Signaling-Biased and Constitutively Active Dopamine D2 Receptor Variant.
D2 receptor
Dopamine
G protein
allelic variant
arrestin
biased signaling
constitutive activity
Journal
ACS chemical neuroscience
ISSN: 1948-7193
Titre abrégé: ACS Chem Neurosci
Pays: United States
ID NLM: 101525337
Informations de publication
Date de publication:
02 06 2021
02 06 2021
Historique:
pubmed:
12
5
2021
medline:
22
6
2021
entrez:
11
5
2021
Statut:
ppublish
Résumé
A dopamine D2 receptor mutation was recently identified in a family with a novel hyperkinetic movement disorder. Compared to the wild type D2 receptor, the novel allelic variant D2-I
Identifiants
pubmed: 33974399
doi: 10.1021/acschemneuro.0c00712
pmc: PMC8528033
mid: NIHMS1708496
doi:
Substances chimiques
Dopamine Agonists
0
Receptors, Dopamine D2
0
Quinpirole
20OP60125T
Cyclic AMP
E0399OZS9N
Types de publication
Journal Article
Research Support, N.I.H., Extramural
Research Support, Non-U.S. Gov't
Research Support, U.S. Gov't, Non-P.H.S.
Langues
eng
Sous-ensembles de citation
IM
Pagination
1873-1884Subventions
Organisme : NIDA NIH HHS
ID : R01 DA034388
Pays : United States
Organisme : BLRD VA
ID : I01 BX003279
Pays : United States
Organisme : NIDA NIH HHS
ID : R01 DA004523
Pays : United States
Organisme : NIDA NIH HHS
ID : F31 DA047007
Pays : United States
Organisme : NINDS NIH HHS
ID : R21 NS117713
Pays : United States
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