown with BrainUp-10® (p = 0.0222).
CONCLUSION
Data show that BrainUp-10® produces a statistically significant improvement in apathy, ameliorating neuropsychiatric distress of patients. There were no compound-related adverse events. BrainUp-10® technology may enable patients to receive the benefits for their cognitive and behavioral problems.

Identifiants

pubmed: 33935080
pii: JAD201501
doi: 10.3233/JAD-201501
doi:

Substances chimiques

Cholinesterase Inhibitors 0

Types de publication

Journal Article Multicenter Study Randomized Controlled Trial Research Support, Non-U.S. Gov't

Langues

eng

Sous-ensembles de citation

IM

Pagination

1231-1241

Auteurs

Leonardo Guzman-Martinez (L)

Laboratory of Neuroscience and Functional Medicine, Faculty of Sciences, International Center for Biomedicine (ICC), University of Chile, Santiago, Chile.

Gonzalo A Farías (GA)

Department of Neurology, Faculty of Medicine, University of Chile, Santiago, Chile.
Center for Advanced Clinical Investigation (CICA), Faculty of Medicine, University of Chile, Santiago, Chile.

José P Tapia (JP)

Laboratory of Neuroscience and Functional Medicine, Faculty of Sciences, International Center for Biomedicine (ICC), University of Chile, Santiago, Chile.

María P Sánchez (MP)

Faculty of Chemistry and Biology, University of Santiago of Chile, Santiago, Chile.

Patricio Fuentes (P)

Department of Neurology, Faculty of Medicine, University of Chile, Santiago, Chile.
Center for Advanced Clinical Investigation (CICA), Faculty of Medicine, University of Chile, Santiago, Chile.

Sergio Gloger (S)

Biomedica Research Group, Santiago, Chile.

Ricardo B Maccioni (RB)

Laboratory of Neuroscience and Functional Medicine, Faculty of Sciences, International Center for Biomedicine (ICC), University of Chile, Santiago, Chile.
Department of Neurology, Faculty of Medicine, University of Chile, Santiago, Chile.
Center for Advanced Clinical Investigation (CICA), Faculty of Medicine, University of Chile, Santiago, Chile.

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